GB1475795A - Steroid 21-thioesters - Google Patents

Steroid 21-thioesters

Info

Publication number
GB1475795A
GB1475795A GB2399274A GB2399274A GB1475795A GB 1475795 A GB1475795 A GB 1475795A GB 2399274 A GB2399274 A GB 2399274A GB 2399274 A GB2399274 A GB 2399274A GB 1475795 A GB1475795 A GB 1475795A
Authority
GB
United Kingdom
Prior art keywords
thioesters
steroid
mercaptopregna
jouveinal
trimethylacetate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB2399274A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Jouveinal SA
Original Assignee
Jouveinal SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Jouveinal SA filed Critical Jouveinal SA
Publication of GB1475795A publication Critical patent/GB1475795A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
GB2399274A 1973-05-30 1974-05-30 Steroid 21-thioesters Expired GB1475795A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7319734A FR2231374B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1973-05-30 1973-05-30

Publications (1)

Publication Number Publication Date
GB1475795A true GB1475795A (en) 1977-06-10

Family

ID=9120281

Family Applications (1)

Application Number Title Priority Date Filing Date
GB2399274A Expired GB1475795A (en) 1973-05-30 1974-05-30 Steroid 21-thioesters

Country Status (7)

Country Link
US (1) US4014909A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
JP (1) JPS5136273B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BE (1) BE815590A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (1) CA1041083A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FR (1) FR2231374B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GB (1) GB1475795A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NL (1) NL163221C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4861765A (en) * 1985-06-26 1989-08-29 Jouveinal 21-alkyl-, cycloalkyl- or aryl-substituted thio steroids and pharmaceutical compositions containing them
US5420120A (en) * 1993-12-17 1995-05-30 Alcon Laboratories, Inc. Anti-inflammatory glucocorticoid compounds for topical ophthalmic use
GB2311290A (en) * 1996-03-20 1997-09-24 Losbanos Ltd Manufacture of steroids

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6144070Y2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * 1978-05-15 1986-12-12
FR2442856A1 (fr) * 1978-12-01 1980-06-27 Sipsy Procede de preparation de steroides
US4262940A (en) * 1978-12-15 1981-04-21 The Johnson Corporation Internally compensated self-aligning rotary joint
FR2510582B1 (fr) 1981-07-30 1986-05-30 Sipsy Steroides esterifies en la position 17 et thio-esterifies en la position 21, leur procede de preparation et leur application comme medicament
FR2529894B2 (fr) * 1981-07-30 1986-07-25 Jouveinal Steroides esterifies en la position 17 et thio-esterifies en la position 21 et leur application comme medicament
FR2551069B1 (fr) * 1983-08-26 1986-07-25 Jouveinal Sa 17-oxo-21-thioesters d'hydrocortisone, leur preparation et leurs applications comme medicament
JPS6175974U (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * 1984-10-24 1986-05-22
US5116829A (en) * 1990-04-23 1992-05-26 Kao Corporation Steroid compounds
US5439901A (en) * 1993-07-23 1995-08-08 The Procter & Gamble Company Cyproterone thiopivalate
US5602094A (en) * 1994-03-29 1997-02-11 Goddard; David Treatment of tumors
EP1238285A1 (en) * 1999-11-30 2002-09-11 Akzo Nobel N.V. Steroid compounds for steroid receptor binding assays
EP1663999A2 (en) * 2003-08-29 2006-06-07 Ranbaxy Laboratories, Ltd. Inhibitors of phosphodiesterase type-iv
EP1694655A2 (en) * 2003-11-26 2006-08-30 Ranbaxy Laboratories Limited Phosphodiesterase inhibitors
US20080009535A1 (en) * 2004-08-30 2008-01-10 Sarala Balachandran Inhibitors of phosphodiesterase type-IV
EP1934219A1 (en) 2005-09-16 2008-06-25 Ranbaxy Laboratories Limited Substituted pyrazolo [3,4-b] pyridines as phosphodiesterase inhibitors
CA2626612A1 (en) 2005-10-19 2007-04-26 Ranbaxy Laboratories Limited Pharmaceutical compositions of muscarinic receptor antagonists
JP2009512677A (ja) * 2005-10-19 2009-03-26 ランバクシー ラボラトリーズ リミテッド ホスホジエステラーゼタイプｉｖ阻害剤の組成物
US20100029728A1 (en) * 2006-09-22 2010-02-04 Ranbaxy Laboratories Limited Phosphodiesterase inhibitors
CN101616901A (zh) * 2006-09-22 2009-12-30 兰贝克赛实验室有限公司 Iv型磷酸二酯酶的抑制剂
EP1958947A1 (en) 2007-02-15 2008-08-20 Ranbaxy Laboratories Limited Inhibitors of phosphodiesterase type 4
WO2008111009A1 (en) * 2007-03-14 2008-09-18 Ranbaxy Laboratories Limited Pyrazolo [3, 4-b] pyridine derivatives as phosphodiesterase inhibitors
NZ579645A (en) 2007-03-14 2012-01-12 Ranbaxy Lab Ltd Pyrazolo (3, 4-b) pyridine derivatives as phosphodiesterase inhibitors
CN102099368A (zh) * 2007-12-21 2011-06-15 先灵公司 作为糖皮质激素受体激动剂的c-21硫醚
EP2111861A1 (en) 2008-04-21 2009-10-28 Ranbaxy Laboratories Limited Compositions of phosphodiesterase type IV inhibitors
EP3153502B1 (fr) * 2013-09-25 2018-12-19 H4 Pharma Procédé de synthèse d'un sel minéral de l'acide pivalique en tant que produit intermédiaire

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2814632A (en) * 1957-02-21 1957-11-26 Schering Corp Steroid compounds and methods for their manufacture
FR1187M (fr) * 1961-03-17 1962-03-19 Roussel Uclaf Nouveau médicament notamment pour le traitement des manifestations inflammatoires d'origine rhumatismale arthritique ou infectieuse.
DE2044831A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * 1969-09-18 1971-03-25
CH566349A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * 1969-12-24 1975-09-15 Ciba Geigy Ag
US3803133A (en) * 1972-12-15 1974-04-09 Squibb & Sons Inc 21-sulfinyl steroids

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4861765A (en) * 1985-06-26 1989-08-29 Jouveinal 21-alkyl-, cycloalkyl- or aryl-substituted thio steroids and pharmaceutical compositions containing them
US5420120A (en) * 1993-12-17 1995-05-30 Alcon Laboratories, Inc. Anti-inflammatory glucocorticoid compounds for topical ophthalmic use
GB2311290A (en) * 1996-03-20 1997-09-24 Losbanos Ltd Manufacture of steroids

Also Published As

Publication number Publication date
FR2231374A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1974-12-27
DE2357778B2 (de) 1977-02-17
NL7407176A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1974-12-03
US4014909A (en) 1977-03-29
DE2357778A1 (de) 1974-12-19
FR2231374B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1976-10-22
NL163221C (nl) 1980-08-15
BE815590A (fr) 1974-09-16
CA1041083A (fr) 1978-10-24
JPS5136273B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1976-10-07
NL163221B (nl) 1980-03-17
JPS5030863A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1975-03-27

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Legal Events

Date Code Title Description
PS Patent sealed [section 19, patents act 1949]
PE20 Patent expired after termination of 20 years

Effective date: 19940529