FI902763A0 - Heterocyklisk foerening med antagonistisk aktivitet mot serotonin 2-receptor. - Google Patents

Heterocyklisk foerening med antagonistisk aktivitet mot serotonin 2-receptor.

Info

Publication number
FI902763A0
FI902763A0 FI902763A FI902763A FI902763A0 FI 902763 A0 FI902763 A0 FI 902763A0 FI 902763 A FI902763 A FI 902763A FI 902763 A FI902763 A FI 902763A FI 902763 A0 FI902763 A0 FI 902763A0
Authority
FI
Finland
Prior art keywords
antagonistic activity
heterocyclic
receptor
serotonin
foerening
Prior art date
Application number
FI902763A
Other languages
English (en)
Inventor
Yoshifumi Watanabe
Hiroyuki Usui
Toshiro Shibano
Tsuyoshi Tanaka
Yoshiyuki Morishima
Original Assignee
Daiichi Seiyaku Co
Yasuoka Megumi
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP1310346A external-priority patent/JPH03170431A/ja
Application filed by Daiichi Seiyaku Co, Yasuoka Megumi filed Critical Daiichi Seiyaku Co
Publication of FI902763A0 publication Critical patent/FI902763A0/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI902763A 1989-06-05 1990-06-04 Heterocyklisk foerening med antagonistisk aktivitet mot serotonin 2-receptor. FI902763A0 (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP14239789 1989-06-05
JP18861789 1989-07-20
JP20203989 1989-08-03
JP1310346A JPH03170431A (ja) 1989-11-29 1989-11-29 心臓疾患治療剤

Publications (1)

Publication Number Publication Date
FI902763A0 true FI902763A0 (fi) 1990-06-04

Family

ID=27472451

Family Applications (1)

Application Number Title Priority Date Filing Date
FI902763A FI902763A0 (fi) 1989-06-05 1990-06-04 Heterocyklisk foerening med antagonistisk aktivitet mot serotonin 2-receptor.

Country Status (17)

Country Link
US (1) US5232924A (fi)
EP (1) EP0401707B1 (fi)
KR (1) KR910000755A (fi)
CN (1) CN1049161A (fi)
AT (1) ATE111911T1 (fi)
AU (1) AU628579B2 (fi)
CA (1) CA2018220A1 (fi)
DE (1) DE69012653T2 (fi)
DK (1) DK0401707T3 (fi)
ES (1) ES2064530T3 (fi)
FI (1) FI902763A0 (fi)
HU (1) HUT54365A (fi)
IL (1) IL94592A (fi)
NO (1) NO174712C (fi)
NZ (1) NZ233917A (fi)
PT (1) PT94270A (fi)
YU (1) YU108790A (fi)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5552397A (en) * 1992-05-18 1996-09-03 E. R. Squibb & Sons, Inc. Substituted azepinone dual inhibitors of angiotensin converting enzyme and neutral exdopeptidase
CA2108245A1 (en) * 1992-11-04 1994-05-05 Gary J. Grover Method for treating myocardial ischemia employing serotonin receptor antagonists
TW200608978A (en) * 2004-05-28 2006-03-16 Speedel Experimenta Ag Organic compounds
US9150546B2 (en) 2009-02-13 2015-10-06 Shionogi & Co., Ltd. Triazine derivative and pharmaceutical composition comprising the same
CN103153968B (zh) 2010-08-10 2016-02-03 盐野义制药株式会社 三唑衍生物及含有其的具有镇痛作用的药物组合物
JP6075621B2 (ja) 2010-08-10 2017-02-08 塩野義製薬株式会社 新規複素環誘導体およびそれらを含有する医薬組成物
WO2013074390A1 (en) * 2011-11-14 2013-05-23 Merck Sharp & Dohme Corp. Triazolopyridinone pde10 inhibitors
WO2013118855A1 (ja) 2012-02-09 2013-08-15 塩野義製薬株式会社 複素環および炭素環誘導体
TWI637949B (zh) 2013-06-14 2018-10-11 塩野義製藥股份有限公司 胺基三衍生物及含有其等之醫藥組合物
CN113185521A (zh) * 2021-05-08 2021-07-30 新乡市润宇新材料科技有限公司 一种环丙基开环制备四氢吡咯并[1,2-a]1,3,5-三嗪-4-酮类化合物的方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH498132A (de) * 1968-05-06 1970-10-31 Agripat Sa Verfahren zur Herstellung neuer Pyrido (1,2-a)-s-triazindione
GB1328205A (en) * 1970-10-13 1973-08-30 Lilly Industries Ltd Oxazolo-triazines
US4340597A (en) * 1981-04-13 1982-07-20 Schering Corporation 1-Substituted-4-aryl-1,2,5,6-tetrahydro and hexahydropyridines
DE3173762D1 (de) * 1981-06-15 1986-03-27 Nippon Soda Co Thiazolinotriazine derivatives
DE3126837A1 (de) * 1981-07-08 1983-01-27 Hoechst Ag, 6000 Frankfurt Triazino-(2,1-a)isochinolinderivate

Also Published As

Publication number Publication date
EP0401707B1 (en) 1994-09-21
US5232924A (en) 1993-08-03
HU903489D0 (en) 1990-10-28
DE69012653T2 (de) 1995-02-09
PT94270A (pt) 1991-02-08
DK0401707T3 (da) 1994-10-17
NO902439L (no) 1990-12-06
NO902439D0 (no) 1990-06-01
ATE111911T1 (de) 1994-10-15
CN1049161A (zh) 1991-02-13
AU628579B2 (en) 1992-09-17
CA2018220A1 (en) 1990-12-05
AU5629590A (en) 1990-12-06
NO174712C (no) 1994-06-22
IL94592A (en) 1994-07-31
EP0401707A1 (en) 1990-12-12
HUT54365A (en) 1991-02-28
YU108790A (en) 1991-10-31
IL94592A0 (en) 1991-04-15
DE69012653D1 (de) 1994-10-27
KR910000755A (ko) 1991-01-30
ES2064530T3 (es) 1995-02-01
NZ233917A (en) 1991-04-26
NO174712B (no) 1994-03-14

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Legal Events

Date Code Title Description
FD Application lapsed
MM Patent lapsed

Owner name: DAIICHI PHARMACEUTICAL CO., LTD.