FR2775441B1 - Matrice pour la preparation de microparticules ou de nanoparticules, procede de fabrication de telles particules et particules obtenues - Google Patents

Matrice pour la preparation de microparticules ou de nanoparticules, procede de fabrication de telles particules et particules obtenues

Info

Publication number
FR2775441B1
FR2775441B1 FR9802578A FR9802578A FR2775441B1 FR 2775441 B1 FR2775441 B1 FR 2775441B1 FR 9802578 A FR9802578 A FR 9802578A FR 9802578 A FR9802578 A FR 9802578A FR 2775441 B1 FR2775441 B1 FR 2775441B1
Authority
FR
France
Prior art keywords
particles
microparticles
nanoparticles
matrix
producing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR9802578A
Other languages
English (en)
Other versions
FR2775441A1 (fr
Inventor
Philippe Grisoni
Marc Pauly
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BASF Health and Care Products France SAS
Original Assignee
Laboratoires Serobiologiques SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Laboratoires Serobiologiques SA filed Critical Laboratoires Serobiologiques SA
Priority to FR9802578A priority Critical patent/FR2775441B1/fr
Priority to JP2000533215A priority patent/JP2002504425A/ja
Priority to EP99904918A priority patent/EP1060011A1/fr
Priority to PCT/FR1999/000385 priority patent/WO1999043426A1/fr
Priority to AU25256/99A priority patent/AU2525699A/en
Publication of FR2775441A1 publication Critical patent/FR2775441A1/fr
Application granted granted Critical
Publication of FR2775441B1 publication Critical patent/FR2775441B1/fr
Priority to US10/388,658 priority patent/US20030180235A1/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/51Nanocapsules; Nanoparticles
    • A61K9/5107Excipients; Inactive ingredients
    • A61K9/5123Organic compounds, e.g. fats, sugars
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/02Cosmetics or similar toiletry preparations characterised by special physical form
    • A61K8/11Encapsulated compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/34Alcohols
    • A61K8/342Alcohols having more than seven atoms in an unbroken chain
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/37Esters of carboxylic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/37Esters of carboxylic acids
    • A61K8/375Esters of carboxylic acids the alcohol moiety containing more than one hydroxy group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/60Sugars; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/64Proteins; Peptides; Derivatives or degradation products thereof
    • A61K8/645Proteins of vegetable origin; Derivatives or degradation products thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/67Vitamins
    • A61K8/678Tocopherol, i.e. vitamin E
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/92Oils, fats or waxes; Derivatives thereof, e.g. hydrogenation products thereof
    • A61K8/922Oils, fats or waxes; Derivatives thereof, e.g. hydrogenation products thereof of vegetable origin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q17/00Barrier preparations; Preparations brought into direct contact with the skin for affording protection against external influences, e.g. sunlight, X-rays or other harmful rays, corrosive materials, bacteria or insect stings
    • A61Q17/04Topical preparations for affording protection against sunlight or other radiation; Topical sun tanning preparations
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00Preparations for care of the skin
    • A61Q19/06Preparations for care of the skin for countering cellulitis
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B01PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01JCHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2/00Processes or devices for granulating materials, e.g. fertilisers in general; Rendering particulate materials free flowing in general, e.g. making them hydrophobic
    • B01J2/02Processes or devices for granulating materials, e.g. fertilisers in general; Rendering particulate materials free flowing in general, e.g. making them hydrophobic by dividing the liquid material into drops, e.g. by spraying, and solidifying the drops
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B82NANOTECHNOLOGY
    • B82YSPECIFIC USES OR APPLICATIONS OF NANOSTRUCTURES; MEASUREMENT OR ANALYSIS OF NANOSTRUCTURES; MANUFACTURE OR TREATMENT OF NANOSTRUCTURES
    • B82Y5/00Nanobiotechnology or nanomedicine, e.g. protein engineering or drug delivery
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2800/00Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
    • A61K2800/20Chemical, physico-chemical or functional or structural properties of the composition as a whole
    • A61K2800/28Rubbing or scrubbing compositions; Peeling or abrasive compositions; Containing exfoliants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2800/00Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
    • A61K2800/40Chemical, physico-chemical or functional or structural properties of particular ingredients
    • A61K2800/41Particular ingredients further characterized by their size
    • A61K2800/413Nanosized, i.e. having sizes below 100 nm
FR9802578A 1998-02-27 1998-02-27 Matrice pour la preparation de microparticules ou de nanoparticules, procede de fabrication de telles particules et particules obtenues Expired - Fee Related FR2775441B1 (fr)

Priority Applications (6)

Application Number Priority Date Filing Date Title
FR9802578A FR2775441B1 (fr) 1998-02-27 1998-02-27 Matrice pour la preparation de microparticules ou de nanoparticules, procede de fabrication de telles particules et particules obtenues
JP2000533215A JP2002504425A (ja) 1998-02-27 1999-02-19 ミクロ粒子又はナノ粒子製造用マトリックス、前記粒子の製造方法及び得られる粒子
EP99904918A EP1060011A1 (fr) 1998-02-27 1999-02-19 Matrice pour la preparation de microparticules ou de nanoparticules, procede de fabrication de telles particules et particules obtenues
PCT/FR1999/000385 WO1999043426A1 (fr) 1998-02-27 1999-02-19 Matrice pour la preparation de microparticules ou de nanoparticules, procede de fabrication de telles particules et particules obtenues
AU25256/99A AU2525699A (en) 1998-02-27 1999-02-19 Matrix for preparing microparticles or nanoparticles, method for making said particles and resulting particles
US10/388,658 US20030180235A1 (en) 1998-02-27 2003-03-17 Matrix for preparing microparticles or nanoparticles, method for making said particles and resulting particles

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9802578A FR2775441B1 (fr) 1998-02-27 1998-02-27 Matrice pour la preparation de microparticules ou de nanoparticules, procede de fabrication de telles particules et particules obtenues

Publications (2)

Publication Number Publication Date
FR2775441A1 FR2775441A1 (fr) 1999-09-03
FR2775441B1 true FR2775441B1 (fr) 2000-04-28

Family

ID=9523602

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9802578A Expired - Fee Related FR2775441B1 (fr) 1998-02-27 1998-02-27 Matrice pour la preparation de microparticules ou de nanoparticules, procede de fabrication de telles particules et particules obtenues

Country Status (5)

Country Link
EP (1) EP1060011A1 (fr)
JP (1) JP2002504425A (fr)
AU (1) AU2525699A (fr)
FR (1) FR2775441B1 (fr)
WO (1) WO1999043426A1 (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2000067728A2 (fr) * 1999-05-07 2000-11-16 Pharmasol Gmbh Particules lipidiques a base de melanges de lipides liquides et solides et procede pour les produire
FR2809011B1 (fr) * 2000-05-22 2002-11-15 Sederma Sa Utilisation du beurre de karite incorpore dans les microcapsules fixees sur tout textile pour augmenter l'hydratation cutanee
FR2814380B1 (fr) 2000-09-25 2002-11-08 Serobiologiques Lab Sa Poudre de microcapsules et procede d'obtention
JP2006514047A (ja) * 2002-12-19 2006-04-27 アクセス ビジネス グループ インターナショナル リミテッド ライアビリティ カンパニー 水溶性ビタミンeによる皮膚細胞再生の促進
AU2003239845A1 (en) * 2003-05-07 2004-11-26 Ifac Gmbh And Co.Kg Compositions for the targetted release of fragrances and aromas
US20070077286A1 (en) * 2003-12-24 2007-04-05 Tsutomu Ishihara Drug-containing nanoparticle, process for producing the same and parenterally administered preparation from the nanoparticle
JP4851067B2 (ja) * 2004-01-28 2012-01-11 ホソカワミクロン株式会社 ナノ粒子含有組成物およびその製造方法
KR101197489B1 (ko) * 2005-09-05 2012-11-09 가부시키가이샤 시세이도 셀프태닝 화장료
EP1967173A1 (fr) * 2007-03-06 2008-09-10 Peter Greven Hautschutz GmbH & Co. KG Produit de nettoyage de la peau avec des particules comprenant de l'huile de ricin hydrogenée
FR2918296B1 (fr) 2007-07-05 2009-09-18 Oreal Capsules de type noyau/ecorce et procede de preparation
US8613956B2 (en) 2008-06-23 2013-12-24 International Flora Technologies, Ltd. Cosmetic particles that transform from hard to soft particles comprising hydrogenated long-chain triglyceride oils
JP5406962B2 (ja) * 2012-06-14 2014-02-05 花王株式会社 ナノ粒子の製造方法
FR3000084B1 (fr) * 2012-12-20 2015-02-27 Coatex Sas Microparticules d'agent actif
EP2982363A1 (fr) * 2014-08-04 2016-02-10 Omya International AG Système à deux composants pour formulations cosmétiques
JP2021518355A (ja) * 2018-03-15 2021-08-02 セレシン・インコーポレーテッド 高い薬物充填量の中鎖脂肪酸トリグリセリドを有する医薬組成物およびそれに関連する方法
WO2020100409A1 (fr) * 2018-11-16 2020-05-22 株式会社マンダム Composition nettoyante pour la peau

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0143608B1 (fr) * 1983-11-25 1992-07-22 Ciba Specialty Chemicals Water Treatments Limited Production et utilisation de billes polymères

Also Published As

Publication number Publication date
EP1060011A1 (fr) 2000-12-20
JP2002504425A (ja) 2002-02-12
AU2525699A (en) 1999-09-15
WO1999043426A1 (fr) 1999-09-02
FR2775441A1 (fr) 1999-09-03

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Legal Events

Date Code Title Description
TP Transmission of property
ST Notification of lapse

Effective date: 20151030