FI940775L - alfa-fenyyli-isoseriinijohdannaisten valmistusmentelmä ja niiden käyttö - Google Patents
alfa-fenyyli-isoseriinijohdannaisten valmistusmentelmä ja niiden käyttö Download PDFInfo
- Publication number
- FI940775L FI940775L FI940775A FI940775A FI940775L FI 940775 L FI940775 L FI 940775L FI 940775 A FI940775 A FI 940775A FI 940775 A FI940775 A FI 940775A FI 940775 L FI940775 L FI 940775L
- Authority
- FI
- Finland
- Prior art keywords
- preparing alpha
- phenylisoserine derivatives
- phenylisoserine
- derivatives
- alpha
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C231/00—Preparation of carboxylic acid amides
- C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C269/06—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups by reactions not involving the formation of carbamate groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Epoxy Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR919110398A FR2680506B1 (fr) | 1991-08-19 | 1991-08-19 | Procede de preparation de derives de la beta-phenylisoserine et leur utilisation. |
| PCT/FR1992/000795 WO1993004038A1 (fr) | 1991-08-19 | 1992-08-17 | PROCEDE DE PREPARATION DE DERIVES DE LA β-PHENYLISOSERINE ET LEUR UTILISATION |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| FI940775A0 FI940775A0 (fi) | 1994-02-18 |
| FI940775A7 FI940775A7 (fi) | 1994-02-18 |
| FI940775L true FI940775L (fi) | 1994-02-18 |
Family
ID=9416254
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI940775A FI940775L (fi) | 1991-08-19 | 1992-08-17 | alfa-fenyyli-isoseriinijohdannaisten valmistusmentelmä ja niiden käyttö |
Country Status (16)
| Country | Link |
|---|---|
| EP (2) | EP0599973A1 (OSRAM) |
| JP (1) | JPH06510033A (OSRAM) |
| AU (1) | AU2490492A (OSRAM) |
| CA (1) | CA2113827A1 (OSRAM) |
| CZ (1) | CZ35494A3 (OSRAM) |
| FI (1) | FI940775L (OSRAM) |
| FR (1) | FR2680506B1 (OSRAM) |
| HU (1) | HUT68255A (OSRAM) |
| MX (1) | MX9204635A (OSRAM) |
| NO (1) | NO940027D0 (OSRAM) |
| NZ (1) | NZ243972A (OSRAM) |
| SK (1) | SK19094A3 (OSRAM) |
| TW (1) | TW222620B (OSRAM) |
| WO (1) | WO1993004038A1 (OSRAM) |
| YU (1) | YU78092A (OSRAM) |
| ZA (1) | ZA926189B (OSRAM) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5646176A (en) * | 1992-12-24 | 1997-07-08 | Bristol-Myers Squibb Company | Phosphonooxymethyl ethers of taxane derivatives |
| US5684175A (en) * | 1993-02-05 | 1997-11-04 | Napro Biotherapeutics, Inc. | C-2' hydroxyl-benzyl protected, N-carbamate protected (2R, 3S)- 3-phenylisoserine and production process therefor |
| EP1260507A1 (en) * | 1993-02-05 | 2002-11-27 | Bryn Mawr College | Synthesis of taxol, analogs and intermediates with variable A-nng side chains |
| US5580899A (en) * | 1995-01-09 | 1996-12-03 | The Liposome Company, Inc. | Hydrophobic taxane derivatives |
| US5675025A (en) * | 1995-06-07 | 1997-10-07 | Napro Biotherapeutics, Inc. | Paclitaxel synthesis from precursor compounds and methods of producing the same |
| US6051600A (en) * | 1995-09-12 | 2000-04-18 | Mayhew; Eric | Liposomal hydrolysis-promoting hydrophobic taxane derivatives |
| US6107332A (en) | 1995-09-12 | 2000-08-22 | The Liposome Company, Inc. | Hydrolysis-promoting hydrophobic taxane derivatives |
| US5688977A (en) * | 1996-02-29 | 1997-11-18 | Napro Biotherapeutics, Inc. | Method for docetaxel synthesis |
| US6107497A (en) * | 1996-02-29 | 2000-08-22 | Napro Biotherapeutics, Inc. | Intermediate for use in docetaxel synthesis and production method therefor |
| US5750737A (en) * | 1996-09-25 | 1998-05-12 | Sisti; Nicholas J. | Method for paclitaxel synthesis |
| US6025516A (en) * | 1998-10-14 | 2000-02-15 | Chiragene, Inc. | Resolution of 2-hydroxy-3-amino-3-phenylpropionamide and its conversion to C-13 sidechain of taxanes |
| US6452025B1 (en) | 2001-04-25 | 2002-09-17 | Napro Biotherapeutics, Inc. | Three-step conversion of protected taxane ester to paclitaxel |
| DE60309847T2 (de) * | 2002-02-27 | 2007-10-18 | Ferring B.V. | Zwischenprodukte und verfahren zur herstellung von heptapeptid-oxytocinanaloga |
| AU2013274101B2 (en) | 2012-06-15 | 2017-09-07 | The Brigham And Women's Hospital, Inc. | Compositions for treating cancer and methods for making the same |
| US10426753B2 (en) | 2014-04-03 | 2019-10-01 | Invictus Oncology Pvt. Ltd. | Supramolecular combinatorial therapeutics |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2629819B1 (fr) * | 1988-04-06 | 1990-11-16 | Rhone Poulenc Sante | Procede de preparation de derives de la baccatine iii et de la desacetyl-10 baccatine iii |
| FR2629818B1 (fr) * | 1988-04-06 | 1990-11-16 | Centre Nat Rech Scient | Procede de preparation du taxol |
| FR2662441B1 (fr) * | 1990-05-22 | 1992-10-23 | Rhone Poulenc Sante | Procede de preparation enantioselective de derives de la phenylisoserine. |
| FR2662440B1 (fr) * | 1990-05-22 | 1992-07-31 | Rhone Poulenc Sante | Procede de preparation stereoselective de derives de la phenylisoserine. |
-
1991
- 1991-08-19 FR FR919110398A patent/FR2680506B1/fr not_active Expired - Fee Related
-
1992
- 1992-08-11 MX MX9204635A patent/MX9204635A/es unknown
- 1992-08-17 HU HU9400478A patent/HUT68255A/hu unknown
- 1992-08-17 FI FI940775A patent/FI940775L/fi not_active Application Discontinuation
- 1992-08-17 CA CA002113827A patent/CA2113827A1/fr not_active Abandoned
- 1992-08-17 TW TW081106473A patent/TW222620B/zh active
- 1992-08-17 AU AU24904/92A patent/AU2490492A/en not_active Abandoned
- 1992-08-17 WO PCT/FR1992/000795 patent/WO1993004038A1/fr not_active Ceased
- 1992-08-17 EP EP92918283A patent/EP0599973A1/fr not_active Ceased
- 1992-08-17 CZ CS94354A patent/CZ35494A3/cs unknown
- 1992-08-17 NZ NZ243972A patent/NZ243972A/en unknown
- 1992-08-17 SK SK190-94A patent/SK19094A3/sk unknown
- 1992-08-17 EP EP92402293A patent/EP0528729A1/fr active Pending
- 1992-08-17 JP JP5504146A patent/JPH06510033A/ja active Pending
- 1992-08-17 ZA ZA926189A patent/ZA926189B/xx unknown
- 1992-08-19 YU YU78092A patent/YU78092A/sh unknown
-
1994
- 1994-01-04 NO NO940027A patent/NO940027D0/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO1993004038A1 (fr) | 1993-03-04 |
| FR2680506B1 (fr) | 1994-09-02 |
| NO940027L (no) | 1994-01-04 |
| CA2113827A1 (fr) | 1993-03-04 |
| TW222620B (OSRAM) | 1994-04-21 |
| MX9204635A (es) | 1993-02-01 |
| FR2680506A1 (fr) | 1993-02-26 |
| ZA926189B (en) | 1993-03-01 |
| HU9400478D0 (en) | 1994-06-28 |
| YU78092A (sh) | 1995-10-03 |
| AU2490492A (en) | 1993-03-16 |
| CZ35494A3 (en) | 1994-07-13 |
| SK19094A3 (en) | 1994-09-07 |
| FI940775A0 (fi) | 1994-02-18 |
| HUT68255A (en) | 1995-06-28 |
| EP0599973A1 (fr) | 1994-06-08 |
| NZ243972A (en) | 1994-11-25 |
| FI940775A7 (fi) | 1994-02-18 |
| EP0528729A1 (fr) | 1993-02-24 |
| NO940027D0 (no) | 1994-01-04 |
| JPH06510033A (ja) | 1994-11-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD | Application lapsed |