FI48067C - Analogiamenetelmä terapeuttisesti vaikuttavien uusien 1-(3,5-dihalogee ni-4-hydroksifenyyli)-2-(2-fenoksi- tai 2-bentsyyli-isopropyyliamino)- propanolien ja niiden happoadditiosuolojen valmistamiseksi - Google Patents

Analogiamenetelmä terapeuttisesti vaikuttavien uusien 1-(3,5-dihalogee ni-4-hydroksifenyyli)-2-(2-fenoksi- tai 2-bentsyyli-isopropyyliamino)- propanolien ja niiden happoadditiosuolojen valmistamiseksi

Info

Publication number
FI48067C
FI48067C FI680050A FI5068A FI48067C FI 48067 C FI48067 C FI 48067C FI 680050 A FI680050 A FI 680050A FI 5068 A FI5068 A FI 5068A FI 48067 C FI48067 C FI 48067C
Authority
FI
Finland
Prior art keywords
benzylisopropylamino
propanols
dihalogen
hydroxyphenyl
phenoxy
Prior art date
Application number
FI680050A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI48067B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html
Inventor
Fourneau
Delourme
Original Assignee
Applic Scient Et Soc D
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Applic Scient Et Soc D filed Critical Applic Scient Et Soc D
Publication of FI48067B publication Critical patent/FI48067B/fi
Application granted granted Critical
Publication of FI48067C publication Critical patent/FI48067C/fi

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FI680050A 1967-01-10 1968-01-09 Analogiamenetelmä terapeuttisesti vaikuttavien uusien 1-(3,5-dihalogee ni-4-hydroksifenyyli)-2-(2-fenoksi- tai 2-bentsyyli-isopropyyliamino)- propanolien ja niiden happoadditiosuolojen valmistamiseksi FI48067C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR90478A FR6087M (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1967-01-10 1967-01-10
FR133258A FR6934M (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1967-01-10 1967-12-21

Publications (2)

Publication Number Publication Date
FI48067B FI48067B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1974-02-28
FI48067C true FI48067C (fi) 1974-06-10

Family

ID=26174501

Family Applications (1)

Application Number Title Priority Date Filing Date
FI680050A FI48067C (fi) 1967-01-10 1968-01-09 Analogiamenetelmä terapeuttisesti vaikuttavien uusien 1-(3,5-dihalogee ni-4-hydroksifenyyli)-2-(2-fenoksi- tai 2-bentsyyli-isopropyyliamino)- propanolien ja niiden happoadditiosuolojen valmistamiseksi

Country Status (13)

Country Link
US (1) US3542870A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AT (1) AT278750B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BE (1) BE709012A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CH (1) CH485658A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DE (1) DE1668930C3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DK (1) DK120400B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ES (1) ES349044A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FI (1) FI48067C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FR (2) FR6087M (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GB (1) GB1146139A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
SE (1) SE349020B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
SU (1) SU456406A3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
YU (1) YU34272B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3163871D1 (en) 1980-07-09 1984-07-05 Draco Ab 1-(dihydroxyphenyl)-2-amino-ethanol derivatives; preparation, compositions and intermediates
JPS6058927A (ja) * 1983-09-09 1985-04-05 Nippon Mejifuijitsukusu Kk 放射能標識血小板製剤
US4699928A (en) * 1984-07-13 1987-10-13 Merrell Dow Pharmaceuticals Inc. Fluoroallylamine derivatives
US6650943B1 (en) 2000-04-07 2003-11-18 Advanced Bionics Corporation Fully implantable neurostimulator for cavernous nerve stimulation as a therapy for erectile dysfunction and other sexual dysfunction
US6885895B1 (en) * 2001-04-26 2005-04-26 Advanced Bionics Corporation Methods and systems for electrical and/or drug stimulation as a therapy for erectile dysfunction
PL375713A1 (en) 2002-08-19 2005-12-12 Pfizer Products Inc. Combination therapy for hyperproliferative diseases
WO2005089741A2 (en) * 2004-03-17 2005-09-29 Sosei R&D Ltd. The treatment of inflammatory disorders and pain using beta-aminoalcohols
US7741317B2 (en) 2005-10-21 2010-06-22 Bristol-Myers Squibb Company LXR modulators
US7888376B2 (en) 2005-11-23 2011-02-15 Bristol-Myers Squibb Company Heterocyclic CETP inhibitors
US8383660B2 (en) 2006-03-10 2013-02-26 Pfizer Inc. Dibenzyl amine compounds and derivatives
US7919506B2 (en) 2006-03-10 2011-04-05 Pfizer Inc. Dibenzyl amine compounds and derivatives
ES2382009T3 (es) 2006-12-01 2012-06-04 Bristol-Myers Squibb Company Derivados de N-((3-bencil)-2,2-(bis-fenil-)-propan-1-amina como inhibidores de CETP para el tratamiento de aterosclerosis y enfermedades cardiovasculares
EP2986599A1 (en) 2013-04-17 2016-02-24 Pfizer Inc. N-piperidin-3-ylbenzamide derivatives for treating cardiovascular diseases
WO2016055901A1 (en) 2014-10-08 2016-04-14 Pfizer Inc. Substituted amide compounds
MX2021008533A (es) 2019-01-18 2021-08-19 Astrazeneca Ab Inhibidores de la pcsk9 y metodos de uso de los mismos.

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2661372A (en) * 1953-12-01 Pharmacologically valuable stereo
GB789033A (en) * 1954-10-23 1958-01-15 Philips Nv Improvements in or relating to substituted aralkyl-phenyl-alkylamines
FR1165845A (fr) * 1955-05-28 1958-10-29 Philips Nv Amines secondaires portant des substituants et leur préparation
GB800718A (en) * 1955-05-28 1958-09-03 Philips Nv Novel substituted alkylamines and processes for their production
BE630296A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * 1962-03-31
NL130079C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * 1963-06-28
FR3654M (fr) * 1963-11-08 1965-11-02 Raymond Michel β(-3:5 diiodo-4 hydroxyphényl) βhydroxy αméthyl n méthyléthylamine-synthese et a titre d'hypertenseur a action prolongée, son utilisation dans le traitement des collapsus cardiovasculaires.

Also Published As

Publication number Publication date
YU4668A (en) 1978-10-31
AT278750B (de) 1970-02-10
DK120400B (da) 1971-05-24
DE1668930A1 (de) 1971-09-16
FR6087M (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1968-06-04
SE349020B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1972-09-18
SU456406A3 (ru) 1975-01-05
GB1146139A (en) 1969-03-19
FI48067B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1974-02-28
CH485658A (fr) 1970-02-15
FR6934M (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1969-05-05
US3542870A (en) 1970-11-24
YU34272B (en) 1979-04-30
DE1668930B2 (de) 1973-08-02
BE709012A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1968-05-16
DE1668930C3 (de) 1974-02-28
ES349044A1 (es) 1969-08-16

Similar Documents

Publication Publication Date Title
FI48067C (fi) Analogiamenetelmä terapeuttisesti vaikuttavien uusien 1-(3,5-dihalogee ni-4-hydroksifenyyli)-2-(2-fenoksi- tai 2-bentsyyli-isopropyyliamino)- propanolien ja niiden happoadditiosuolojen valmistamiseksi
AT289066B (de) Verfahren zur Herstellung von neuen substituierten 1-Amino-2-hydroxy-3-[2'-cyclopentyl- bzw. -(Δ2-cyclopentenyl)-phenoxy]-propanen, deren optisch aktiven Isomeren und Salzen
FI51936C (fi) Menetelmä terapeuttisesti käytettävien 3,4-dihydronaftalenonioksi-2-hy droksipropyyliamiinien ja näiden happo-additiosuolojen valmistamiseksi .
FI49720C (fi) Menetelmä terapeuttisesti vaikuttavien 2-metyyli-3-karbonihappoamidoki noksaliini-di-N-oksidien-(1,4) valmistamiseksi.
DK127599B (da) Analogifremgangsmåde til fremstilling af terapeutisk virksomme 2,4-diaminosubstituerede quinazolin-forbindelser eller syreadditionssalte heraf.
FI49409C (fi) Menetelmä farmakologisesti aktiivisten kinuklidiini-2- ja kinuklidiini -3-karboksyylihapon anilidien ja niiden terapeuttisesti hyväksyttävien suolojen valmistamiseksi.
DK119768B (da) Analogifremgangsmåde til fremstilling af terapeutisk virksomme pyridinsubstituerede malonater eller farmaceutisk acceptable syreadditionssalte deraf.
FI49718C (fi) Menetelmä terapeuttisesti vaikuttavien 2-halogeenimetyyli-3-karbonihap poamidokinoksaliini-di-N-oksidien-(1,4) valmistamiseksi.
DK121236B (da) Analogifremgangsmåde til fremstilling af terapeutisk aktive, basisk substituerede amider af N-substituerede antranilsyrer, eller syreadditionssalte deraf.
FI50420C (fi) Menetelmä terapeuttisesti aktiivisten 4-pyrimidinyyli-1,4-dihydropyrid iinijohdannaisten valmistamiseksi
IT1064102B (it) Procedimento per la preparazione di acido 6 amino penicillanico
FI48576C (fi) Menetelmä terapeuttisesti aktiivisten alfa-fluori-malonihappojohdannai sten valmistamiseksi.
NL145542B (nl) Werkwijze ter bereiding van therapeutisch werkzame carbaminezuurderivaten.
DK118613B (da) Fremgangsmåde til fremstilling af terapeutisk aktive 3,4-dihydroxyphenyl-alkanolaminer eller syreadditionssalte heraf.
FI46955C (fi) Menetelmä terapeuttisesti vaikuttavan 1-p-klooribentsoyyli-2-alempi-al kyyli-5-alempi-alkoksi-3-indolyyli-etikkahapon valmistamiseksi
FI45175C (fi) Menetelmä 18-metyyli-19-nor-17alfa-hydroksi-progesteronien ja niiden 1 7alfa-esterien valmistamiseksi.
SE403773B (sv) Forfarande for framstellning av vissa alfa-aminoalkyl-4-hydroxi-3(alkylsulfonylmetyl) bensylalkoholer eller farmaceutiskt acceptabla syraadditionssalter derav
IT1036002B (it) Procedimento per al preparazione di acido 6,7di idrossicumarin 4 metisolfonico e dei suoi sali
FI52572C (fi) Menetelmä terapeuttisesti käytettävien, heksahydro-1H-atsepiiniyhdiste iden vasemmalle kiertävien optisten isomeerien sekä näiden happoadditi osuolojen ja kvaternääristen ammoniumsuolojen valmistamiseksi.
FI49416C (fi) Menetelmä uusien farmakologisesti aktiivisten bentsofuraani-2-karbonih appojohdannaisten valmistamiseksi.
FI49021C (fi) Menetelmä terapeuttisesti vaikuttavien substituoitujen p-alkenyylioksi -ja p-alkynyylioksifenyylietikkahappojen tai niiden suolojen valmistam iseksi.
FI42566C (fi) Menetelmä terapeuttisesti vaikuttavan 2-£5',6',7',8'-tetrahydronaftyyli-(1')-amino|-imidatsoliinin valmistamiseksi
FI44229C (fi) Menetelmä analgeettisten beeta-tyydyttämättömien-beeta-hydroksi-beeta-fenyylietyyliamiinien ja niiden happoadditiosuolojen valmistamiseksi
FI50877C (fi) Menetelmä sienten kasvua estävinä aineina käytettävien N-trityyli-imid atsolien ja niiden suolojen valmistamiseksi.
FI36795A (fi) Menetelmä N-(2,3-dimetyylifenyyli)-antraniilihapon valmistamiseksi