FI914007L - 4-substituerade dihydropyrido (4,3-d) pyrimidiner som smaertslindrande och lokala inflammationshaemmande medel vid vaord av hudsjukdomar. - Google Patents

4-substituerade dihydropyrido (4,3-d) pyrimidiner som smaertslindrande och lokala inflammationshaemmande medel vid vaord av hudsjukdomar. Download PDF

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Publication number
FI914007L
FI914007L FI914007A FI914007A FI914007L FI 914007 L FI914007 L FI 914007L FI 914007 A FI914007 A FI 914007A FI 914007 A FI914007 A FI 914007A FI 914007 L FI914007 L FI 914007L
Authority
FI
Finland
Prior art keywords
vaord
smaertslindrande
lokala
inflammationshaemmande
hudsjukdomar
Prior art date
Application number
FI914007A
Other languages
English (en)
Finnish (fi)
Other versions
FI914007A7 (fi
FI914007A0 (fi
Inventor
Richard Charles Effland
Joseph Thomas Klein
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of FI914007A0 publication Critical patent/FI914007A0/fi
Publication of FI914007A7 publication Critical patent/FI914007A7/fi
Publication of FI914007L publication Critical patent/FI914007L/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/06Peri-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/485Morphinan derivatives, e.g. morphine, codeine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Neurosurgery (AREA)
  • Dermatology (AREA)
  • Emergency Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
FI914007A 1990-08-27 1991-08-23 4-substituerade dihydropyrido (4,3-d) pyrimidiner som smaertslindrande och lokala inflammationshaemmande medel vid vaord av hudsjukdomar. FI914007L (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/573,414 US5059602A (en) 1990-08-27 1990-08-27 4-substituted dihydropyrido(4,3-d)pyrimidines as analgesics and topical antiinflammatory agents for the treatment of skin disorders

Publications (3)

Publication Number Publication Date
FI914007A0 FI914007A0 (fi) 1991-08-23
FI914007A7 FI914007A7 (fi) 1992-02-28
FI914007L true FI914007L (fi) 1992-02-28

Family

ID=24291905

Family Applications (1)

Application Number Title Priority Date Filing Date
FI914007A FI914007L (fi) 1990-08-27 1991-08-23 4-substituerade dihydropyrido (4,3-d) pyrimidiner som smaertslindrande och lokala inflammationshaemmande medel vid vaord av hudsjukdomar.

Country Status (22)

Country Link
US (1) US5059602A (cs)
EP (1) EP0480155B1 (cs)
JP (1) JP3083180B2 (cs)
KR (1) KR100218562B1 (cs)
AT (1) ATE133670T1 (cs)
AU (1) AU635150B2 (cs)
CA (1) CA2049850C (cs)
CZ (1) CZ280569B6 (cs)
DE (1) DE69116788T2 (cs)
DK (1) DK0480155T3 (cs)
ES (1) ES2082894T3 (cs)
FI (1) FI914007L (cs)
GR (1) GR3019085T3 (cs)
HU (1) HUT59923A (cs)
IE (1) IE72086B1 (cs)
IL (1) IL99305A (cs)
NO (1) NO913331L (cs)
NZ (1) NZ239516A (cs)
PT (1) PT98773B (cs)
SG (1) SG48250A1 (cs)
YU (1) YU144391A (cs)
ZA (1) ZA916738B (cs)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5095019A (en) * 1990-08-27 1992-03-10 Hoechst-Roussel Pharmaceuticals Inc. 4-substituted dihydropyrido(4,3-D)pyrimidines as analgesics and topical antiinflammatory agents for the treatment of skin disorders
US6031105A (en) * 1996-04-09 2000-02-29 Pfizer Inc Substituted pyridines
US6008361A (en) * 1996-04-09 1999-12-28 Pfizer Inc. Substituted pyridines
US6760616B2 (en) 2000-05-18 2004-07-06 Nu Vasive, Inc. Tissue discrimination and applications in medical procedures
US20030129186A1 (en) 2001-07-25 2003-07-10 Biomarin Pharmaceutical Inc. Compositions and methods for modulating blood-brain barrier transport
CN101287411B (zh) 2005-04-28 2013-03-06 普罗秋斯生物医学公司 药物信息系统及其用途
WO2006117762A2 (en) 2005-05-03 2006-11-09 Ranbaxy Laboratories Limited Antimicrobial agents
JP2009533315A (ja) * 2006-04-10 2009-09-17 ランバクシー ラボラトリーズ リミテッド 抗菌剤
CN101594878A (zh) 2006-09-18 2009-12-02 雷普特药品公司 通过给予受体相关蛋白(rap)-缀合物对肝病症的治疗
ES2728225T3 (es) 2009-02-20 2019-10-23 2 Bbb Medicines B V Sistema de administración de fármacos a base de glutatión
KR101909711B1 (ko) 2009-05-06 2018-12-19 라보라토리 스킨 케어, 인크. 활성제-칼슘 포스페이트 입자 복합체를 포함하는 피부 전달 조성물 및 이들을 이용하는 방법
US20120077778A1 (en) 2010-09-29 2012-03-29 Andrea Bourdelais Ladder-Frame Polyether Conjugates

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1197466B (de) * 1962-03-22 1965-07-29 Thomae Gmbh Dr K Verfahren zur Herstellung von neuen 5, 6, 7, 8-Tetrahydropyrido-[4, 3-d]pyrimidinen
US3635973A (en) * 1969-11-20 1972-01-18 Sherwin Williams Co Method of preparing 3-substituted pyridopyrimidinediones and lumazines
US3962264A (en) * 1972-09-27 1976-06-08 Pfizer Inc. Process for making 2-amino nicotinonitrile
DE3438351A1 (de) * 1984-10-19 1986-04-24 Gödecke AG, 1000 Berlin 4-alkoxy-pyrido(2,3-d)pyrimidin-derivate, verfahren zu deren herstellung und deren verwendung
DE3502590A1 (de) * 1985-01-26 1986-07-31 Gödecke AG, 1000 Berlin 5-alkoxy-pyrido(4,3-d)pyrimidin-derivate, verfahren zu deren herstellung und deren verwendung
DE3502742A1 (de) * 1985-01-28 1986-07-31 Gödecke AG, 1000 Berlin 5-oxo-pyrido(4,3-d)pyrimidin-derivate, verfahren zu deren herstellung und deren verwendung

Also Published As

Publication number Publication date
HU912786D0 (en) 1992-01-28
PT98773B (pt) 1999-01-29
DE69116788D1 (de) 1996-03-14
ZA916738B (en) 1992-04-29
IL99305A (en) 1997-02-18
CA2049850C (en) 2002-03-05
IL99305A0 (en) 1992-07-15
CA2049850A1 (en) 1992-02-28
IE72086B1 (en) 1997-03-12
HUT59923A (en) 1992-07-28
JP3083180B2 (ja) 2000-09-04
CS262491A3 (en) 1992-06-17
US5059602A (en) 1991-10-22
AU8271991A (en) 1992-03-05
NO913331L (no) 1992-02-28
NO913331D0 (no) 1991-08-26
FI914007A7 (fi) 1992-02-28
CZ280569B6 (cs) 1996-02-14
YU144391A (sh) 1995-03-27
PT98773A (pt) 1992-07-31
JPH04230684A (ja) 1992-08-19
ES2082894T3 (es) 1996-04-01
FI914007A0 (fi) 1991-08-23
IE913010A1 (en) 1992-03-11
DE69116788T2 (de) 1996-07-18
KR100218562B1 (ko) 1999-09-01
AU635150B2 (en) 1993-03-11
EP0480155B1 (en) 1996-01-31
EP0480155A3 (en) 1992-04-29
KR920004387A (ko) 1992-03-27
SG48250A1 (en) 1998-04-17
GR3019085T3 (en) 1996-05-31
ATE133670T1 (de) 1996-02-15
NZ239516A (en) 1994-04-27
EP0480155A2 (en) 1992-04-15
DK0480155T3 (da) 1996-06-10

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