FI944013A0 - Välituotteiden valmistus kinoliiniantibioottien synteesissä - Google Patents

Välituotteiden valmistus kinoliiniantibioottien synteesissä

Info

Publication number
FI944013A0
FI944013A0 FI944013A FI944013A FI944013A0 FI 944013 A0 FI944013 A0 FI 944013A0 FI 944013 A FI944013 A FI 944013A FI 944013 A FI944013 A FI 944013A FI 944013 A0 FI944013 A0 FI 944013A0
Authority
FI
Finland
Prior art keywords
intermediates
synthesis
preparation
quinoline antibiotics
quinoline
Prior art date
Application number
FI944013A
Other languages
English (en)
Swedish (sv)
Other versions
FI106022B (fi
FI944013A (fi
Inventor
Tamim F Braish
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI944013A0 publication Critical patent/FI944013A0/fi
Publication of FI944013A publication Critical patent/FI944013A/fi
Application granted granted Critical
Publication of FI106022B publication Critical patent/FI106022B/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Indole Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
FI944013A 1992-03-02 1994-09-01 Menetelmä (1a, 5a, 6a)-3-(N-substituoitu)-6-[(N-suojattu) - amino]-3-atsabisyklo[3.1.0]heksaani-välituotteen valmistamiseksi kinoliiniantibioottien synteesissä ja menetelmän välituotteita FI106022B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US84436792 1992-03-02
US07/844,367 US5256791A (en) 1992-03-02 1992-03-02 Preparation of intermediates in the synthesis of quinoline antibiotics
US9300008 1993-01-07
PCT/US1993/000008 WO1993018001A1 (en) 1992-03-02 1993-01-07 Preparation of intermediates in the synthesis of quinoline antibiotics

Publications (3)

Publication Number Publication Date
FI944013A0 true FI944013A0 (fi) 1994-09-01
FI944013A FI944013A (fi) 1994-09-01
FI106022B FI106022B (fi) 2000-11-15

Family

ID=25292537

Family Applications (1)

Application Number Title Priority Date Filing Date
FI944013A FI106022B (fi) 1992-03-02 1994-09-01 Menetelmä (1a, 5a, 6a)-3-(N-substituoitu)-6-[(N-suojattu) - amino]-3-atsabisyklo[3.1.0]heksaani-välituotteen valmistamiseksi kinoliiniantibioottien synteesissä ja menetelmän välituotteita

Country Status (22)

Country Link
US (2) US5256791A (fi)
EP (1) EP0629189B1 (fi)
JP (1) JP2564247B2 (fi)
KR (2) KR0135626B1 (fi)
CN (1) CN1037100C (fi)
AT (1) ATE156480T1 (fi)
AU (1) AU667872B2 (fi)
CA (1) CA2131160C (fi)
DE (1) DE69312913T2 (fi)
DK (1) DK0629189T3 (fi)
ES (1) ES2105217T3 (fi)
FI (1) FI106022B (fi)
GR (1) GR3024789T3 (fi)
HU (1) HU215837B (fi)
IL (1) IL104818A (fi)
MX (1) MX9301138A (fi)
MY (1) MY107723A (fi)
NO (1) NO300681B1 (fi)
NZ (1) NZ246768A (fi)
TW (1) TW211002B (fi)
WO (1) WO1993018001A1 (fi)
ZA (1) ZA931428B (fi)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5475116A (en) * 1994-04-29 1995-12-12 Pfizer Inc. Aza bicyclo[3,1,0]hexane intermediates useful in the synthesis of quinolones
US5929240A (en) * 1994-12-12 1999-07-27 Pfizer Inc. Process and intermediates for preparing naphthyridonecarboxylic acid salts
JPH0912547A (ja) * 1995-06-23 1997-01-14 Chisso Corp ニューキノロン系化合物中間体の製造方法
GB9524466D0 (en) * 1995-11-30 1996-01-31 Pfizer Ltd Process
JPH1087617A (ja) * 1996-07-09 1998-04-07 Pfizer Inc キノリン系抗生物質の合成に有用な中間体の製法
GB9614422D0 (en) * 1996-07-09 1996-09-04 Pfizer Ltd Novel process
US6057455A (en) * 1996-07-09 2000-05-02 Pfizer, Inc. Preparation of intermediates useful in the synthesis of quinoline antibiotics
HN1998000106A (es) 1997-08-01 1999-01-08 Pfizer Prod Inc Composiciones parenterales de alatroflaxacino
DE19733439A1 (de) * 1997-08-02 1999-02-04 Bayer Ag Neue 6-endo-Amino-3-azabicyclo(3.1.0)hexande, Verfahren zu deren Herstellung und deren Verwendung zur Herstellung von Chinolon- und Naphthyridincarbonsäure-Derviaten mit verbesserten Eigenschaften
PA8464701A1 (es) * 1998-01-16 2000-09-29 Pfizer Prod Inc Procedimiento e intermedios para preparar naftiridonas
US7019142B2 (en) 1998-01-16 2006-03-28 Pfizer Inc. Process for preparing naphthyridones and intermediates
US6184380B1 (en) * 1999-01-25 2001-02-06 Pfizer Inc. Process for preparing naphthyridones and intermediates
WO2008010061A2 (en) * 2006-07-17 2008-01-24 Glenmark Pharmaceuticals S.A. 3-azabicyclo [3.1.0] hexane vanilloid receptor ligands, pharmaceutical compositions containing them, and processes for their preparation
WO2020243423A1 (en) 2019-05-31 2020-12-03 Ikena Oncology, Inc. Tead inhibitors and uses thereof
CN114466839A (zh) 2019-05-31 2022-05-10 医肯纳肿瘤学公司 Tead抑制剂和其用途
WO2023151188A1 (zh) * 2022-02-08 2023-08-17 上海皓元医药股份有限公司 一种抗病毒药物中间体的绿色合成方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4183857A (en) * 1978-07-06 1980-01-15 Shell Oil Company 3-Benzyl-3-azabicyclo(3.1.0)hexane-2,4-dione
EP0010799B1 (en) * 1978-10-27 1982-05-19 Shell Internationale Researchmaatschappij B.V. A process for the preparation of 3-azabicyclo(3.1.0)hexane derivatives and modifications thereof
JPH0676400B2 (ja) * 1987-08-25 1994-09-28 大日本製薬株式会社 新規ピリドンカルボン酸誘導体、そのエステルおよびその塩
US5196548A (en) * 1989-05-11 1993-03-23 Pfizer Inc. Preparation of diazabicyclic Intermediates
PL166381B1 (pl) * 1989-08-16 1995-05-31 Pfizer Sposób wytwarzania nowych podstawionych kwasów 7-azabicyklochinolonokarboksylowych PL PL PL PL
US5200527A (en) * 1991-04-08 1993-04-06 Lonza Ltd. Process for the production of 2-azabicyclo [2.2.1] hept-5-en-3-one

Also Published As

Publication number Publication date
KR950700251A (ko) 1995-01-16
IL104818A0 (en) 1993-06-10
MY107723A (en) 1996-05-30
ZA931428B (en) 1994-09-01
JP2564247B2 (ja) 1996-12-18
NO943243L (no) 1994-09-01
FI106022B (fi) 2000-11-15
DK0629189T3 (da) 1997-12-08
NO943243D0 (no) 1994-09-01
DE69312913T2 (de) 1997-11-20
HUT70497A (en) 1995-10-30
AU3430093A (en) 1993-10-05
CA2131160A1 (en) 1993-09-16
US5298629A (en) 1994-03-29
WO1993018001A1 (en) 1993-09-16
US5256791A (en) 1993-10-26
AU667872B2 (en) 1996-04-18
KR0135626B1 (ko) 1998-04-23
HU215837B (en) 2001-03-28
CN1037100C (zh) 1998-01-21
MX9301138A (es) 1994-01-31
GR3024789T3 (en) 1998-01-30
ATE156480T1 (de) 1997-08-15
NZ246768A (en) 1995-09-26
EP0629189A1 (en) 1994-12-21
CA2131160C (en) 1997-11-18
ES2105217T3 (es) 1997-10-16
HU9402530D0 (en) 1994-11-28
DE69312913D1 (de) 1997-09-11
IL104818A (en) 1997-09-30
CN1076440A (zh) 1993-09-22
JPH07500349A (ja) 1995-01-12
NO300681B1 (no) 1997-07-07
TW211002B (en) 1993-08-11
EP0629189B1 (en) 1997-08-06
FI944013A (fi) 1994-09-01

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