GB1385578A - 5- 3-iodopropargyloxy pyrimidines and a method of preparing same - Google Patents
5- 3-iodopropargyloxy pyrimidines and a method of preparing sameInfo
- Publication number
- GB1385578A GB1385578A GB5540172A GB5540172A GB1385578A GB 1385578 A GB1385578 A GB 1385578A GB 5540172 A GB5540172 A GB 5540172A GB 5540172 A GB5540172 A GB 5540172A GB 1385578 A GB1385578 A GB 1385578A
- Authority
- GB
- United Kingdom
- Prior art keywords
- ethylthio
- pyrimidine
- methoxy
- hydroxy
- give
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- -1 benzylthio Chemical group 0.000 abstract 3
- QGZKDVFQNNGYKY-UHFFFAOYSA-N Ammonia Chemical compound N QGZKDVFQNNGYKY-UHFFFAOYSA-N 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- NGAWZVYNUUHVJQ-UHFFFAOYSA-N 2-ethylsulfanyl-5-methoxy-1h-pyrimidin-6-one Chemical compound CCSC1=NC=C(OC)C(=O)N1 NGAWZVYNUUHVJQ-UHFFFAOYSA-N 0.000 abstract 1
- AAYHVAIEYCLGGO-UHFFFAOYSA-N 2-ethylsulfanyl-5-methoxypyrimidine Chemical compound C(C)SC1=NC=C(C=N1)OC AAYHVAIEYCLGGO-UHFFFAOYSA-N 0.000 abstract 1
- PSKTVUXBXHTWIS-UHFFFAOYSA-N 2-ethylsulfanylpyrimidin-5-ol Chemical compound CCSC1=NC=C(O)C=N1 PSKTVUXBXHTWIS-UHFFFAOYSA-N 0.000 abstract 1
- 125000001494 2-propynyl group Chemical group [H]C#CC([H])([H])* 0.000 abstract 1
- OBWADCOQFAXTJE-UHFFFAOYSA-N 4-chloro-2-ethylsulfanyl-5-methoxypyrimidine Chemical compound C(C)SC1=NC=C(C(=N1)Cl)OC OBWADCOQFAXTJE-UHFFFAOYSA-N 0.000 abstract 1
- CDFYFTSELDPCJA-UHFFFAOYSA-N 5-methoxy-2-sulfanylidene-1h-pyrimidin-4-one Chemical compound COC1=CNC(=S)NC1=O CDFYFTSELDPCJA-UHFFFAOYSA-N 0.000 abstract 1
- ZCYVEMRRCGMTRW-UHFFFAOYSA-N 7553-56-2 Chemical compound [I] ZCYVEMRRCGMTRW-UHFFFAOYSA-N 0.000 abstract 1
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 abstract 1
- 241000233866 Fungi Species 0.000 abstract 1
- HCHKCACWOHOZIP-UHFFFAOYSA-N Zinc Chemical compound [Zn] HCHKCACWOHOZIP-UHFFFAOYSA-N 0.000 abstract 1
- 150000008044 alkali metal hydroxides Chemical class 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000004644 alkyl sulfinyl group Chemical group 0.000 abstract 1
- 125000004390 alkyl sulfonyl group Chemical group 0.000 abstract 1
- 125000004414 alkyl thio group Chemical group 0.000 abstract 1
- 229910021529 ammonia Inorganic materials 0.000 abstract 1
- 230000001857 anti-mycotic effect Effects 0.000 abstract 1
- DENRZWYUOJLTMF-UHFFFAOYSA-N diethyl sulfate Chemical compound CCOS(=O)(=O)OCC DENRZWYUOJLTMF-UHFFFAOYSA-N 0.000 abstract 1
- 239000003085 diluting agent Substances 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 230000002083 iodinating effect Effects 0.000 abstract 1
- 229910052740 iodine Inorganic materials 0.000 abstract 1
- 239000011630 iodine Substances 0.000 abstract 1
- 230000001717 pathogenic effect Effects 0.000 abstract 1
- RLOWWWKZYUNIDI-UHFFFAOYSA-N phosphinic chloride Chemical compound ClP=O RLOWWWKZYUNIDI-UHFFFAOYSA-N 0.000 abstract 1
- LTXJLQINBYSQFU-UHFFFAOYSA-N pyrimidin-5-ol Chemical compound OC1=CN=CN=C1 LTXJLQINBYSQFU-UHFFFAOYSA-N 0.000 abstract 1
- 230000000699 topical effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/56—One oxygen atom and one sulfur atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/34—One oxygen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/52—Two oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CS860971A CS158984B1 (en:Method) | 1971-12-15 | 1971-12-15 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1385578A true GB1385578A (en) | 1975-02-26 |
Family
ID=5436887
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB5540172A Expired GB1385578A (en) | 1971-12-15 | 1972-11-30 | 5- 3-iodopropargyloxy pyrimidines and a method of preparing same |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US3907797A (en:Method) |
| JP (1) | JPS5426557B2 (en:Method) |
| AT (1) | AT319254B (en:Method) |
| BE (1) | BE792632A (en:Method) |
| CA (1) | CA989839A (en:Method) |
| CH (1) | CH578541A5 (en:Method) |
| CS (1) | CS158984B1 (en:Method) |
| DK (1) | DK133044C (en:Method) |
| FI (1) | FI56002C (en:Method) |
| FR (1) | FR2163727B1 (en:Method) |
| GB (1) | GB1385578A (en:Method) |
| NL (1) | NL172653C (en:Method) |
| SE (1) | SE393110B (en:Method) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2484416A1 (fr) * | 1980-06-13 | 1981-12-18 | Spofa Vereinigte Pharma Werke | Derives 4-(3-iodopropargyloxy) pyrimidine et procede pour la production de ces derives |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4170704A (en) * | 1978-04-20 | 1979-10-09 | Givaudan Corporation | Iodopropargyl pyridyl and picolinyl ethers and thioethers as paint fungicides |
| US4220577A (en) * | 1978-04-20 | 1980-09-02 | Givaudan Corporation | Iodopropargyl pyridyl and picolinyl ethers and thioethers as paint fungicides |
| US4729987A (en) * | 1978-07-28 | 1988-03-08 | The Dow Chemical Company | Insecticidal O,O-diethyl-O-(2-(1,1-dimethylethyl)-5-pyrimidinyl)-phosphorothioate |
| US4654329A (en) * | 1978-07-28 | 1987-03-31 | The Dow Chemical Company | Insecticidal, miticidal or nematocidal phosphorus esters of 5-pyrimidinols |
| US4379930A (en) * | 1981-09-14 | 1983-04-12 | The Dow Chemical Company | Preparation of 2-t-butyl-5-hydroxypyrimidine |
| CA1198261A (en) * | 1983-04-29 | 1985-12-24 | Gordon M. Cameron | Liquid sulphur dioxide manufacture |
| DE3423623A1 (de) * | 1984-06-27 | 1986-01-02 | Bayer Ag, 5090 Leverkusen | Verfahren zur herstellung von phosphorsaeurederivaten und zwischenprodukten |
| DE3423622A1 (de) * | 1984-06-27 | 1986-01-02 | Bayer Ag, 5090 Leverkusen | Verfahren zur herstellung von phosphorsaeurederivaten und zwischenprodukten |
| US6838463B2 (en) * | 2000-09-19 | 2005-01-04 | Sumitomo Chemical Company, Limited | Pyrimidine compounds and their use |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL38815A0 (en) * | 1971-03-05 | 1972-04-27 | Ciba Geigy Ag | Iodoethynyl compounds,their manufacture and their use |
-
0
- BE BE792632D patent/BE792632A/xx not_active IP Right Cessation
-
1971
- 1971-12-15 CS CS860971A patent/CS158984B1/cs unknown
-
1972
- 1972-11-17 SE SE7215006A patent/SE393110B/xx unknown
- 1972-11-20 CH CH1686472A patent/CH578541A5/xx not_active IP Right Cessation
- 1972-11-22 DK DK583172A patent/DK133044C/da not_active IP Right Cessation
- 1972-11-27 FI FI3349/72A patent/FI56002C/fi active
- 1972-11-30 GB GB5540172A patent/GB1385578A/en not_active Expired
- 1972-12-09 JP JP12306472A patent/JPS5426557B2/ja not_active Expired
- 1972-12-11 AT AT1052172A patent/AT319254B/de not_active IP Right Cessation
- 1972-12-11 NL NLAANVRAGE7216815,A patent/NL172653C/xx not_active IP Right Cessation
- 1972-12-14 US US314991A patent/US3907797A/en not_active Expired - Lifetime
- 1972-12-14 CA CA159,124A patent/CA989839A/en not_active Expired
- 1972-12-15 FR FR7244892A patent/FR2163727B1/fr not_active Expired
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2484416A1 (fr) * | 1980-06-13 | 1981-12-18 | Spofa Vereinigte Pharma Werke | Derives 4-(3-iodopropargyloxy) pyrimidine et procede pour la production de ces derives |
Also Published As
| Publication number | Publication date |
|---|---|
| DE2259784B2 (de) | 1976-02-19 |
| FR2163727A1 (en:Method) | 1973-07-27 |
| FR2163727B1 (en:Method) | 1983-07-01 |
| CH578541A5 (en:Method) | 1976-08-13 |
| FI56002B (fi) | 1979-07-31 |
| AT319254B (de) | 1974-12-10 |
| CA989839A (en) | 1976-05-25 |
| BE792632A (fr) | 1973-03-30 |
| CS158984B1 (en:Method) | 1974-12-27 |
| DK133044B (da) | 1976-03-15 |
| DK133044C (da) | 1976-08-16 |
| NL172653C (nl) | 1983-10-03 |
| SE393110B (sv) | 1977-05-02 |
| DE2259784A1 (de) | 1973-06-28 |
| JPS4864078A (en:Method) | 1973-09-05 |
| FI56002C (fi) | 1979-11-12 |
| NL7216815A (en:Method) | 1973-06-13 |
| NL172653B (nl) | 1983-05-02 |
| JPS5426557B2 (en:Method) | 1979-09-04 |
| US3907797A (en) | 1975-09-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed [section 19, patents act 1949] | ||
| PCNP | Patent ceased through non-payment of renewal fee |