GB1234060A - - Google Patents

Info

Publication number
GB1234060A
GB1234060A GB1234060DA GB1234060A GB 1234060 A GB1234060 A GB 1234060A GB 1234060D A GB1234060D A GB 1234060DA GB 1234060 A GB1234060 A GB 1234060A
Authority
GB
United Kingdom
Prior art keywords
cbo
phe
gly
ome
arg
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GB1234060A publication Critical patent/GB1234060A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1002—Tetrapeptides with the first amino acid being neutral
    • C07K5/1016—Tetrapeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06026—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atom, i.e. Gly or Ala
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06034—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms
    • C07K5/06052—Val-amino acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06086—Dipeptides with the first amino acid being basic
    • C07K5/06095—Arg-amino acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06104—Dipeptides with the first amino acid being acidic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0812—Tripeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1002—Tetrapeptides with the first amino acid being neutral
    • C07K5/1005—Tetrapeptides with the first amino acid being neutral and aliphatic
    • C07K5/1008—Tetrapeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atoms, i.e. Gly, Ala

Abstract

1,234,060. Peptides. BOFORS A.B. 23 Oct., 1968 [24 Oct., 1967], No. 50397/68. Heading C2C. Novel compound I where R 1 is H, butyl, isobutyl, sec-butyl or benzyl; m is 0 or 1; X is -(NHCH 2 CO-) n1 , n 1 is 0-3; R 3 is carboxy-, carbalkoxy- or carbamido-alkyl where the alkyl has 1-6C; Y is of Formula II p is 0 or 1; n 2 is 2, 3 or 4; R 4 is H, guanyl, or carbamyl; n is 2, 3 or 4; R 2 is alkoxy, alkenyloxy or cycloalkoxy of up to 8C; -NR 5 R 6 , -gly-pro-arg-R 7 ; R 5 and R 6 are H or alkyl, alkenyl or cycloalkyl of up to 8C and R 7 is alkoxy, alkenyloxy or cycloalkoxy of up to 8C or -NR 5 R 6 are prepared by conventional methods of peptide chemistry. Intermediates isolated are H- or CBO - valarg(NO 2 ) - OMe; CBO - gly - gly - val - arg(NO 2 )- OMe; CBO - ala - glu(OMe) - OH; CBO - gly- NHNHCOOtBu; H - gly - NHNHCOOtBu; CBO - phe - leu - OEt; CBO - phe - leu- NHNH 2 ; CBO - glu(OMe) - gly - NHNHCOOt- Bu; CBO - ala - glu(OMe) - gly - NHNHCOOt- Bu; CBO - phe - leu - ala - glu(OMe) - gly- NHNHCOOtBu; CBO - phe - arg(NO 2 )- OMe; CBO - val - arg(NO 2 ) - NH 2 ; CBO- phe - arg(NO 2 ) - NH 2 ; CBO - phe - leu - alaglu(OMe) - gly - gly - gly - val - arg(NO 2 )- OMe; CBO - phe - leu - ala - glu(OMe) - gly- N 3 ; CBO - phe - val - arg(NO 2 ) - OMe; CBO- phe - gly - val - arg(NO 2 ) - OMe; CBO - phegly - gly - val - arg(NO 2 ) - OEt; CBO - phegly - gly - gly - val - arg(NO 2 ) - OMe; CBO- phe - phe - val - arg(NO 2 )OMe; CBO - phe - leuval - arg(NO 2 ) - OMe; CBO - val - arg(NO 2 )- NH 2 ; CBO - phe - arg(NO 2 ) - NH 2 ; CBO - pheval - arg(NO 2 ) - NH 2 ; CBO - arg(NO 2 ) - arg- (NO 2 ) - OMe; CBO - phe - val - OMe; CBO- phe - val - NHNH 2 ; CBO - phe - phe - OMe; CBO - phe - phe - NHNH 2 ; CBO - phe - gly- OEt; CBO - phe - gly - gly - OEt; CBO - phegly - NHNH 2 ; and CBO - phe - gly - gly- NHNH 2 .
GB1234060D 1967-10-24 1968-10-23 Expired GB1234060A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE1455767A SE348465B (en) 1967-10-24 1967-10-24

Publications (1)

Publication Number Publication Date
GB1234060A true GB1234060A (en) 1971-06-03

Family

ID=20299296

Family Applications (1)

Application Number Title Priority Date Filing Date
GB1234060D Expired GB1234060A (en) 1967-10-24 1968-10-23

Country Status (8)

Country Link
JP (1) JPS4823070B1 (en)
CH (1) CH535206A (en)
DK (1) DK123709B (en)
FI (1) FI49153C (en)
FR (1) FR8346M (en)
GB (1) GB1234060A (en)
NO (1) NO122126B (en)
SE (1) SE348465B (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111606971A (en) * 2019-02-24 2020-09-01 长沙理工大学 Preparation method of FAGG

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6139350Y2 (en) * 1980-08-18 1986-11-11
JPS62146989U (en) * 1986-03-11 1987-09-17

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111606971A (en) * 2019-02-24 2020-09-01 长沙理工大学 Preparation method of FAGG
CN111606971B (en) * 2019-02-24 2023-05-26 长沙理工大学 Preparation method of FAPGG

Also Published As

Publication number Publication date
JPS4823070B1 (en) 1973-07-11
SE348465B (en) 1972-09-04
DE1804022B2 (en) 1976-05-06
FI49153C (en) 1975-04-10
CH535206A (en) 1973-03-31
NO122126B (en) 1971-05-24
FR8346M (en) 1970-12-21
DK123709B (en) 1972-07-24
DE1804022A1 (en) 1969-05-14

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Legal Events

Date Code Title Description
PS Patent sealed
PLE Entries relating assignments, transmissions, licences in the register of patents
PCNP Patent ceased through non-payment of renewal fee