FR2662691A1 - Derive de la dichloroaniline. - Google Patents

Derive de la dichloroaniline. Download PDF

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Publication number
FR2662691A1
FR2662691A1 FR9106741A FR9106741A FR2662691A1 FR 2662691 A1 FR2662691 A1 FR 2662691A1 FR 9106741 A FR9106741 A FR 9106741A FR 9106741 A FR9106741 A FR 9106741A FR 2662691 A1 FR2662691 A1 FR 2662691A1
Authority
FR
France
Prior art keywords
compound
formula
solution
amino
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR9106741A
Other languages
English (en)
French (fr)
Other versions
FR2662691B1 (US07122547-20061017-C00273.png
Inventor
Judkins Brian David
Evans Brian
Meadows James David
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Group Ltd
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB909012465A external-priority patent/GB9012465D0/en
Priority claimed from GB919104645A external-priority patent/GB9104645D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of FR2662691A1 publication Critical patent/FR2662691A1/fr
Application granted granted Critical
Publication of FR2662691B1 publication Critical patent/FR2662691B1/fr
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/28Radicals substituted by singly-bound oxygen or sulphur atoms
    • C07D213/30Oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FR9106741A 1990-06-05 1991-06-04 Derive de la dichloroaniline. Granted FR2662691A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB909012465A GB9012465D0 (en) 1990-06-05 1990-06-05 Chemical compounds
GB919104645A GB9104645D0 (en) 1991-03-05 1991-03-05 Chemical compound

Publications (2)

Publication Number Publication Date
FR2662691A1 true FR2662691A1 (fr) 1991-12-06
FR2662691B1 FR2662691B1 (US07122547-20061017-C00273.png) 1994-04-22

Family

ID=26297165

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9106741A Granted FR2662691A1 (fr) 1990-06-05 1991-06-04 Derive de la dichloroaniline.

Country Status (25)

Country Link
EP (1) EP0460924A1 (US07122547-20061017-C00273.png)
JP (1) JPH05117236A (US07122547-20061017-C00273.png)
KR (1) KR920000717A (US07122547-20061017-C00273.png)
AP (1) AP251A (US07122547-20061017-C00273.png)
AT (1) AT399874B (US07122547-20061017-C00273.png)
AU (1) AU635424B2 (US07122547-20061017-C00273.png)
BE (1) BE1005612A5 (US07122547-20061017-C00273.png)
CA (1) CA2043850A1 (US07122547-20061017-C00273.png)
CH (1) CH682322A5 (US07122547-20061017-C00273.png)
DE (1) DE4118293A1 (US07122547-20061017-C00273.png)
DK (1) DK106991A (US07122547-20061017-C00273.png)
ES (1) ES2036920B1 (US07122547-20061017-C00273.png)
FI (1) FI912679A (US07122547-20061017-C00273.png)
FR (1) FR2662691A1 (US07122547-20061017-C00273.png)
GB (1) GB2244709B (US07122547-20061017-C00273.png)
GR (1) GR1001309B (US07122547-20061017-C00273.png)
IE (1) IE911898A1 (US07122547-20061017-C00273.png)
IL (1) IL98363A0 (US07122547-20061017-C00273.png)
IT (1) IT1245868B (US07122547-20061017-C00273.png)
LU (1) LU87945A1 (US07122547-20061017-C00273.png)
MY (1) MY106672A (US07122547-20061017-C00273.png)
NL (1) NL9100960A (US07122547-20061017-C00273.png)
OA (1) OA09501A (US07122547-20061017-C00273.png)
PT (1) PT97858A (US07122547-20061017-C00273.png)
SE (1) SE500706C2 (US07122547-20061017-C00273.png)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9104650D0 (en) * 1991-03-05 1991-04-17 Glaxo Group Ltd Medicaments
ZA994264B (en) 1998-07-01 2000-01-25 Warner Lambert Co Stereoisomers with high affinity for adrenergic receptors.
US7232837B2 (en) 1999-06-29 2007-06-19 Mcneil-Ppc, Inc. Stereoisomers with high affinity for adrenergic receptors
GB0014546D0 (en) 2000-06-14 2000-08-09 Glaxo Group Ltd A novel process
FR2960153B1 (fr) * 2010-05-20 2012-08-17 Centre Nat Rech Scient Nouveaux bras autoreactifs et prodrogues les comprenant

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2165542A (en) * 1984-10-17 1986-04-16 Glaxo Group Ltd Dichloroaniline derivatives
GB2187734A (en) * 1986-02-12 1987-09-16 Glaxo Group Ltd Dichloroaniline derivatives

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1618005A1 (de) * 1966-09-22 1971-09-09 Thomae Gmbh Dr K Verfahren zur Herstellung von neuen Amino-dihalogen-phenyl-aethylaminen
EP0021636B1 (en) * 1979-06-16 1982-12-01 Beecham Group Plc Secondary amines, their preparation and use in pharmaceutical compositions
ES8802416A1 (es) * 1986-04-15 1988-06-01 Glaxo Group Ltd Un procedimiento para la preparacion de derivados de dicloroanilina.

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2165542A (en) * 1984-10-17 1986-04-16 Glaxo Group Ltd Dichloroaniline derivatives
GB2187734A (en) * 1986-02-12 1987-09-16 Glaxo Group Ltd Dichloroaniline derivatives

Also Published As

Publication number Publication date
IE911898A1 (en) 1991-12-18
GR910100242A (en) 1992-08-25
EP0460924A1 (en) 1991-12-11
GB9111946D0 (en) 1991-07-24
LU87945A1 (fr) 1993-01-15
AP9100271A0 (en) 1991-07-31
AT399874B (de) 1995-08-25
IL98363A0 (en) 1992-07-15
ES2036920B1 (es) 1994-02-16
JPH05117236A (ja) 1993-05-14
FI912679A (fi) 1991-12-06
ES2036920A1 (es) 1993-06-01
OA09501A (en) 1992-11-15
ITRM910387A1 (it) 1992-12-04
FI912679A0 (fi) 1991-06-04
NL9100960A (nl) 1992-01-02
KR920000717A (ko) 1992-01-29
BE1005612A5 (fr) 1993-11-23
GB2244709B (en) 1994-02-09
DK106991D0 (da) 1991-06-04
SE9101687L (sv) 1991-12-06
AU7812791A (en) 1991-12-12
SE9101687D0 (sv) 1991-06-04
DE4118293A1 (de) 1991-12-12
IT1245868B (it) 1994-10-25
FR2662691B1 (US07122547-20061017-C00273.png) 1994-04-22
ATA112891A (de) 1994-12-15
SE500706C2 (sv) 1994-08-15
GB2244709A (en) 1991-12-11
MY106672A (en) 1995-07-31
AP251A (en) 1993-04-20
GR1001309B (el) 1993-08-31
CA2043850A1 (en) 1991-12-06
AU635424B2 (en) 1993-03-18
DK106991A (da) 1991-12-06
PT97858A (pt) 1992-03-31
ITRM910387A0 (it) 1991-06-04
CH682322A5 (US07122547-20061017-C00273.png) 1993-08-31

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