FR2418233A2 - Antibiotic syn isomers of oxime(s) - of 3-alkylthio or acylamino 7-amino thiazolyl acetamido cephalosporanic acids - Google Patents

Antibiotic syn isomers of oxime(s) - of 3-alkylthio or acylamino 7-amino thiazolyl acetamido cephalosporanic acids

Info

Publication number
FR2418233A2
FR2418233A2 FR7805060A FR7805060A FR2418233A2 FR 2418233 A2 FR2418233 A2 FR 2418233A2 FR 7805060 A FR7805060 A FR 7805060A FR 7805060 A FR7805060 A FR 7805060A FR 2418233 A2 FR2418233 A2 FR 2418233A2
Authority
FR
France
Prior art keywords
alkylthio
acylamino
oxime
antibiotic
syn isomers
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7805060A
Other languages
French (fr)
Other versions
FR2418233B2 (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Roussel Uclaf SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf SA filed Critical Roussel Uclaf SA
Priority to FR7805060A priority Critical patent/FR2418233A2/en
Publication of FR2418233A2 publication Critical patent/FR2418233A2/en
Application granted granted Critical
Publication of FR2418233B2 publication Critical patent/FR2418233B2/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/59—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3 with hetero atoms directly attached in position 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)

Abstract

Synisomers of cephalosporanic acid derivs. of formula (I) are new: (where Ra is H or a 1-4C (un)satd. alkyl, R3 is 1-4C alkylthio or a radical R4-CO-NH- where R4 is 1-4C alkyl; A is H, or one equiv of an alkali or alkaline earth metal, magnesium or an aminated organic base) (I) are antibiotics active against Gram positive and negative bacteria.
FR7805060A 1978-02-22 1978-02-22 Antibiotic syn isomers of oxime(s) - of 3-alkylthio or acylamino 7-amino thiazolyl acetamido cephalosporanic acids Granted FR2418233A2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FR7805060A FR2418233A2 (en) 1978-02-22 1978-02-22 Antibiotic syn isomers of oxime(s) - of 3-alkylthio or acylamino 7-amino thiazolyl acetamido cephalosporanic acids

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7805060A FR2418233A2 (en) 1978-02-22 1978-02-22 Antibiotic syn isomers of oxime(s) - of 3-alkylthio or acylamino 7-amino thiazolyl acetamido cephalosporanic acids

Publications (2)

Publication Number Publication Date
FR2418233A2 true FR2418233A2 (en) 1979-09-21
FR2418233B2 FR2418233B2 (en) 1982-10-08

Family

ID=9204904

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7805060A Granted FR2418233A2 (en) 1978-02-22 1978-02-22 Antibiotic syn isomers of oxime(s) - of 3-alkylthio or acylamino 7-amino thiazolyl acetamido cephalosporanic acids

Country Status (1)

Country Link
FR (1) FR2418233A2 (en)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0057422A2 (en) * 1981-02-02 1982-08-11 Fujisawa Pharmaceutical Co., Ltd. New cephem compounds, processes for preparation thereof and pharmaceutical composition containing them
FR2550200A1 (en) * 1983-08-01 1985-02-08 Fujisawa Pharmaceutical Co PROCESS FOR THE PREPARATION OF CEPHEM COMPOUNDS WITH ANTIMICROBIAL ACTIVITY AND NEW PRODUCTS THUS OBTAINED

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2123544A1 (en) * 1971-01-29 1972-09-08 Glaxo Lab Ltd
FR2293935A1 (en) * 1974-12-13 1976-07-09 Lilly Co Eli 3- (SUBSTITUTE THIO) CEPHALOSPORINS ANTIBIOTICS
FR2301260A1 (en) * 1975-02-20 1976-09-17 Ciba Geigy Ag Amino-cephem derivs prepn. - by reacting 3-hydroxy-3-cephem-4-carboxylic acid derivs with amines (NL240876)

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2123544A1 (en) * 1971-01-29 1972-09-08 Glaxo Lab Ltd
FR2293935A1 (en) * 1974-12-13 1976-07-09 Lilly Co Eli 3- (SUBSTITUTE THIO) CEPHALOSPORINS ANTIBIOTICS
FR2301260A1 (en) * 1975-02-20 1976-09-17 Ciba Geigy Ag Amino-cephem derivs prepn. - by reacting 3-hydroxy-3-cephem-4-carboxylic acid derivs with amines (NL240876)

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0057422A2 (en) * 1981-02-02 1982-08-11 Fujisawa Pharmaceutical Co., Ltd. New cephem compounds, processes for preparation thereof and pharmaceutical composition containing them
EP0057422A3 (en) * 1981-02-02 1983-11-23 Fujisawa Pharmaceutical Co., Ltd. New cephem compounds, processes for preparation thereof and pharmaceutical composition containing them
FR2550200A1 (en) * 1983-08-01 1985-02-08 Fujisawa Pharmaceutical Co PROCESS FOR THE PREPARATION OF CEPHEM COMPOUNDS WITH ANTIMICROBIAL ACTIVITY AND NEW PRODUCTS THUS OBTAINED
EP0133678A2 (en) * 1983-08-01 1985-03-06 Fujisawa Pharmaceutical Co., Ltd. New cephem compounds, processes for preparation thereof and pharmaceutical compositions containing them
EP0133678A3 (en) * 1983-08-01 1986-03-19 Fujisawa Pharmaceutical Co., Ltd. New cephem compounds, processes for preparation thereof and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
FR2418233B2 (en) 1982-10-08

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