FI914007L - 4-substituerade dihydropyrido (4,3-d) pyrimidiner som smaertslindrande och lokala inflammationshaemmande medel vid vaord av hudsjukdomar. - Google Patents

4-substituerade dihydropyrido (4,3-d) pyrimidiner som smaertslindrande och lokala inflammationshaemmande medel vid vaord av hudsjukdomar. Download PDF

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Publication number
FI914007L
FI914007L FI914007A FI914007A FI914007L FI 914007 L FI914007 L FI 914007L FI 914007 A FI914007 A FI 914007A FI 914007 A FI914007 A FI 914007A FI 914007 L FI914007 L FI 914007L
Authority
FI
Finland
Prior art keywords
vaord
smaertslindrande
lokala
inflammationshaemmande
hudsjukdomar
Prior art date
Application number
FI914007A
Other languages
English (en)
Finnish (fi)
Other versions
FI914007A7 (fi
FI914007A0 (fi
Inventor
Richard Charles Effland
Joseph Thomas Klein
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of FI914007A0 publication Critical patent/FI914007A0/fi
Publication of FI914007A7 publication Critical patent/FI914007A7/fi
Publication of FI914007L publication Critical patent/FI914007L/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/06Peri-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/485Morphinan derivatives, e.g. morphine, codeine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Emergency Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
FI914007A 1990-08-27 1991-08-23 4-substituerade dihydropyrido (4,3-d) pyrimidiner som smaertslindrande och lokala inflammationshaemmande medel vid vaord av hudsjukdomar. FI914007L (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/573,414 US5059602A (en) 1990-08-27 1990-08-27 4-substituted dihydropyrido(4,3-d)pyrimidines as analgesics and topical antiinflammatory agents for the treatment of skin disorders

Publications (3)

Publication Number Publication Date
FI914007A0 FI914007A0 (fi) 1991-08-23
FI914007A7 FI914007A7 (fi) 1992-02-28
FI914007L true FI914007L (fi) 1992-02-28

Family

ID=24291905

Family Applications (1)

Application Number Title Priority Date Filing Date
FI914007A FI914007L (fi) 1990-08-27 1991-08-23 4-substituerade dihydropyrido (4,3-d) pyrimidiner som smaertslindrande och lokala inflammationshaemmande medel vid vaord av hudsjukdomar.

Country Status (22)

Country Link
US (1) US5059602A (cs)
EP (1) EP0480155B1 (cs)
JP (1) JP3083180B2 (cs)
KR (1) KR100218562B1 (cs)
AT (1) ATE133670T1 (cs)
AU (1) AU635150B2 (cs)
CA (1) CA2049850C (cs)
CZ (1) CZ280569B6 (cs)
DE (1) DE69116788T2 (cs)
DK (1) DK0480155T3 (cs)
ES (1) ES2082894T3 (cs)
FI (1) FI914007L (cs)
GR (1) GR3019085T3 (cs)
HU (1) HUT59923A (cs)
IE (1) IE72086B1 (cs)
IL (1) IL99305A (cs)
NO (1) NO913331L (cs)
NZ (1) NZ239516A (cs)
PT (1) PT98773B (cs)
SG (1) SG48250A1 (cs)
YU (1) YU144391A (cs)
ZA (1) ZA916738B (cs)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5095019A (en) * 1990-08-27 1992-03-10 Hoechst-Roussel Pharmaceuticals Inc. 4-substituted dihydropyrido(4,3-D)pyrimidines as analgesics and topical antiinflammatory agents for the treatment of skin disorders
US6008361A (en) * 1996-04-09 1999-12-28 Pfizer Inc. Substituted pyridines
US6031105A (en) * 1996-04-09 2000-02-29 Pfizer Inc Substituted pyridines
EP1289415A4 (en) 2000-05-18 2008-12-03 Nuvasive Inc TISSUE DISTRACTION AND APPLICATIONS IN MEDICAL PROCEDURES
CA2450073C (en) 2001-07-25 2017-08-29 Biomarin Pharmaceutical Inc. Compositions and methods for modulating blood-brain barrier transport
EP2671508B1 (en) 2005-04-28 2020-09-16 Proteus Digital Health, Inc. Pharma-informatics system
KR20080014812A (ko) * 2005-05-03 2008-02-14 랜박시 래보러터리스 리미티드 항균제
JP2009533315A (ja) * 2006-04-10 2009-09-17 ランバクシー ラボラトリーズ リミテッド 抗菌剤
WO2008036682A2 (en) 2006-09-18 2008-03-27 Raptor Pharmaceutical Inc. Treatment of liver disorders by administration of receptor-associated protein (rap)-conjugates
CN102316902B (zh) 2009-02-20 2014-09-24 to-BBB控股股份有限公司 基于谷胱甘肽的药物递送系统
IL255113B (en) 2009-05-06 2022-09-01 Laboratory Skin Care Inc Dermal delivery compositions comprising active agent-calcium phosphate particle complexes and methods of using the same
US20120077778A1 (en) 2010-09-29 2012-03-29 Andrea Bourdelais Ladder-Frame Polyether Conjugates

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1197466B (de) * 1962-03-22 1965-07-29 Thomae Gmbh Dr K Verfahren zur Herstellung von neuen 5, 6, 7, 8-Tetrahydropyrido-[4, 3-d]pyrimidinen
US3635973A (en) * 1969-11-20 1972-01-18 Sherwin Williams Co Method of preparing 3-substituted pyridopyrimidinediones and lumazines
US3962264A (en) * 1972-09-27 1976-06-08 Pfizer Inc. Process for making 2-amino nicotinonitrile
DE3438351A1 (de) * 1984-10-19 1986-04-24 Gödecke AG, 1000 Berlin 4-alkoxy-pyrido(2,3-d)pyrimidin-derivate, verfahren zu deren herstellung und deren verwendung
DE3502590A1 (de) * 1985-01-26 1986-07-31 Gödecke AG, 1000 Berlin 5-alkoxy-pyrido(4,3-d)pyrimidin-derivate, verfahren zu deren herstellung und deren verwendung
DE3502742A1 (de) * 1985-01-28 1986-07-31 Gödecke AG, 1000 Berlin 5-oxo-pyrido(4,3-d)pyrimidin-derivate, verfahren zu deren herstellung und deren verwendung

Also Published As

Publication number Publication date
IL99305A (en) 1997-02-18
ATE133670T1 (de) 1996-02-15
KR920004387A (ko) 1992-03-27
DK0480155T3 (da) 1996-06-10
YU144391A (sh) 1995-03-27
FI914007A7 (fi) 1992-02-28
NO913331D0 (no) 1991-08-26
KR100218562B1 (ko) 1999-09-01
SG48250A1 (en) 1998-04-17
IE913010A1 (en) 1992-03-11
DE69116788T2 (de) 1996-07-18
HU912786D0 (en) 1992-01-28
GR3019085T3 (en) 1996-05-31
HUT59923A (en) 1992-07-28
NZ239516A (en) 1994-04-27
AU8271991A (en) 1992-03-05
CS262491A3 (en) 1992-06-17
NO913331L (no) 1992-02-28
EP0480155A2 (en) 1992-04-15
CZ280569B6 (cs) 1996-02-14
EP0480155B1 (en) 1996-01-31
JPH04230684A (ja) 1992-08-19
DE69116788D1 (de) 1996-03-14
US5059602A (en) 1991-10-22
AU635150B2 (en) 1993-03-11
EP0480155A3 (en) 1992-04-29
IL99305A0 (en) 1992-07-15
ZA916738B (en) 1992-04-29
CA2049850A1 (en) 1992-02-28
PT98773A (pt) 1992-07-31
IE72086B1 (en) 1997-03-12
CA2049850C (en) 2002-03-05
ES2082894T3 (es) 1996-04-01
PT98773B (pt) 1999-01-29
JP3083180B2 (ja) 2000-09-04
FI914007A0 (fi) 1991-08-23

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