FI944014A0 - Makrolidien desosaminojohdannaiset immuunivastetta heikentävinä aineina ja sieniä vastustavina aineina - Google Patents

Makrolidien desosaminojohdannaiset immuunivastetta heikentävinä aineina ja sieniä vastustavina aineina

Info

Publication number
FI944014A0
FI944014A0 FI944014A FI944014A FI944014A0 FI 944014 A0 FI944014 A0 FI 944014A0 FI 944014 A FI944014 A FI 944014A FI 944014 A FI944014 A FI 944014A FI 944014 A0 FI944014 A0 FI 944014A0
Authority
FI
Finland
Prior art keywords
macrolides
pct
immunosuppressants
antifungal agents
desosamine
Prior art date
Application number
FI944014A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI944014A (fi
Inventor
James R Hauske
Gary R Schulte
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI944014A publication Critical patent/FI944014A/fi
Publication of FI944014A0 publication Critical patent/FI944014A0/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
FI944014A 1992-03-02 1994-09-01 Makrolidien desosaminojohdannaiset immuunivastetta heikentävinä aineina ja sieniä vastustavina aineina FI944014A0 (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US84435092A 1992-03-02 1992-03-02
PCT/US1993/000426 WO1993018042A1 (fr) 1992-03-02 1993-01-27 Derives de desosamino de macrolides utiles comme immunosuppresseurs et antifongiques

Publications (2)

Publication Number Publication Date
FI944014A FI944014A (fi) 1994-09-01
FI944014A0 true FI944014A0 (fi) 1994-09-01

Family

ID=25292478

Family Applications (1)

Application Number Title Priority Date Filing Date
FI944014A FI944014A0 (fi) 1992-03-02 1994-09-01 Makrolidien desosaminojohdannaiset immuunivastetta heikentävinä aineina ja sieniä vastustavina aineina

Country Status (12)

Country Link
US (2) US5506233A (fr)
EP (1) EP0629203B1 (fr)
JP (1) JPH07500613A (fr)
AT (1) ATE205496T1 (fr)
CA (1) CA2131371A1 (fr)
DE (1) DE69330747T2 (fr)
DK (1) DK0629203T3 (fr)
ES (1) ES2160593T3 (fr)
FI (1) FI944014A0 (fr)
GR (1) GR3037059T3 (fr)
PT (1) PT629203E (fr)
WO (1) WO1993018042A1 (fr)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2182004C1 (ru) * 2001-02-22 2002-05-10 Общество С Ограниченной Ответственностью "Научно-Технологическая Фармацевтическая Фирма "Полисан" Лекарственный препарат для парентерального применения
EP1554572B1 (fr) 2001-07-25 2009-10-14 Raptor Pharmaceutical Inc. Compositions et procedes de modulation du transport a travers la barriere hematho-encephalique
US7452692B2 (en) * 2002-02-13 2008-11-18 Teva Gyógyszergyár Zártkörüen Müködö Részvénytársaság Method for extracting a macrolide from biomatter
MXPA04007847A (es) 2002-02-13 2005-02-24 Biogal Gyogyszergyar Metodo para extraer un macrolido de biomateria.
US20060169199A1 (en) * 2003-03-31 2006-08-03 Vilmos Keri Crystallization and purification of macrolides
ES2229975T1 (es) * 2003-03-31 2005-05-01 Teva Gyogyszergyar Reszvenytarsasag Cristalizacion y purificacion de macrolidos.
US7160867B2 (en) * 2003-05-16 2007-01-09 Isotechnika, Inc. Rapamycin carbohydrate derivatives
DK1558622T3 (da) * 2003-07-24 2008-02-25 Teva Gyogyszergyar Zartkoeruee Fremgangsmåde til oprensning af macrolider
CA2571710A1 (fr) 2004-06-24 2006-11-02 Nicholas Valiante Immuno-potentialisateurs a petites molecules et analyses visant a detecter leur presence
MX2007005867A (es) * 2004-12-22 2007-07-04 Teva Gyogyszergyar Zartkoeruen Mukoedo Reszvenytarsasag Metodo de purificar macrolidos.
US20060154953A1 (en) * 2005-01-05 2006-07-13 Vilmos Keri Amorphous tacrolimus and preparation thereof
EP2671508B1 (fr) 2005-04-28 2020-09-16 Proteus Digital Health, Inc. Système pharma-informatique
DE602007006601D1 (de) * 2006-03-15 2010-07-01 Teva Gyogyszergyar Zartkoeruee Verfahren zur reinigung von tacrolimus
JP2009203162A (ja) * 2006-06-05 2009-09-10 Astellas Pharma Inc マクロライド化合物の新規製造法
EP2063905B1 (fr) 2006-09-18 2014-07-30 Raptor Pharmaceutical Inc Traitement des troubles hépatiques par l'administration de conjugués de protéine associée au récepteur (rap)
EP4218718A3 (fr) 2009-05-06 2024-04-24 Laboratory Skin Care, Inc. Compositions pour libération dermique comprenant des complexes principe actif-particule de phosphate de calcium et procédés d'utilisation associés
US20120077778A1 (en) 2010-09-29 2012-03-29 Andrea Bourdelais Ladder-Frame Polyether Conjugates

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4894366A (en) * 1984-12-03 1990-01-16 Fujisawa Pharmaceutical Company, Ltd. Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same
AU6286690A (en) * 1989-08-18 1991-04-03 Fisons Plc Macrocyclic compounds
IE904050A1 (en) * 1989-11-13 1991-05-22 Merck & Co Inc Aminomacrolides and derivatives having immunosuppressive¹activity
EP0466365A3 (en) * 1990-07-03 1992-04-15 Merck & Co. Inc. Novel immunosuppressant fermentation products of a microorganism

Also Published As

Publication number Publication date
DE69330747D1 (de) 2001-10-18
EP0629203A1 (fr) 1994-12-21
US5563135A (en) 1996-10-08
ES2160593T3 (es) 2001-11-16
EP0629203B1 (fr) 2001-09-12
DE69330747T2 (de) 2002-05-29
FI944014A (fi) 1994-09-01
US5506233A (en) 1996-04-09
DK0629203T3 (da) 2001-11-12
PT629203E (pt) 2002-01-30
GR3037059T3 (en) 2002-01-31
ATE205496T1 (de) 2001-09-15
CA2131371A1 (fr) 1993-09-16
JPH07500613A (ja) 1995-01-19
WO1993018042A1 (fr) 1993-09-16

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