FI950488A0 - Kinuklidiinijohdannaisia skvaleenisyntaasi-inhibiittoreina - Google Patents

Kinuklidiinijohdannaisia skvaleenisyntaasi-inhibiittoreina

Info

Publication number
FI950488A0
FI950488A0 FI950488A FI950488A FI950488A0 FI 950488 A0 FI950488 A0 FI 950488A0 FI 950488 A FI950488 A FI 950488A FI 950488 A FI950488 A FI 950488A FI 950488 A0 FI950488 A0 FI 950488A0
Authority
FI
Finland
Prior art keywords
pct
derivatives
hydroxy
squalene synthase
alkyl
Prior art date
Application number
FI950488A
Other languages
English (en)
Swedish (sv)
Other versions
FI950488A (fi
Inventor
Keith Blakeney Mallion
George Robert Brown
Paul Robert Owen Whittamore
Original Assignee
Zeneca Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zeneca Ltd filed Critical Zeneca Ltd
Publication of FI950488A0 publication Critical patent/FI950488A0/fi
Publication of FI950488A publication Critical patent/FI950488A/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Enzymes And Modification Thereof (AREA)
FI950488A 1992-08-06 1995-02-03 Kinuklidiinijohdannaisia skvaleenisyntaasi-inhibiittoreina FI950488A (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB929216721A GB9216721D0 (en) 1992-08-06 1992-08-06 Therapeutic heterocyclic derivatives
PCT/GB1993/001648 WO1994003451A1 (en) 1992-08-06 1993-08-04 Quinuclidine derivatives as squalene synthase inhibitors

Publications (2)

Publication Number Publication Date
FI950488A0 true FI950488A0 (fi) 1995-02-03
FI950488A FI950488A (fi) 1995-03-10

Family

ID=10719936

Family Applications (1)

Application Number Title Priority Date Filing Date
FI950488A FI950488A (fi) 1992-08-06 1995-02-03 Kinuklidiinijohdannaisia skvaleenisyntaasi-inhibiittoreina

Country Status (13)

Country Link
US (1) US5691349A (fi)
EP (1) EP0654032B1 (fi)
JP (1) JPH08500098A (fi)
AT (1) ATE159255T1 (fi)
AU (1) AU4721193A (fi)
CA (2) CA2141806A1 (fi)
DE (1) DE69314649T2 (fi)
FI (1) FI950488A (fi)
GB (2) GB9216721D0 (fi)
IL (1) IL106583A0 (fi)
TW (1) TW231292B (fi)
WO (1) WO1994003451A1 (fi)
ZA (1) ZA935655B (fi)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL109451A0 (en) * 1993-04-29 1994-07-31 Zeneca Ltd Heterocyclic derivatives
GB9412145D0 (en) * 1994-06-17 1994-08-10 Zeneca Ltd Heterocycles
US5556990A (en) * 1994-12-16 1996-09-17 Rhone-Poulenc Rorer Pharmaceuticals Inc. Polyarylcarbamoylaza- and -carbamoylalkanedioic acids
AU7247898A (en) * 1997-04-11 1998-11-11 Eli Lilly And Company Composition for treating pain
US6284910B1 (en) 1998-12-15 2001-09-04 University Of Kentucky Research Foundation Farnesyl pyrophosphate analogs
US6433168B1 (en) * 1999-07-26 2002-08-13 Sumika Fine Chemicals Co., Ltd. Highly pure phenothiazine compound, production method thereof, production method of intermediate therefor, and hydrate and novel crystal as starting materials for the intermediate
PL370087A1 (en) * 2001-10-17 2005-05-16 Ucb, S.A. Quinuclidine derivatives, processes for preparing them and their uses as m2 and/or m3 muscarinic receptor inhibitors
GB0127731D0 (en) * 2001-11-20 2002-01-09 Coin Controls Coin handling apparatus
CN117380646B (zh) * 2023-12-12 2024-03-12 柞水县宝华矿业有限公司 一种石英砂除杂清洗装置

Family Cites Families (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3405134A (en) * 1965-08-17 1968-10-08 Colgate Palmolive Co Quinuclidyl esters of aromatic acids
NL6715600A (fi) * 1966-12-02 1968-06-04
US3534053A (en) * 1967-05-24 1970-10-13 American Home Prod Quinuclidine derivatives
US3763168A (en) * 1968-09-09 1973-10-02 Sterling Drug Inc N-(3-quinuclidinyl) acylanilides
US3655675A (en) * 1968-09-09 1972-04-11 Sterling Drug Inc N-(n-heteryl)-acylanilides
US3725410A (en) * 1970-07-15 1973-04-03 American Home Prod 3-aminomethyl-3-quinuclidinols
US3679690A (en) * 1971-03-18 1972-07-25 Sterling Drug Inc Certain n-(pyridyl) propionanilides
FR2183565B1 (fi) * 1972-05-10 1975-12-26 Cerm Cent Europ Rech Mauvernay
CA1014958A (en) * 1973-10-05 1977-08-02 Jacques Moleyre .alpha.-QUINUCLIDYLMETHYL PHENYL KETONES
SU495310A1 (ru) * 1974-03-05 1975-12-15 Всесоюзный Научно-Исследовательский Химико-Фармацевтический Институт Им.С.Орджоникидзе Хинуклидил-3-диарал(гетерил) карбинолы, про вл ющие антигистаминную, антисеротониновую и антиаллергическую активность и способ их получени
US4038402A (en) * 1974-03-05 1977-07-26 Mikhail Emmanuilovich Kaminka Method of effecting antihistaminic, antiserotonin and antiallergic actions
US4599344A (en) * 1984-10-31 1986-07-08 Schering A.G. Quinuclidines and quinuclidinium salts as antiarrhythmic agents
CH667657A5 (de) * 1985-01-07 1988-10-31 Sandoz Ag Carbocyclische und heterocyclische carbonylmethylen- und methylpiperidine und -pyrrolidine.
NZ225999A (en) * 1987-09-10 1992-04-28 Merck Sharp & Dohme Azacyclic- or azabicyclic-substituted thiadiazole derivatives and pharmaceutical compositions
IL88156A (en) * 1987-11-13 1997-02-18 Novo Nordisk As Azacyclic compounds their preparation and pharmaceutical compositions containing them
EP0322182A3 (en) * 1987-12-22 1992-01-02 Beecham Group Plc Azabicyclic compounds, process for their preparation and pharmaceutical compositions containing them
DK730588A (da) * 1988-02-03 1989-08-04 Asta Pharma Ag Anvendelse af pyridin-2-ethere eller pyridin-2-thioethere med en nitrogenholdig cycloalifatisk ring som antidepressivt laegemiddel
NZ227841A (en) * 1988-02-12 1991-08-27 Merck Sharp & Dohme Heterocyclic compounds with at least two non-condensed five membered rings and pharmaceutical compositions
DK175029B1 (da) * 1988-04-01 2004-05-03 Sankyo Co 2-(heterocyclylthio)carbapenemderivater, farmaceutiske midler indeholdende dem, fremgangsmåde til fremstilling deraf samt deres anvendelse som antibiotika
US5242914A (en) * 1988-04-01 1993-09-07 Sankyo Company, Limited 2-(heterocyclylthio) carbapenem derivatives, their preparation and their use as antibiotics
US5286864A (en) * 1988-11-22 1994-02-15 Boehringer Ingelheim Kg Quinuclidines, their use as medicaments and processes for their preparation
DE3839385A1 (de) * 1988-11-22 1990-05-23 Boehringer Ingelheim Kg Neue quinuclidine, ihre herstellung als arzneimittel und verfahren zu ihrer herstellung
GB8918061D0 (en) * 1989-08-08 1989-09-20 Merck Sharp & Dohme Therapeutic agents
YU84791A (sh) * 1990-05-19 1994-06-10 Boehringer Ingelheim Kg. Biciklicni 1-aza-cikloalkalni
DE4116582A1 (de) * 1990-05-19 1991-11-21 Boehringer Ingelheim Kg Bicyclische 1-aza-cycloalkane
ZA92278B (en) * 1991-02-01 1992-10-28 Akzo Nv 3-quinuclidine derivatives
AU1752792A (en) * 1991-03-08 1992-10-06 Rhone-Poulenc Rorer International (Holdings) Inc. Multicyclic tertiary amine polyaromatic squalene synthetase inhibitors
US5385912A (en) * 1991-03-08 1995-01-31 Rhone-Poulenc Rorer Pharmaceuticals Inc. Multicyclic tertiary amine polyaromatic squalene synthase inhibitors
US5135935A (en) * 1991-05-17 1992-08-04 Merck & Co., Inc. Squalene synthetase inhibitors
GB9201749D0 (en) * 1992-01-28 1992-03-11 Smithkline Beecham Plc Medicaments
GB9202443D0 (en) * 1992-02-05 1992-03-18 Fujisawa Pharmaceutical Co A novel substituted-acetamide compound and a process for the preparation thereof

Also Published As

Publication number Publication date
CA2101901A1 (en) 1994-02-07
DE69314649T2 (de) 1998-03-05
ZA935655B (en) 1994-02-08
TW231292B (fi) 1994-10-01
EP0654032B1 (en) 1997-10-15
DE69314649D1 (de) 1997-11-20
ATE159255T1 (de) 1997-11-15
IL106583A0 (en) 1993-12-08
CA2141806A1 (en) 1994-02-17
WO1994003451A1 (en) 1994-02-17
FI950488A (fi) 1995-03-10
GB9315510D0 (en) 1993-09-08
AU4721193A (en) 1994-03-03
US5691349A (en) 1997-11-25
JPH08500098A (ja) 1996-01-09
EP0654032A1 (en) 1995-05-24
GB9216721D0 (en) 1992-09-23

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Legal Events

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