FI885622A0 - Menetelmä 7 -/(Z)-2-(5-amino-1,2,4-tiadiatsol-3-yyli)-2-metoksi-iminoasetamido/-3-(1-imidatso/1,2-b/-pyridatsinium)metyyli-3-kefeemi-4-karboksylaatti-hydrokloridin kiteiden valmistamiseksi - Google Patents

Menetelmä 7 -/(Z)-2-(5-amino-1,2,4-tiadiatsol-3-yyli)-2-metoksi-iminoasetamido/-3-(1-imidatso/1,2-b/-pyridatsinium)metyyli-3-kefeemi-4-karboksylaatti-hydrokloridin kiteiden valmistamiseksi

Info

Publication number
FI885622A0
FI885622A0 FI885622A FI885622A FI885622A0 FI 885622 A0 FI885622 A0 FI 885622A0 FI 885622 A FI885622 A FI 885622A FI 885622 A FI885622 A FI 885622A FI 885622 A0 FI885622 A0 FI 885622A0
Authority
FI
Finland
Prior art keywords
methoxyiminoacetamido
pyridazinium
cephem
thiadiazol
imidazo
Prior art date
Application number
FI885622A
Other languages
English (en)
Swedish (sv)
Other versions
FI90873C (fi
FI90873B (fi
FI885622A (fi
Inventor
Yoshiharu Maeda
Yukio Mizuno
Akira Nakatani
Mitsuhisa Yamano
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of FI885622A0 publication Critical patent/FI885622A0/fi
Publication of FI885622A publication Critical patent/FI885622A/fi
Application granted granted Critical
Publication of FI90873B publication Critical patent/FI90873B/fi
Publication of FI90873C publication Critical patent/FI90873C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/38—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof
    • C07D501/46—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof with the 7-amino radical acylated by carboxylic acids containing hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI885622A 1987-12-04 1988-12-02 Menetelmä 7 -/(Z)-2-(5-amino-1,2,4-tiadiatsol-3-yyli)-2-metoksi-iminoasetamido/-3-(1-imidatso/1,2-b/-pyridatsinium)metyyli-3-kefeemi-4-karboksylaatti-hydrokloridin kiteiden valmistamiseksi FI90873C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP30835187 1987-12-04
JP30835187 1987-12-04

Publications (4)

Publication Number Publication Date
FI885622A0 true FI885622A0 (fi) 1988-12-02
FI885622A FI885622A (fi) 1989-06-05
FI90873B FI90873B (fi) 1993-12-31
FI90873C FI90873C (fi) 1994-04-11

Family

ID=17980012

Family Applications (1)

Application Number Title Priority Date Filing Date
FI885622A FI90873C (fi) 1987-12-04 1988-12-02 Menetelmä 7 -/(Z)-2-(5-amino-1,2,4-tiadiatsol-3-yyli)-2-metoksi-iminoasetamido/-3-(1-imidatso/1,2-b/-pyridatsinium)metyyli-3-kefeemi-4-karboksylaatti-hydrokloridin kiteiden valmistamiseksi

Country Status (13)

Country Link
US (1) US4978752A (fi)
EP (1) EP0319019A3 (fi)
KR (1) KR890009943A (fi)
CN (1) CN1020611C (fi)
AU (1) AU615966B2 (fi)
DK (1) DK670488A (fi)
FI (1) FI90873C (fi)
HU (1) HU206218B (fi)
NO (1) NO171313C (fi)
NZ (1) NZ227190A (fi)
PT (1) PT89142B (fi)
RU (1) RU2007407C1 (fi)
ZA (1) ZA888903B (fi)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE89826T1 (de) * 1985-03-01 1993-06-15 Takeda Chemical Industries Ltd Antibakterielle verbindungen, ihre herstellung und verwendung.
ATE267831T1 (de) * 1999-09-30 2004-06-15 Otsuka Kagaku Kk Kristalle von cephemderivaten und verfahren zu ihrer herstellung
AU3465901A (en) * 2000-03-03 2001-09-17 Boehringer Ingelheim Pharma Material processing by repeated solvent expansion-contraction
CA2430934C (en) * 2000-12-01 2011-06-21 Takeda Chemical Industries, Ltd. A method of producing sustained-release preparations of a bioactive substance using high-pressure gas
EP1354581A4 (en) * 2000-12-26 2007-07-04 Takeda Pharmaceutical POROUS SUBSTANCE AND METHOD FOR THE PRODUCTION THEREOF
AT413282B (de) * 2002-02-01 2006-01-15 Sandoz Ag Kristalline salze der 7-(((5-amino-1,2,4-thiadiazol-3-yl) (fluoromethoxy-imino)acetyl)amino)-3- ((imino-1-piperazinylmethyl)
EP1606293B1 (en) * 2003-03-27 2009-08-19 Basilea Pharmaceutica AG Cephalosporin in crystalline form
ATE543817T1 (de) * 2003-07-29 2012-02-15 Dainippon Sumitomo Pharma Co Verfahren zur herstellung einer imidverbindung
US7621299B2 (en) 2003-10-03 2009-11-24 Cabot Corporation Method and apparatus for filling a vessel with particulate matter
WO2010089729A1 (en) 2009-02-09 2010-08-12 Ranbaxy Laboratories Limited Processes for the preparation of cefozopran, its salts and polymorphic forms thereof
CN105153201B (zh) * 2015-08-29 2017-08-22 济南康和医药科技有限公司 一种盐酸头孢唑兰的制备方法
CN108227795A (zh) * 2017-12-05 2018-06-29 国网浙江余姚市供电有限公司 一种电网设施配电安全监控系统

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO165842C (no) * 1984-04-23 1991-04-17 Takeda Chemical Industries Ltd Analogifremgangsmaate for fremstilling av terapeutisk aktive cefem-forbindelser.
NO166283C (no) * 1985-03-01 1991-06-26 Takeda Chemical Industries Ltd Analogifremgangsmaate for fremstilling av terapeutisk aktive 7beta-(2-(5-amino-1,2,4-tiadiazol-3-yl)-2(z)-substituertoksyiminoacetamido)-3-(heterocyclylmetyl)-3-cefem-4-karboksylsyrederivater.

Also Published As

Publication number Publication date
NZ227190A (en) 1990-08-28
FI90873C (fi) 1994-04-11
NO171313C (no) 1993-02-24
DK670488D0 (da) 1988-12-01
CN1034727A (zh) 1989-08-16
FI90873B (fi) 1993-12-31
AU2574988A (en) 1989-06-29
AU615966B2 (en) 1991-10-17
NO885295D0 (no) 1988-11-28
FI885622A (fi) 1989-06-05
EP0319019A2 (en) 1989-06-07
DK670488A (da) 1989-06-05
PT89142A (pt) 1989-12-29
US4978752A (en) 1990-12-18
HUT50346A (en) 1990-01-29
NO171313B (no) 1992-11-16
HU206218B (en) 1992-09-28
PT89142B (pt) 1993-09-30
CN1020611C (zh) 1993-05-12
EP0319019A3 (en) 1991-01-16
ZA888903B (en) 1990-07-25
KR890009943A (ko) 1989-08-05
RU2007407C1 (ru) 1994-02-15
NO885295L (no) 1989-06-05

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Owner name: TAKEDA CHEMICAL INDUSTRIES, LTD.