FR2959510B1 - Derives de pyrido[3,2-d]pyrimidine, leurs procedes de preparation et leurs utilisations therapeutiques - Google Patents
Derives de pyrido[3,2-d]pyrimidine, leurs procedes de preparation et leurs utilisations therapeutiquesInfo
- Publication number
- FR2959510B1 FR2959510B1 FR1053277A FR1053277A FR2959510B1 FR 2959510 B1 FR2959510 B1 FR 2959510B1 FR 1053277 A FR1053277 A FR 1053277A FR 1053277 A FR1053277 A FR 1053277A FR 2959510 B1 FR2959510 B1 FR 2959510B1
- Authority
- FR
- France
- Prior art keywords
- pyrido
- processes
- preparation
- therapeutic uses
- pyrimidine derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR1053277A FR2959510B1 (fr) | 2010-04-28 | 2010-04-28 | Derives de pyrido[3,2-d]pyrimidine, leurs procedes de preparation et leurs utilisations therapeutiques |
PCT/FR2011/050959 WO2011135259A1 (fr) | 2010-04-28 | 2011-04-28 | Dérivés de pyrido[3,2-d]pyrimidine, leurs procédés de préparation et leurs utilisations thérapeutiques |
US13/695,001 US20130109693A1 (en) | 2010-04-28 | 2011-04-28 | Derivatives of pyrido [3,2-d] pyrimidine, methods for preparation thereof and therapeutic uses thereof |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR1053277A FR2959510B1 (fr) | 2010-04-28 | 2010-04-28 | Derives de pyrido[3,2-d]pyrimidine, leurs procedes de preparation et leurs utilisations therapeutiques |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2959510A1 FR2959510A1 (fr) | 2011-11-04 |
FR2959510B1 true FR2959510B1 (fr) | 2013-04-26 |
Family
ID=42745002
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR1053277A Expired - Fee Related FR2959510B1 (fr) | 2010-04-28 | 2010-04-28 | Derives de pyrido[3,2-d]pyrimidine, leurs procedes de preparation et leurs utilisations therapeutiques |
Country Status (3)
Country | Link |
---|---|
US (1) | US20130109693A1 (fr) |
FR (1) | FR2959510B1 (fr) |
WO (1) | WO2011135259A1 (fr) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US10235668B1 (en) | 2012-04-25 | 2019-03-19 | Wells Fargo Bank, N.A. | System and method for a mobile wallet |
US10192217B1 (en) * | 2012-04-25 | 2019-01-29 | Wells Fargo Bank, N.A. | System and method for receipt tracking in a mobile wallet |
FR2994572B1 (fr) * | 2012-08-17 | 2015-04-17 | Centre Nat Rech Scient | Pyrido[3,2-d]pyrimidines trisubstituees, leurs procedes de preparation et leurs utilisation en therapeutique |
SG11201601138PA (en) * | 2013-08-23 | 2016-03-30 | Neupharma Inc | Certain chemical entities, compositions, and methods |
AU2016220219B2 (en) | 2015-02-17 | 2020-05-14 | Neupharma, Inc. | Certain chemical entities, compositions, and methods |
CN107108615B (zh) | 2015-03-04 | 2020-11-20 | 吉利德科学公司 | Toll样受体调节性4,6-二氨基-吡啶并[3,2-D]嘧啶化合物 |
JP7101165B2 (ja) | 2016-08-15 | 2022-07-14 | ニューファーマ, インコーポレイテッド | 特定の化学的実体、組成物、および方法 |
US10640499B2 (en) | 2016-09-02 | 2020-05-05 | Gilead Sciences, Inc. | Toll like receptor modulator compounds |
EP3507276B1 (fr) | 2016-09-02 | 2021-11-03 | Gilead Sciences, Inc. | Composés modulateurs du recepteur de type toll |
GB201700814D0 (en) * | 2017-01-17 | 2017-03-01 | Liverpool School Tropical Medicine | Compounds |
FR3066761B1 (fr) * | 2017-05-23 | 2020-10-30 | Centre Nat Rech Scient | Nouveaux composes inhibiteurs des canaux ioniques |
CN111094289B (zh) * | 2018-07-03 | 2022-11-22 | 江苏恒瑞医药股份有限公司 | 吡啶并嘧啶类衍生物、其制备方法及其在医药上的应用 |
TW202210480A (zh) | 2019-04-17 | 2022-03-16 | 美商基利科學股份有限公司 | 類鐸受體調節劑之固體形式 |
TW202212339A (zh) | 2019-04-17 | 2022-04-01 | 美商基利科學股份有限公司 | 類鐸受體調節劑之固體形式 |
TW202115056A (zh) | 2019-06-28 | 2021-04-16 | 美商基利科學股份有限公司 | 類鐸受體調節劑化合物的製備方法 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2008543888A (ja) * | 2005-06-24 | 2008-12-04 | ギリアード サイエンシーズ, インコーポレイテッド | ピリド(3,2−d)ピリミジン、およびC型肝炎を治療するのに有用な医薬組成物 |
WO2008024977A2 (fr) * | 2006-08-24 | 2008-02-28 | Serenex, Inc. | Dérivés d'isoquinoline, quinazoline et phtalazine |
-
2010
- 2010-04-28 FR FR1053277A patent/FR2959510B1/fr not_active Expired - Fee Related
-
2011
- 2011-04-28 US US13/695,001 patent/US20130109693A1/en not_active Abandoned
- 2011-04-28 WO PCT/FR2011/050959 patent/WO2011135259A1/fr active Application Filing
Also Published As
Publication number | Publication date |
---|---|
WO2011135259A1 (fr) | 2011-11-03 |
US20130109693A1 (en) | 2013-05-02 |
FR2959510A1 (fr) | 2011-11-04 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |
Effective date: 20151231 |