FI64799C - Foerfarande foer framstaellning av terapeutiskt anvaendbara sustituerade bensendisulfonamider - Google Patents

Foerfarande foer framstaellning av terapeutiskt anvaendbara sustituerade bensendisulfonamider Download PDF

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Publication number
FI64799C
FI64799C FI753392A FI753392A FI64799C FI 64799 C FI64799 C FI 64799C FI 753392 A FI753392 A FI 753392A FI 753392 A FI753392 A FI 753392A FI 64799 C FI64799 C FI 64799C
Authority
FI
Finland
Prior art keywords
compound
formula
amino
give
product
Prior art date
Application number
FI753392A
Other languages
English (en)
Finnish (fi)
Other versions
FI64799B (fi
FI753392A (xx
Inventor
Helmut Hugo Mrozik
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/616,331 external-priority patent/US4064239A/en
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of FI753392A publication Critical patent/FI753392A/fi
Publication of FI64799B publication Critical patent/FI64799B/fi
Application granted granted Critical
Publication of FI64799C publication Critical patent/FI64799C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/30Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/37Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
    • C07C311/38Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring having sulfur atoms of sulfonamide groups and amino groups bound to carbon atoms of six-membered rings of the same carbon skeleton
    • C07C311/39Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring having sulfur atoms of sulfonamide groups and amino groups bound to carbon atoms of six-membered rings of the same carbon skeleton having the nitrogen atom of at least one of the sulfonamide groups bound to hydrogen atoms or to an acyclic carbon atom
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/10Organic substances
    • A23K20/111Aromatic compounds
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/10Organic substances
    • A23K20/116Heterocyclic compounds
    • A23K20/121Heterocyclic compounds containing oxygen or sulfur as hetero atom
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23KFODDER
    • A23K20/00Accessory food factors for animal feeding-stuffs
    • A23K20/10Organic substances
    • A23K20/116Heterocyclic compounds
    • A23K20/137Heterocyclic compounds containing two hetero atoms, of which at least one is nitrogen
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/63Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00Preparation of halogenated hydrocarbons
    • C07C17/013Preparation of halogenated hydrocarbons by addition of halogens
    • C07C17/04Preparation of halogenated hydrocarbons by addition of halogens to unsaturated halogenated hydrocarbons
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00Preparation of halogenated hydrocarbons
    • C07C17/26Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton
    • C07C17/263Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by condensation reactions
    • C07C17/2637Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by condensation reactions between a compound containing only oxygen and possibly halogen as hetero-atoms and a halogenated hydrocarbon
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/07Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by halogen atoms
    • C07C205/11Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by halogen atoms having nitro groups bound to carbon atoms of six-membered aromatic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Polymers & Plastics (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Husbandry (AREA)
  • Zoology (AREA)
  • Engineering & Computer Science (AREA)
  • Food Science & Technology (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
FI753392A 1974-12-16 1975-12-02 Foerfarande foer framstaellning av terapeutiskt anvaendbara sustituerade bensendisulfonamider FI64799C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US53335274A 1974-12-16 1974-12-16
US53335274 1974-12-16
US61633175 1975-09-26
US05/616,331 US4064239A (en) 1974-12-16 1975-09-26 Halogenated unsaturated alkyl benzenedisulfonamides as anthelmintics

Publications (3)

Publication Number Publication Date
FI753392A FI753392A (xx) 1976-06-17
FI64799B FI64799B (fi) 1983-09-30
FI64799C true FI64799C (fi) 1984-01-10

Family

ID=27064157

Family Applications (1)

Application Number Title Priority Date Filing Date
FI753392A FI64799C (fi) 1974-12-16 1975-12-02 Foerfarande foer framstaellning av terapeutiskt anvaendbara sustituerade bensendisulfonamider

Country Status (16)

Country Link
AR (1) AR218216A1 (xx)
CA (1) CA1058194A (xx)
DE (1) DE2556122C2 (xx)
DK (1) DK145756C (xx)
FI (1) FI64799C (xx)
FR (1) FR2294710A1 (xx)
GB (1) GB1485897A (xx)
IE (1) IE42203B1 (xx)
IL (1) IL48610A (xx)
LU (1) LU74019A1 (xx)
NL (2) NL187394C (xx)
NO (1) NO142667C (xx)
NZ (1) NZ179477A (xx)
OA (1) OA05183A (xx)
PH (1) PH12041A (xx)
SE (1) SE426817B (xx)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107868024A (zh) * 2017-10-25 2018-04-03 浙江海正药业股份有限公司 克洛索隆的晶型及其制备方法和用途
CN113773235B (zh) * 2021-08-20 2022-06-17 北大方正集团有限公司 一种氯舒隆的合成方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1483222A (fr) * 1965-06-24 1967-06-02 Merck & Co Inc Production de nouveaux dérivés, substitués à l'azote, de la 5-chloro-2, 4-disulfamoylaniline
SE410598B (sv) * 1973-05-11 1979-10-22 Merck & Co Inc Forfarande for framstellning av bensendisulfonamider med anthelmintisk verkan

Also Published As

Publication number Publication date
IE42203L (en) 1976-06-16
DE2556122A1 (de) 1976-06-24
NL930115I1 (nl) 1993-10-18
DK544775A (da) 1976-06-17
GB1485897A (en) 1977-09-14
DK145756C (da) 1983-08-08
LU74019A1 (xx) 1976-11-11
FI64799B (fi) 1983-09-30
AU8743575A (en) 1977-06-16
AR218216A1 (es) 1980-05-30
PH12041A (en) 1978-10-16
OA05183A (fr) 1981-01-31
NZ179477A (en) 1978-04-03
SE7513569L (sv) 1976-06-17
DK145756B (da) 1983-02-21
NL7514163A (nl) 1976-06-18
IL48610A0 (en) 1976-02-29
NL187394B (nl) 1991-04-16
IE42203B1 (en) 1980-06-18
IL48610A (en) 1979-10-31
FI753392A (xx) 1976-06-17
NO142667B (no) 1980-06-16
NO142667C (no) 1980-09-24
DE2556122C2 (de) 1986-05-22
FR2294710A1 (fr) 1976-07-16
SE426817B (sv) 1983-02-14
NL187394C (nl) 1991-09-16
NO754087L (xx) 1976-06-17
FR2294710B1 (xx) 1979-09-21
CA1058194A (en) 1979-07-10

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Legal Events

Date Code Title Description
MM Patent lapsed
MM Patent lapsed

Owner name: MERCK & CO INC.