FI972284A - cis-(+)-3-(4,6-dihydroksikroman-3-yylimetyyli)-4-metoksianiliinin valmistusmenetelmiä ja niissä käytettyjä välituotteita - Google Patents

cis-(+)-3-(4,6-dihydroksikroman-3-yylimetyyli)-4-metoksianiliinin valmistusmenetelmiä ja niissä käytettyjä välituotteita Download PDF

Info

Publication number
FI972284A
FI972284A FI972284A FI972284A FI972284A FI 972284 A FI972284 A FI 972284A FI 972284 A FI972284 A FI 972284A FI 972284 A FI972284 A FI 972284A FI 972284 A FI972284 A FI 972284A
Authority
FI
Finland
Prior art keywords
methoxyaniline
ylmethyl
cis
dihydroxycroman
compounds
Prior art date
Application number
FI972284A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI972284A0 (fi
Inventor
George J Quallich
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI972284A0 publication Critical patent/FI972284A0/fi
Publication of FI972284A publication Critical patent/FI972284A/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/22Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Pyrane Compounds (AREA)
FI972284A 1994-11-30 1997-05-29 cis-(+)-3-(4,6-dihydroksikroman-3-yylimetyyli)-4-metoksianiliinin valmistusmenetelmiä ja niissä käytettyjä välituotteita FI972284A (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/346,955 US5539128A (en) 1994-11-30 1994-11-30 Processes and intermediates for preparing cis(+)3-[4,6-dihydroxy chroman-3-ylmethyl]-4-methoxyaniline
PCT/IB1995/000846 WO1996016955A1 (en) 1994-11-30 1995-10-06 Processes and intermediates for preparing cis(+)3-[4,-6-dihydroxychroman-3-ylmethyl]-4-methoxyaniline

Publications (2)

Publication Number Publication Date
FI972284A0 FI972284A0 (fi) 1997-05-29
FI972284A true FI972284A (fi) 1997-05-29

Family

ID=23361728

Family Applications (1)

Application Number Title Priority Date Filing Date
FI972284A FI972284A (fi) 1994-11-30 1997-05-29 cis-(+)-3-(4,6-dihydroksikroman-3-yylimetyyli)-4-metoksianiliinin valmistusmenetelmiä ja niissä käytettyjä välituotteita

Country Status (12)

Country Link
US (1) US5539128A (da)
EP (1) EP0794951B1 (da)
JP (1) JP3041049B2 (da)
AT (1) ATE191715T1 (da)
CA (1) CA2204604C (da)
DE (1) DE69516305T2 (da)
DK (1) DK0794951T3 (da)
ES (1) ES2144628T3 (da)
FI (1) FI972284A (da)
GR (1) GR3033608T3 (da)
PT (1) PT794951E (da)
WO (1) WO1996016955A1 (da)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU713701B2 (en) * 1996-09-16 1999-12-09 Pfizer Inc. Processes and intermediates for preparing substituted chromanol derivatives

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4661596A (en) * 1985-02-21 1987-04-28 American Home Products Corporation Quinolinyl (or pyridinyl) methoxy substituted naphthalene compounds as antiallergic agents
US5059609A (en) * 1987-10-19 1991-10-22 Pfizer Inc. Substituted tetralins, chromans and related compounds in the treatment of asthma, arthritis and related diseases
WO1990015801A1 (en) * 1989-06-22 1990-12-27 Pfizer Inc. Substituted sulfonamides and related compounds in the treatment of asthma, arthritis and related diseases
US4987231A (en) * 1989-08-04 1991-01-22 Pfizer Inc. Optical resolution method for 3R-(3-carboxybenzyl)-6-(5-fluoro-2-benzothiazolyl)methoxy-4R-chromanol
CZ100095A3 (en) * 1992-10-21 1995-11-15 Pfizer Sulfonamide derivatives of hydroxy substituted alicyclic or heterocyclic compounds with condensed benzene nucleus and pharmaceutical preparations based thereon

Also Published As

Publication number Publication date
ES2144628T3 (es) 2000-06-16
EP0794951A1 (en) 1997-09-17
FI972284A0 (fi) 1997-05-29
DE69516305T2 (de) 2001-02-15
WO1996016955A1 (en) 1996-06-06
DK0794951T3 (da) 2000-07-10
EP0794951B1 (en) 2000-04-12
ATE191715T1 (de) 2000-04-15
CA2204604C (en) 2002-02-19
MX9703989A (es) 1997-09-30
CA2204604A1 (en) 1996-06-06
PT794951E (pt) 2000-07-31
GR3033608T3 (en) 2000-10-31
DE69516305D1 (de) 2000-05-18
US5539128A (en) 1996-07-23
JPH10500143A (ja) 1998-01-06
JP3041049B2 (ja) 2000-05-15

Similar Documents

Publication Publication Date Title
FI932229A (fi) Azabicykliska bryggderivat
AU1889392A (en) Fluoroalkoxybenzylamino derivatives of nitrogen containing heterocycles
ATE224374T1 (de) 1,2-substituierte imidazolylverbindungen zur behandlung von entzündungen
DE3681518D1 (de) Pyridinderivate, deren herstellung und anwendung.
FI931765A0 (fi) Steroidderivat foer behandling av prostatahypertrofi, deras framstaellning och anvaendningar
DE69523155D1 (de) Benzimidazolonderivate mit zentraler dopaminerger aktivität
CA2238283A1 (en) Method for identifying compounds for inhibition of neoplastic lesions, pharmaceutical compositions from such compounds and uses of such compounds and compositions for treating neoplastic lesions
DK0654041T3 (da) Peptidyl-4-amino-2,2-difluor-3-oxo-1,6-hexandisyre-derivater som anto-inflammatoriske midler
AU2351095A (en) Benzimidazole derivatives having dopaminergic activity
FI972284A0 (fi) cis-(+)-3-(4,6-dihydroksikroman-3-yylimetyyli)-4-metoksianiliinin valmistusmenetelmiä ja niissä käytettyjä välituotteita
MA22926A1 (fr) Procede pour la preparation de nouveaux composes.
CA2083361A1 (en) Fish production
DE69310353T2 (de) 2,3,4,5-tetrahydro-1h-3-benzazepine und ihre pharmazeutisch verträglichen säureadditionssalze
CA2175352A1 (en) 3-Aryl-4-Alkyl and 4,5-Dialkyl-4H-1,2,4-Triazoles Useful as Memory Enhancers
AU2178099A (en) Azetidinecarboxamide derivatives for treating cns disorders
ES2004215A6 (es) Procedimiento para preparar quinazolinas tetraciclicas
ES8308828A1 (es) "procedimiento para la preparacion de (+)-6-metoxi-x-metil-2-naftalen-acetato de n,n"-bis-(4-clorofenil)-1,12-diimino-2,4,11-13-tetraaza-tetradecandiimidoamida".
KR970702869A (ko) 항종양성 인돌로피롤로카르바졸 유도체(antitumor indolopyprolocarbazole derivative)
SE8800480D0 (sv) Arylamider av alfa-hexametyleniminokarbonsyror och hydroklorider av dessa arylamider
MY104184A (en) A sampled data phase locking system