FR2397418A1 - Esters de penicilline utilisables comme medicaments et procede pour leur preparation - Google Patents

Esters de penicilline utilisables comme medicaments et procede pour leur preparation

Info

Publication number
FR2397418A1
FR2397418A1 FR7820783A FR7820783A FR2397418A1 FR 2397418 A1 FR2397418 A1 FR 2397418A1 FR 7820783 A FR7820783 A FR 7820783A FR 7820783 A FR7820783 A FR 7820783A FR 2397418 A1 FR2397418 A1 FR 2397418A1
Authority
FR
France
Prior art keywords
preparation
medicinal products
esters
penicillin esters
penicillin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
FR7820783A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Beecham Group PLC
Original Assignee
Beecham Group PLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beecham Group PLC filed Critical Beecham Group PLC
Publication of FR2397418A1 publication Critical patent/FR2397418A1/fr
Pending legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/429—Thiazoles condensed with heterocyclic ring systems
    • A61K31/43—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Cette invention concerne une classe d'esters de la pénicilline dénommée nafcilline. Ces esters répondent à la formule générale :
FR7820783A 1977-07-14 1978-07-12 Esters de penicilline utilisables comme medicaments et procede pour leur preparation Pending FR2397418A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB2958377 1977-07-14

Publications (1)

Publication Number Publication Date
FR2397418A1 true FR2397418A1 (fr) 1979-02-09

Family

ID=10293839

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7820783A Pending FR2397418A1 (fr) 1977-07-14 1978-07-12 Esters de penicilline utilisables comme medicaments et procede pour leur preparation

Country Status (4)

Country Link
US (1) US4215120A (fr)
JP (1) JPS5419993A (fr)
DE (1) DE2831031A1 (fr)
FR (1) FR2397418A1 (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5324463B2 (ja) * 2006-12-10 2013-10-23 チョンシー ユー β−ラクタム抗生物質の経皮送達システム
US9969751B2 (en) 2009-06-10 2018-05-15 Techfields Pharma Co., Ltd. High penetration prodrug compositions of antimicrobials and antimicrobial-related compounds
RU2016115906A (ru) * 2009-06-10 2018-11-28 Текфилдз Байокем Ко., Лтд. Композиции или пролекарства противомикробных и родственных противомикробным соединений, обладающие высокой проникающей способностью
IN2014KN02583A (fr) 2012-05-16 2015-05-08 Techfields Pharma Co Ltd
JP5795343B2 (ja) * 2013-01-23 2015-10-14 チョンシー ユー β−ラクタム抗生物質の経皮送達システム
CN104356143B (zh) * 2014-10-27 2017-08-29 桂林南药股份有限公司 一种萘夫西林酸的制备方法

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1021654A (fr) * 1949-07-07 1953-02-23 Lphivens Kemiske Fabrik Ved A Procédé de production d'éthers-sels aminés de pénicilline et de composés qui s'y rattachent
DE2725695A1 (de) * 1976-06-11 1977-12-22 Beecham Group Ltd Arzneipraeparate fuer eine orale verabreichung

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB675422A (en) * 1949-07-07 1952-07-09 Knud Abildgaard Elling Preparation of amino esters of penicillin and salts thereof
US3157639A (en) * 1959-08-19 1964-11-17 Beecham Group Ltd Synthetic penicillins
ES428213A1 (es) * 1974-07-12 1976-07-16 Andreu Sa Dr Procedimiento para la obtencion de esteres dialquilaminoal-quilicos de penicilina.
GB1578730A (en) * 1976-06-24 1980-11-05 Beecham Group Ltd Esters of penicillin antibiotics

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1021654A (fr) * 1949-07-07 1953-02-23 Lphivens Kemiske Fabrik Ved A Procédé de production d'éthers-sels aminés de pénicilline et de composés qui s'y rattachent
DE2725695A1 (de) * 1976-06-11 1977-12-22 Beecham Group Ltd Arzneipraeparate fuer eine orale verabreichung

Also Published As

Publication number Publication date
US4215120A (en) 1980-07-29
JPS5419993A (en) 1979-02-15
DE2831031A1 (de) 1979-02-01

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