GB0402118D0 - Polymorphic forms of a GABAA agonist - Google Patents

Polymorphic forms of a GABAA agonist

Info

Publication number
GB0402118D0
GB0402118D0 GBGB0402118.4A GB0402118A GB0402118D0 GB 0402118 D0 GB0402118 D0 GB 0402118D0 GB 0402118 A GB0402118 A GB 0402118A GB 0402118 D0 GB0402118 D0 GB 0402118D0
Authority
GB
United Kingdom
Prior art keywords
polymorphic forms
gabaa agonist
gabaa
agonist
polymorphic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
GBGB0402118.4A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Organon Pharma UK Ltd
Original Assignee
Merck Sharp and Dohme Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=31971783&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=GB0402118(D0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Merck Sharp and Dohme Ltd filed Critical Merck Sharp and Dohme Ltd
Priority to GBGB0402118.4A priority Critical patent/GB0402118D0/en
Publication of GB0402118D0 publication Critical patent/GB0402118D0/en
Priority to ARP050100210A priority patent/AR047511A1/es
Priority to TW094101857A priority patent/TWI345972B/zh
Priority to MYPI20050253A priority patent/MY139525A/en
Priority to PE2005000102A priority patent/PE20050769A1/es
Priority to PT05702040T priority patent/PT1713813E/pt
Priority to CN2005800031615A priority patent/CN1914212B/zh
Priority to PL05702040T priority patent/PL1713813T3/pl
Priority to US11/045,768 priority patent/US7262300B2/en
Priority to JP2006550301A priority patent/JP4917440B2/ja
Priority to AU2005209473A priority patent/AU2005209473B2/en
Priority to GB0501847A priority patent/GB2410434A/en
Priority to NZ548191A priority patent/NZ548191A/en
Priority to UAA200609410A priority patent/UA87487C2/ru
Priority to EA200601404A priority patent/EA009413B1/ru
Priority to MXPA06008595A priority patent/MXPA06008595A/es
Priority to BRPI0506858-4A priority patent/BRPI0506858A/pt
Priority to PCT/GB2005/000288 priority patent/WO2005073237A2/en
Priority to HR20080614T priority patent/HRP20080614T3/xx
Priority to DE602005010975T priority patent/DE602005010975D1/de
Priority to ES05702040T priority patent/ES2314613T3/es
Priority to EP08019457A priority patent/EP2042505A1/en
Priority to AT05702040T priority patent/ATE414088T1/de
Priority to SI200530521T priority patent/SI1713813T1/sl
Priority to DO2005000013A priority patent/DOP2005000013A/es
Priority to HK07102068.6A priority patent/HK1096547B/en
Priority to CA2554536A priority patent/CA2554536C/en
Priority to DK05702040T priority patent/DK1713813T3/da
Priority to EP05702040A priority patent/EP1713813B1/en
Priority to ZA200605307A priority patent/ZA200605307B/en
Priority to IL176863A priority patent/IL176863A0/en
Priority to CO06073254A priority patent/CO5700743A2/es
Priority to EC2006006735A priority patent/ECSP066735A/es
Priority to KR1020067015417A priority patent/KR101210361B1/ko
Priority to MA29278A priority patent/MA28364A1/fr
Priority to NO20063843A priority patent/NO20063843L/no
Priority to US11/827,570 priority patent/US8236958B2/en
Priority to CY20081101439T priority patent/CY1108647T1/el
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Psychology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
GBGB0402118.4A 2004-01-30 2004-01-30 Polymorphic forms of a GABAA agonist Ceased GB0402118D0 (en)

Priority Applications (38)

Application Number Priority Date Filing Date Title
GBGB0402118.4A GB0402118D0 (en) 2004-01-30 2004-01-30 Polymorphic forms of a GABAA agonist
ARP050100210A AR047511A1 (es) 2004-01-30 2005-01-20 Formas poliformicas de un agonista de gabaa
TW094101857A TWI345972B (en) 2004-01-30 2005-01-21 Polymorphic forms of a gabaa agonist
MYPI20050253A MY139525A (en) 2004-01-30 2005-01-24 Polymorphic forms of a gabaa agonist.
PE2005000102A PE20050769A1 (es) 2004-01-30 2005-01-27 Formas polimorficas de un agonista de gabaa
DK05702040T DK1713813T3 (da) 2004-01-30 2005-01-28 Polymorfe former af en gabaa agonist
EP05702040A EP1713813B1 (en) 2004-01-30 2005-01-28 Polymorphic forms of a gabaa agonist
PCT/GB2005/000288 WO2005073237A2 (en) 2004-01-30 2005-01-28 Polymorphic forms of a gabaa agonist
AT05702040T ATE414088T1 (de) 2004-01-30 2005-01-28 Polymorphe formen eines gabaa-agonisten
PL05702040T PL1713813T3 (pl) 2004-01-30 2005-01-28 Polimorficzne postacie agonisty GABAA
US11/045,768 US7262300B2 (en) 2004-01-30 2005-01-28 Polymorphic forms of a GABAA agonist
JP2006550301A JP4917440B2 (ja) 2004-01-30 2005-01-28 Ｇａｂａａアゴニストの多形性形態
AU2005209473A AU2005209473B2 (en) 2004-01-30 2005-01-28 Polymorphic forms of a GABAA agonist
GB0501847A GB2410434A (en) 2004-01-30 2005-01-28 Crystalline forms of a GABAa agonist, Gaboxadol
NZ548191A NZ548191A (en) 2004-01-30 2005-01-28 Polymorphic forms of a GABA(A) agonist for neurological or psychiatric disorders
UAA200609410A UA87487C2 (ru) 2004-01-30 2005-01-28 Полиморфные формы габоксадола, агониста gabaа, способ их получения и применение
EA200601404A EA009413B1 (ru) 2004-01-30 2005-01-28 Полиморфные формы габоксадола, агониста gaba
MXPA06008595A MXPA06008595A (es) 2004-01-30 2005-01-28 Formas polimorficas de un agonista gabaa.
BRPI0506858-4A BRPI0506858A (pt) 2004-01-30 2005-01-28 composto, métodos de preparação de monoidrato de gaboxadol cristalino e de anidrato de gaboxadol cristalino, composição farmacêutica, e, uso de um composto
PT05702040T PT1713813E (pt) 2004-01-30 2005-01-28 Formas polimórficas de um agonista de gabaa
HR20080614T HRP20080614T3 (en) 2004-01-30 2005-01-28 Polymorphic forms of a gabaa agonist
DE602005010975T DE602005010975D1 (de) 2004-01-30 2005-01-28 Polymorphe formen eines gabaa-agonisten
ES05702040T ES2314613T3 (es) 2004-01-30 2005-01-28 Formas poliformicas de un agonista gabaa.
EP08019457A EP2042505A1 (en) 2004-01-30 2005-01-28 Polymorphic forms of a GABAa agonist
CN2005800031615A CN1914212B (zh) 2004-01-30 2005-01-28 Gabaa激动剂的多晶型
SI200530521T SI1713813T1 (sl) 2004-01-30 2005-01-28 Polimorfne oblike agonista gabaa
DO2005000013A DOP2005000013A (es) 2004-01-30 2005-01-28 Formas polimórficas de 4,5,6,7-tetrahidroisoxazolo[5,4-c]piridin-3-ol
HK07102068.6A HK1096547B (en) 2004-01-30 2005-01-28 Polymorphic forms of a gabaa agonist
CA2554536A CA2554536C (en) 2004-01-30 2005-01-28 Crystalline forms of gaboxadol monohydrate or anhydrate
ZA200605307A ZA200605307B (en) 2004-01-30 2006-06-27 Polymorphic Forms of a Gabaa agonist
IL176863A IL176863A0 (en) 2004-01-30 2006-07-13 Polymorphic forms of a gaba a agonist
CO06073254A CO5700743A2 (es) 2004-01-30 2006-07-26 Formas polimorficas de un agonista de gaba a
EC2006006735A ECSP066735A (es) 2004-01-30 2006-07-28 Formas polimórficas de un agonista de gabaa
KR1020067015417A KR101210361B1 (ko) 2004-01-30 2006-07-28 다형의 ｇａｂａａ 효능제
MA29278A MA28364A1 (fr) 2004-01-30 2006-08-22 Formes polymorphes d'un agoniste gabaa
NO20063843A NO20063843L (no) 2004-01-30 2006-08-29 Polymorfe formar av en GABA-A-agonist
US11/827,570 US8236958B2 (en) 2004-01-30 2007-07-13 Polymorphic forms of a GABAA agonist
CY20081101439T CY1108647T1 (el) 2004-01-30 2008-12-10 Πολυμορφικες μορφες ενος αγωνιστη gabaa

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0402118.4A GB0402118D0 (en) 2004-01-30 2004-01-30 Polymorphic forms of a GABAA agonist

Publications (1)

Publication Number Publication Date
GB0402118D0 true GB0402118D0 (en) 2004-03-03

Family

ID=31971783

Family Applications (2)

Application Number Title Priority Date Filing Date
GBGB0402118.4A Ceased GB0402118D0 (en) 2004-01-30 2004-01-30 Polymorphic forms of a GABAA agonist
GB0501847A Withdrawn GB2410434A (en) 2004-01-30 2005-01-28 Crystalline forms of a GABAa agonist, Gaboxadol

Family Applications After (1)

Application Number Title Priority Date Filing Date
GB0501847A Withdrawn GB2410434A (en) 2004-01-30 2005-01-28 Crystalline forms of a GABAa agonist, Gaboxadol

Country Status (34)

Country Link
US (2) US7262300B2 (https=)
EP (2) EP1713813B1 (https=)
JP (1) JP4917440B2 (https=)
KR (1) KR101210361B1 (https=)
CN (1) CN1914212B (https=)
AR (1) AR047511A1 (https=)
AT (1) ATE414088T1 (https=)
AU (1) AU2005209473B2 (https=)
BR (1) BRPI0506858A (https=)
CA (1) CA2554536C (https=)
CO (1) CO5700743A2 (https=)
CY (1) CY1108647T1 (https=)
DE (1) DE602005010975D1 (https=)
DK (1) DK1713813T3 (https=)
DO (1) DOP2005000013A (https=)
EA (1) EA009413B1 (https=)
EC (1) ECSP066735A (https=)
ES (1) ES2314613T3 (https=)
GB (2) GB0402118D0 (https=)
HR (1) HRP20080614T3 (https=)
IL (1) IL176863A0 (https=)
MA (1) MA28364A1 (https=)
MX (1) MXPA06008595A (https=)
MY (1) MY139525A (https=)
NO (1) NO20063843L (https=)
NZ (1) NZ548191A (https=)
PE (1) PE20050769A1 (https=)
PL (1) PL1713813T3 (https=)
PT (1) PT1713813E (https=)
SI (1) SI1713813T1 (https=)
TW (1) TWI345972B (https=)
UA (1) UA87487C2 (https=)
WO (1) WO2005073237A2 (https=)
ZA (1) ZA200605307B (https=)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0402118D0 (en) 2004-01-30 2004-03-03 Merck Sharp & Dohme Polymorphic forms of a GABAA agonist
US20060063802A1 (en) 2004-03-29 2006-03-23 Matthieu Guitton Methods for the treatment of tinnitus induced by cochlear excitotoxicity
US8268866B2 (en) 2004-03-29 2012-09-18 Matthieu Guitton Methods for the treatment of tinnitus induced by cochlear excitotoxicity
US9072662B2 (en) 2004-03-29 2015-07-07 Auris Medical Ag Methods for the treatment of tinnitus induced by cochlear excitotoxicity
DE102005004343A1 (de) * 2005-01-25 2006-08-10 Eberhard-Karls-Universität Tübingen Universitätsklinikum Behandlung von Phantomphänomenen
WO2006083682A2 (en) * 2005-01-28 2006-08-10 H.Lundbeck A/S Polymorphic forms of a gabaa agonist
ES2524994T3 (es) 2005-09-28 2014-12-16 Auris Medical Ag Composiciones farmacéuticas para el tratamiento de trastornos del oído interno.
CN102093387B (zh) * 2009-12-10 2012-07-25 天津泰普医药知识产权流转储备中心有限公司 4,5,6,7-四氢异噁唑并[5,4-c]吡啶-3-醇一水合物的晶型化合物
EP2790686B1 (en) 2011-12-12 2021-03-10 Zilentin Ag Treatment of tinnitus through modulation of chloride co-transporter nkcc1 in the auditory system
IL256912B2 (en) 2015-07-17 2024-01-01 Ovid Therapeutics Inc Methods of treating developmental disorders with gaboxadol
EP4233861A3 (en) 2016-08-11 2023-10-11 Ovid Therapeutics, Inc. Compositions for treatment of essential tremor
EP3528807A4 (en) * 2016-11-22 2020-06-17 Ovid Therapeutics Inc METHOD FOR TREATING DEVELOPMENT DISORDERS AND / OR FALLS WITH FLUPIRTIN
US10071083B2 (en) * 2017-02-03 2018-09-11 Ovid Therapeutics Inc Use of gaboxadol in the treatment of tinnitus
JP2020529440A (ja) 2017-08-04 2020-10-08 オービッド・セラピューティクス・インコーポレイテッドＯｖｉｄ Ｔｈｅｒａｐｅｕｔｉｃｓ Ｉｎｃ． 糖尿病および関連する状態の処置におけるガボキサドールの使用
MX2021003302A (es) 2018-09-20 2021-05-13 Ovid Therapeutics Inc Uso de gaboxadol para el tratamiento del sindrome de tourette, los tics y la tartamudez.
US11123332B2 (en) 2018-11-21 2021-09-21 Certego Therapeutics Inc. Gaboxadol for reducing risk of suicide and rapid relief of depression
EP3880201A4 (en) 2018-12-17 2022-07-27 Ovid Therapeutics Inc. USE OF GABOXADOL IN THE TREATMENT OF NON-24 HOUR SLEEP waking disorder
EP4051272A4 (en) 2019-12-18 2023-01-04 Ovid Therapeutics Inc. GABOXADOL FOR THE THERAPEUTIC TREATMENT OF 1P36 DELETION SYNDROME
MX2022014599A (es) 2020-05-20 2022-12-16 Certego Therapeutics Inc Gaboxadol deuterado en anillo y su uso para el tratamiento de trastornos psiquiatricos.

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DK270278A (da) 1977-06-20 1978-12-21 Krogsgaard Larsen P Cycliske aminosyrer
US4315934A (en) 1979-09-24 1982-02-16 Sandoz Ltd. Organic compounds
US4362731A (en) 1980-09-01 1982-12-07 Sandoz Ltd. Myotonolytic use of 4,5,6,7-tetrahydroisoxazolo [5,4-c] pyridin-3-ol and derivatives thereof
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DE19525598C2 (de) 1995-07-13 1997-09-25 Max Planck Gesellschaft Schlafmittel
UA52661C2 (uk) * 1996-06-14 2003-01-15 Ново Нордіск А/С Безводна кристалічна форма гідрохлориду r(-)-n-(4,4-ди(3-метилтієн-2-іл)бут-3-еніл) ніпекотинової кислоти
EP1220658A1 (en) 1999-09-28 2002-07-10 H. Lundbeck A/S Melt granulated composition and modified release dosage form prepared from said composition
AR031473A1 (es) 2000-11-20 2003-09-24 Lundbeck & Co As H Intensificadores de gaba en el tratamiento de enfermedades relacionadas con una reducida actividad neuroesteroide
CA2447417C (en) 2001-05-18 2011-10-04 Lonza Ag Method for the production of solid formulations of sodium 3-hydroxy-3-methylbutyrate
CN1511026A (zh) 2001-05-21 2004-07-07 H��¡�±������޹�˾ 加波沙朵颗粒制剂
CN100491366C (zh) * 2002-09-03 2009-05-27 华晶基因技术有限公司 汉黄芩素用作治疗焦虑症的药物的用途
US20050234093A1 (en) * 2003-06-25 2005-10-20 H. Lundbeck A/S Treatment of depression and other affective disorders
DK1641456T3 (da) * 2003-06-25 2010-06-21 Lundbeck & Co As H Gaboxadol til behandling af depression og andre affektive lidelser
AR045540A1 (es) 2003-09-05 2005-11-02 Lundbeck & Co As H Metodo de elaboracion de 4,5,6,7 tetrahidroisoxazol [5,4-c] piridin-3-ol (thip)
US20070032553A1 (en) 2003-09-10 2007-02-08 Mckernan Ruth Use of gabaa receptor agonists for the treatment of hearing, vestibular and attention disorders, intention tremor and restless leg syndrome
TW200528098A (en) 2003-12-18 2005-09-01 Lundbeck & Co As H Treatment of insomnia in human patients
GB0402118D0 (en) 2004-01-30 2004-03-03 Merck Sharp & Dohme Polymorphic forms of a GABAA agonist
JP2008504306A (ja) 2004-06-29 2008-02-14 ハー・ルンドベック・アクチエゼルスカベット 神経因性疼痛、線維筋痛症または慢性関節リウマチの治療
GB0417558D0 (en) 2004-08-06 2004-09-08 Merck Sharp & Dohme Novel combination therapy
WO2006083682A2 (en) 2005-01-28 2006-08-10 H.Lundbeck A/S Polymorphic forms of a gabaa agonist
WO2006102093A1 (en) 2005-03-18 2006-09-28 Transform Pharmaceuticals, Inc. Gaboxadol forms, compositions thereof, and related methods
US20080262029A1 (en) 2005-04-29 2008-10-23 H. Lundbeck A/S Acid and Base Salt Forms of Gaboxadol

Also Published As

Publication number Publication date
CO5700743A2 (es) 2006-11-30
HK1096547A1 (en) 2007-06-01
CA2554536A1 (en) 2005-08-11
AR047511A1 (es) 2006-01-25
EP2042505A1 (en) 2009-04-01
BRPI0506858A (pt) 2007-05-29
NZ548191A (en) 2010-04-30
WO2005073237A2 (en) 2005-08-11
US8236958B2 (en) 2012-08-07
PE20050769A1 (es) 2005-10-04
ECSP066735A (es) 2006-10-31
EP1713813B1 (en) 2008-11-12
TWI345972B (en) 2011-08-01
US20070259912A1 (en) 2007-11-08
DK1713813T3 (da) 2009-02-16
DOP2005000013A (es) 2005-08-15
WO2005073237A3 (en) 2005-10-20
EP1713813A2 (en) 2006-10-25
KR101210361B1 (ko) 2012-12-10
ES2314613T3 (es) 2009-03-16
GB2410434A (en) 2005-08-03
MY139525A (en) 2009-10-30
CN1914212A (zh) 2007-02-14
TW200534856A (en) 2005-11-01
GB0501847D0 (en) 2005-03-09
NO20063843L (no) 2006-08-29
EA200601404A1 (ru) 2006-12-29
PT1713813E (pt) 2008-12-26
AU2005209473A1 (en) 2005-08-11
ZA200605307B (en) 2007-11-28
JP4917440B2 (ja) 2012-04-18
SI1713813T1 (sl) 2009-02-28
CN1914212B (zh) 2010-10-06
US20050171142A1 (en) 2005-08-04
PL1713813T3 (pl) 2009-04-30
CY1108647T1 (el) 2014-04-09
HRP20080614T3 (en) 2009-01-31
KR20070007070A (ko) 2007-01-12
MXPA06008595A (es) 2006-08-28
ATE414088T1 (de) 2008-11-15
MA28364A1 (fr) 2006-12-01
CA2554536C (en) 2012-09-18
UA87487C2 (ru) 2009-07-27
EA009413B1 (ru) 2007-12-28
JP2007519697A (ja) 2007-07-19
DE602005010975D1 (de) 2008-12-24
IL176863A0 (en) 2006-10-31
AU2005209473B2 (en) 2010-03-04
US7262300B2 (en) 2007-08-28

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