FI844185A0 - N-substituerade isokinolinderivat och foerfarande foer framstaellning daerav. - Google Patents

N-substituerade isokinolinderivat och foerfarande foer framstaellning daerav.

Info

Publication number
FI844185A0
FI844185A0 FI844185A FI844185A FI844185A0 FI 844185 A0 FI844185 A0 FI 844185A0 FI 844185 A FI844185 A FI 844185A FI 844185 A FI844185 A FI 844185A FI 844185 A0 FI844185 A0 FI 844185A0
Authority
FI
Finland
Prior art keywords
alkyl
carbon atoms
phenyl
isokinolinderivat
substituerade
Prior art date
Application number
FI844185A
Other languages
English (en)
Other versions
FI844185L (fi
FI79533C (fi
FI79533B (fi
Inventor
Gabor Bernath
Jenoe Kobor
Ferenc Fueloep
Pal Perjesi
Elemer Ezer
Gyoergy Hajos
Eva Palosi
Laszlo Denes
Laszlo Szporny
Original Assignee
Richter Gedeon Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Vegyeszet filed Critical Richter Gedeon Vegyeszet
Publication of FI844185A0 publication Critical patent/FI844185A0/fi
Publication of FI844185L publication Critical patent/FI844185L/fi
Application granted granted Critical
Publication of FI79533B publication Critical patent/FI79533B/fi
Publication of FI79533C publication Critical patent/FI79533C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/12Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring
    • C07D217/14Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals
    • C07D217/16Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals substituted by oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Transplantation (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
FI844185A 1983-10-25 1984-10-25 Foerfarande foer framstaellning av terapeutiskt anvaendbara n-substituerade isokinolinderivat. FI79533C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU833652A HU189765B (en) 1983-10-25 1983-10-25 Process for preparing n-substituted 1-(bis (hydroxy-metiol)-methyl)-isoquinoline-derivatives
HU365283 1983-10-25

Publications (4)

Publication Number Publication Date
FI844185A0 true FI844185A0 (fi) 1984-10-25
FI844185L FI844185L (fi) 1985-04-26
FI79533B FI79533B (fi) 1989-09-29
FI79533C FI79533C (fi) 1990-01-10

Family

ID=10964925

Family Applications (1)

Application Number Title Priority Date Filing Date
FI844185A FI79533C (fi) 1983-10-25 1984-10-25 Foerfarande foer framstaellning av terapeutiskt anvaendbara n-substituerade isokinolinderivat.

Country Status (9)

Country Link
US (1) US4668688A (fi)
EP (1) EP0142740B1 (fi)
JP (1) JPS60132962A (fi)
AT (1) ATE35133T1 (fi)
CA (1) CA1265141A (fi)
DE (1) DE3472104D1 (fi)
DK (1) DK508484A (fi)
FI (1) FI79533C (fi)
HU (1) HU189765B (fi)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4902695A (en) * 1989-02-13 1990-02-20 Eli Lilly And Company Excitatory amino acid receptor antagonists
US5360568A (en) * 1993-11-12 1994-11-01 Lever Brothers Company, Division Of Conopco, Inc. Imine quaternary salts as bleach catalysts
BR9408038A (pt) * 1993-11-12 1996-12-24 Unilever Nv Composição de branqueamento e processo para branquear um substrato manchado
US5360569A (en) * 1993-11-12 1994-11-01 Lever Brothers Company, Division Of Conopco, Inc. Activation of bleach precursors with catalytic imine quaternary salts
JP5571387B2 (ja) 2007-01-11 2014-08-13 クリティカル・アウトカム・テクノロジーズ・インコーポレイテッド 癌の治療のための化合物および方法
WO2009079797A1 (en) 2007-12-26 2009-07-02 Critical Outcome Technologies, Inc. Compounds and method for treatment of cancer
WO2010006438A1 (en) 2008-07-17 2010-01-21 Critical Outcome Technologies Inc. Thiosemicarbazone inhibitor compounds and cancer treatment methods
US8987272B2 (en) 2010-04-01 2015-03-24 Critical Outcome Technologies Inc. Compounds and method for treatment of HIV

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1199775B (de) * 1960-04-01 1965-09-02 Hoffmann La Roche Verfahren zur Herstellung von analgetisch, hustenlindernd und spasmolytisch wirksamenTetrahydroisochinolinderivaten
US3562280A (en) * 1967-08-30 1971-02-09 Hoffmann La Roche Substituted 1,2,3,4-tetrahydroisoquinolines
DD121321A1 (fi) * 1975-04-24 1976-07-20
HU178454B (en) * 1979-07-02 1982-05-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing new isoquinoline derivatives containing sulphur

Also Published As

Publication number Publication date
EP0142740A1 (en) 1985-05-29
DK508484D0 (da) 1984-10-25
FI844185L (fi) 1985-04-26
US4668688A (en) 1987-05-26
CA1265141A (en) 1990-01-30
JPS60132962A (ja) 1985-07-16
EP0142740B1 (en) 1988-06-15
DE3472104D1 (en) 1988-07-21
FI79533C (fi) 1990-01-10
FI79533B (fi) 1989-09-29
HU189765B (en) 1986-07-28
ATE35133T1 (de) 1988-07-15
DK508484A (da) 1985-04-26

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Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: RICHTER GEDEON VEGYESZETI GYAR R.T.