FR2429221A1 - Procede de preparation de 3-carbamoyloxymethylcephalosporines - Google Patents
Procede de preparation de 3-carbamoyloxymethylcephalosporinesInfo
- Publication number
- FR2429221A1 FR2429221A1 FR7908746A FR7908746A FR2429221A1 FR 2429221 A1 FR2429221 A1 FR 2429221A1 FR 7908746 A FR7908746 A FR 7908746A FR 7908746 A FR7908746 A FR 7908746A FR 2429221 A1 FR2429221 A1 FR 2429221A1
- Authority
- FR
- France
- Prior art keywords
- prodn
- isocyanate
- ceph
- phosphinyl
- carbamoyloxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 239000003242 anti bacterial agent Substances 0.000 title abstract 3
- 229940088710 antibiotic agent Drugs 0.000 title abstract 3
- 229940124587 cephalosporin Drugs 0.000 title abstract 2
- 239000000543 intermediate Substances 0.000 title abstract 2
- 229930186147 Cephalosporin Natural products 0.000 title 1
- -1 methyl cephalosporin Chemical class 0.000 title 1
- FZEVMBJWXHDLDB-ZCFIWIBFSA-N (6r)-5-thia-1-azabicyclo[4.2.0]oct-2-en-8-one Chemical group S1CC=CN2C(=O)C[C@H]21 FZEVMBJWXHDLDB-ZCFIWIBFSA-N 0.000 abstract 2
- 238000006243 chemical reaction Methods 0.000 abstract 2
- SXBDXXFTJVHSAF-ZCFIWIBFSA-N (6r)-5-thia-1-azabicyclo[4.2.0]oct-3-en-8-one Chemical group S1C=CCN2C(=O)C[C@H]21 SXBDXXFTJVHSAF-ZCFIWIBFSA-N 0.000 abstract 1
- 241000894006 Bacteria Species 0.000 abstract 1
- 241001465754 Metazoa Species 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000004414 alkyl thio group Chemical group 0.000 abstract 1
- 230000000903 blocking effect Effects 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 230000007062 hydrolysis Effects 0.000 abstract 1
- 238000006460 hydrolysis reaction Methods 0.000 abstract 1
- 239000012948 isocyanate Substances 0.000 abstract 1
- 150000002513 isocyanates Chemical class 0.000 abstract 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
- C07F9/65613—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings containing the ring system (X = CH2, O, S, NH) optionally with an additional double bond and/or substituents, e.g. cephalosporins and analogs
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Cephalosporin Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB1379978 | 1978-04-07 | ||
| GB1380178 | 1978-04-07 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2429221A1 true FR2429221A1 (fr) | 1980-01-18 |
| FR2429221B1 FR2429221B1 (de) | 1983-04-22 |
Family
ID=26250016
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7908746A Granted FR2429221A1 (fr) | 1978-04-07 | 1979-04-06 | Procede de preparation de 3-carbamoyloxymethylcephalosporines |
Country Status (11)
| Country | Link |
|---|---|
| AU (1) | AU534617B2 (de) |
| DE (1) | DE2914000A1 (de) |
| DK (1) | DK143679A (de) |
| FI (1) | FI791148A (de) |
| FR (1) | FR2429221A1 (de) |
| IE (1) | IE48286B1 (de) |
| IT (1) | IT1117214B (de) |
| NL (1) | NL7902732A (de) |
| NZ (1) | NZ190128A (de) |
| SE (1) | SE7903096L (de) |
| YU (1) | YU82379A (de) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR830000686B1 (ko) * | 1979-04-06 | 1983-03-29 | 헤롤드 월터 마틴 | 세팔로스포린 화합물의 제조방법 |
-
1979
- 1979-04-06 FR FR7908746A patent/FR2429221A1/fr active Granted
- 1979-04-06 YU YU00823/79A patent/YU82379A/xx unknown
- 1979-04-06 SE SE7903096A patent/SE7903096L/ not_active Application Discontinuation
- 1979-04-06 DE DE19792914000 patent/DE2914000A1/de not_active Withdrawn
- 1979-04-06 AU AU45896/79A patent/AU534617B2/en not_active Ceased
- 1979-04-06 DK DK143679A patent/DK143679A/da not_active Application Discontinuation
- 1979-04-06 IT IT48658/79A patent/IT1117214B/it active
- 1979-04-06 NZ NZ190128A patent/NZ190128A/xx unknown
- 1979-04-06 FI FI791148A patent/FI791148A/fi not_active Application Discontinuation
- 1979-04-06 NL NL7902732A patent/NL7902732A/xx not_active Application Discontinuation
- 1979-08-08 IE IE752/79A patent/IE48286B1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DE2914000A1 (de) | 1979-11-15 |
| AU534617B2 (en) | 1984-02-09 |
| IE48286B1 (en) | 1984-11-28 |
| IE790752L (en) | 1979-10-07 |
| SE7903096L (sv) | 1979-12-17 |
| NL7902732A (nl) | 1979-10-09 |
| FI791148A (fi) | 1979-10-08 |
| AU4589679A (en) | 1979-10-11 |
| IT1117214B (it) | 1986-02-17 |
| DK143679A (da) | 1979-10-08 |
| IT7948658A0 (it) | 1979-04-06 |
| NZ190128A (en) | 1982-03-16 |
| YU82379A (en) | 1983-01-21 |
| FR2429221B1 (de) | 1983-04-22 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ST | Notification of lapse |