FI932052A - Fenylsulfonamidendotelinantagonister - Google Patents

Fenylsulfonamidendotelinantagonister Download PDF

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Publication number
FI932052A
FI932052A FI932052A FI932052A FI932052A FI 932052 A FI932052 A FI 932052A FI 932052 A FI932052 A FI 932052A FI 932052 A FI932052 A FI 932052A FI 932052 A FI932052 A FI 932052A
Authority
FI
Finland
Prior art keywords
hydrogen
symbols
fenylsulfonamidendotelinantagonister
cycloalkenylalkyl
co2r
Prior art date
Application number
FI932052A
Other languages
English (en)
Other versions
FI112655B (fi
FI932052A0 (fi
Inventor
Natesan Murugesan
John T Hunt
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of FI932052A0 publication Critical patent/FI932052A0/fi
Publication of FI932052A publication Critical patent/FI932052A/fi
Application granted granted Critical
Publication of FI112655B publication Critical patent/FI112655B/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D261/14—Nitrogen atoms
    • C07D261/16—Benzene-sulfonamido isoxazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D261/18—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems
FI932052A 1992-05-06 1993-05-06 Menetelmä uusien terapeuttisesti käyttökelpoisten fenyylisulfonamidijohdannaisten valmistamiseksi FI112655B (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US87900092A 1992-05-06 1992-05-06
US87900092 1992-05-06

Publications (3)

Publication Number Publication Date
FI932052A0 FI932052A0 (fi) 1993-05-06
FI932052A true FI932052A (fi) 1993-11-07
FI112655B FI112655B (fi) 2003-12-31

Family

ID=25373236

Family Applications (1)

Application Number Title Priority Date Filing Date
FI932052A FI112655B (fi) 1992-05-06 1993-05-06 Menetelmä uusien terapeuttisesti käyttökelpoisten fenyylisulfonamidijohdannaisten valmistamiseksi

Country Status (22)

Country Link
EP (1) EP0569193B1 (fi)
JP (1) JP3286391B2 (fi)
KR (1) KR100277454B1 (fi)
CN (1) CN1066441C (fi)
AT (1) ATE149155T1 (fi)
AU (1) AU659545B2 (fi)
CA (1) CA2095174A1 (fi)
CY (1) CY2016A (fi)
DE (1) DE69308229T2 (fi)
DK (1) DK0569193T3 (fi)
ES (1) ES2100459T3 (fi)
FI (1) FI112655B (fi)
GR (1) GR3023421T3 (fi)
HK (1) HK98197A (fi)
HU (1) HU218938B (fi)
IL (1) IL105481A (fi)
MX (1) MX9302618A (fi)
NO (1) NO303065B1 (fi)
NZ (1) NZ247440A (fi)
PL (1) PL178165B1 (fi)
RU (1) RU2133742C1 (fi)
ZA (1) ZA932914B (fi)

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Also Published As

Publication number Publication date
KR930023337A (ko) 1993-12-18
EP0569193B1 (en) 1997-02-26
ATE149155T1 (de) 1997-03-15
CN1084515A (zh) 1994-03-30
NO931638D0 (no) 1993-05-05
ES2100459T3 (es) 1997-06-16
HU9301305D0 (en) 1993-09-28
HK98197A (en) 1997-08-08
ZA932914B (en) 1993-11-12
PL298828A1 (en) 1993-12-27
HU218938B (hu) 2001-01-29
FI112655B (fi) 2003-12-31
JP3286391B2 (ja) 2002-05-27
DE69308229T2 (de) 1997-07-17
DE69308229D1 (de) 1997-04-03
KR100277454B1 (ko) 2001-01-15
IL105481A0 (en) 1993-08-18
CY2016A (en) 1998-02-20
AU3838293A (en) 1993-11-11
MX9302618A (es) 1994-05-31
PL178165B1 (pl) 2000-03-31
RU2133742C1 (ru) 1999-07-27
NO303065B1 (no) 1998-05-25
EP0569193A1 (en) 1993-11-10
CN1066441C (zh) 2001-05-30
NO931638L (no) 1993-11-08
DK0569193T3 (fi) 1997-03-17
NZ247440A (en) 1995-04-27
CA2095174A1 (en) 1993-11-07
HUT65751A (en) 1994-07-28
GR3023421T3 (en) 1997-08-29
FI932052A0 (fi) 1993-05-06
JPH0649046A (ja) 1994-02-22
IL105481A (en) 1996-12-05
AU659545B2 (en) 1995-05-18

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