FI940591A7 - Uudet 3-(substituoitu tetratsolyyli)-4-okso-4H-pyrido/1,2-a/pyrimidiinit, niiden suolat, niitä sisältävät farmaseuttiset koostumukset ja niiden valmistusmenetelmä - Google Patents

Uudet 3-(substituoitu tetratsolyyli)-4-okso-4H-pyrido/1,2-a/pyrimidiinit, niiden suolat, niitä sisältävät farmaseuttiset koostumukset ja niiden valmistusmenetelmä Download PDF

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Publication number
FI940591A7
FI940591A7 FI940591A FI940591A FI940591A7 FI 940591 A7 FI940591 A7 FI 940591A7 FI 940591 A FI940591 A FI 940591A FI 940591 A FI940591 A FI 940591A FI 940591 A7 FI940591 A7 FI 940591A7
Authority
FI
Finland
Prior art keywords
pyrido
pyrimidines
oxo
salts
novel
Prior art date
Application number
FI940591A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI940591A0 (fi
Inventor
Istvan Hermecz
Jozsef Knoll
Judit Sipos
Klara Gyires
Agnes Horvath
Lelle Vasvari
Laszlo Tardos
Maria Balogh
Zoltan Kapui
Ilona Papp
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Publication of FI940591A0 publication Critical patent/FI940591A0/fi
Publication of FI940591A7 publication Critical patent/FI940591A7/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI940591A 1990-09-25 1994-02-09 Uudet 3-(substituoitu tetratsolyyli)-4-okso-4H-pyrido/1,2-a/pyrimidiinit, niiden suolat, niitä sisältävät farmaseuttiset koostumukset ja niiden valmistusmenetelmä FI940591A7 (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU620590A HU209793B (en) 1990-09-25 1990-09-25 Process for the production of pyrido[1,2-a]pyrimidine-derivatives and pharmaceutical compositions containing the same
PCT/HU1992/000031 WO1993004065A1 (en) 1990-09-25 1992-08-13 NEW 3-(SUBSTITUTED TETRAZOLYL)-4-OXO-4H-PYRIDO-[1,2-a]PYRIMIDINES, SALTS THEREOF, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR PREPARING SAME

Publications (2)

Publication Number Publication Date
FI940591A0 FI940591A0 (fi) 1994-02-09
FI940591A7 true FI940591A7 (fi) 1994-02-09

Family

ID=10971360

Family Applications (1)

Application Number Title Priority Date Filing Date
FI940591A FI940591A7 (fi) 1990-09-25 1994-02-09 Uudet 3-(substituoitu tetratsolyyli)-4-okso-4H-pyrido/1,2-a/pyrimidiinit, niiden suolat, niitä sisältävät farmaseuttiset koostumukset ja niiden valmistusmenetelmä

Country Status (19)

Country Link
US (1) US5475000A (enExample)
EP (1) EP0641340A1 (enExample)
JP (1) JPH06509800A (enExample)
CN (1) CN1071925A (enExample)
AU (1) AU663886B2 (enExample)
BG (1) BG98448A (enExample)
CA (1) CA2114145A1 (enExample)
CZ (1) CZ27694A3 (enExample)
EE (1) EE9400115A (enExample)
FI (1) FI940591A7 (enExample)
HU (1) HU209793B (enExample)
IL (1) IL102788A (enExample)
MX (1) MX9204659A (enExample)
PT (1) PT100774A (enExample)
SI (1) SI9200172A (enExample)
SK (1) SK16594A3 (enExample)
TW (1) TW222632B (enExample)
WO (1) WO1993004065A1 (enExample)
YU (1) YU76092A (enExample)

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3055911A (en) * 1958-04-29 1962-09-25 William G Finnegan Substituted tetrazoles
US4122274A (en) * 1977-05-25 1978-10-24 Bristol-Myers Company 3-Tetrazolo-5,6,7,8-substituted-pyrido[1,2-a]pyrimidin-4-ones
JPS5536447A (en) * 1978-09-07 1980-03-14 Otsuka Pharmaceut Co Ltd Butyramide derivative
US4432986A (en) * 1979-06-18 1984-02-21 Riker Laboratories, Inc. Tetrazoles bonded to certain polycyclic aromatic systems and anti-allergic use thereof
US4474792A (en) * 1979-06-18 1984-10-02 Riker Laboratories, Inc. N-Tetrazolyl benzamides and anti-allergic use thereof
FI73423C (fi) * 1980-02-29 1987-10-09 Otsuka Pharma Co Ltd Foerfarande foer framstaellning av farmakologiskt verksamma tetrazolderivat.
US4457932A (en) * 1983-07-22 1984-07-03 Bristol-Myers Company Anti-ulcer agents
FR2549831A1 (fr) * 1983-07-27 1985-02-01 Rhone Poulenc Agrochimie Nouveaux derives d'acides aryloxybenzoiques, et leur utilisation comme herbicides
US4845227A (en) * 1984-06-18 1989-07-04 Eli Lilly And Company Aromatase inhibitors from azoles
US5237070A (en) * 1985-07-22 1993-08-17 Riker Laboratories, Inc. Substituted DI-t-butylphenols
US5049572A (en) * 1987-04-06 1991-09-17 Riker Laboratories, Inc. Substituted di-t-butylphenols and anti-allergic use thereof
JP2668259B2 (ja) * 1988-02-18 1997-10-27 塩野義製薬株式会社 複素環化合物および抗潰瘍剤
HUT64064A (en) * 1992-02-13 1993-11-29 Chinoin Gyogyszer Es Vegyeszet Process for producing puyrido/1,2-a/pyrimidine derivatives and pharmaceutical compositions comprising same as active ingredient

Also Published As

Publication number Publication date
HUT64954A (en) 1994-03-28
TW222632B (enExample) 1994-04-21
JPH06509800A (ja) 1994-11-02
BG98448A (bg) 1994-11-15
EE9400115A (et) 1995-12-15
IL102788A (en) 1996-03-31
SK16594A3 (en) 1994-08-10
SI9200172A (en) 1993-03-31
HU906205D0 (en) 1991-03-28
YU76092A (sr) 1996-01-09
CN1071925A (zh) 1993-05-12
FI940591A0 (fi) 1994-02-09
MX9204659A (es) 1993-12-31
AU663886B2 (en) 1995-10-26
EP0641340A1 (en) 1995-03-08
CZ27694A3 (en) 1994-08-17
CA2114145A1 (en) 1993-03-04
US5475000A (en) 1995-12-12
WO1993004065A1 (en) 1993-03-04
AU2462892A (en) 1993-03-16
PT100774A (pt) 1993-10-29
HU209793B (en) 1994-11-28

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