ES8800943A1 - Un procedimiento para preparar compuestos imidazoheterociclicos - Google Patents

Un procedimiento para preparar compuestos imidazoheterociclicos

Info

Publication number
ES8800943A1
ES8800943A1 ES555653A ES555653A ES8800943A1 ES 8800943 A1 ES8800943 A1 ES 8800943A1 ES 555653 A ES555653 A ES 555653A ES 555653 A ES555653 A ES 555653A ES 8800943 A1 ES8800943 A1 ES 8800943A1
Authority
ES
Spain
Prior art keywords
alkyl
preparation
pharmaceutical compositions
alkynyloxy
processes
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES555653A
Other languages
English (en)
Other versions
ES555653A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Fujisawa Pharmaceutical Co Ltd
Original Assignee
Fujisawa Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB858514080A external-priority patent/GB8514080D0/en
Priority claimed from GB858530878A external-priority patent/GB8530878D0/en
Application filed by Fujisawa Pharmaceutical Co Ltd filed Critical Fujisawa Pharmaceutical Co Ltd
Publication of ES555653A0 publication Critical patent/ES555653A0/es
Publication of ES8800943A1 publication Critical patent/ES8800943A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Detergent Compositions (AREA)
  • Lubricants (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

PROCEDIMIENTO PARA LA PREPARACION DE COMPUESTOS IMIDAZOHETEROCICLICOS, DE FORMULA GENERAL (I), Y SUS SALES FARMACEUTICAMENTE ACEPTABLES. CONSISTE EN HACER REACCIONAR UN COMPUESTO DE FORMULA GENERAL (II) O UNA SAL DEL MISMO, CON UN COMPUESTO DE FORMULA GENERAL (III), EN LAS QUE R1 ES ALQUENILO INFERIOR, ALQUINILO INFERIOR Y ALCADIENILO INFERIOR; R2 ES HIDROGENO, ALQUILO INFERIOR O ARILO; R3 ES AR(ALQUILO INFERIOR) QUE PUEDE TENER 1 A 3 SUSTITUYENTES; X ES OXIGENO O NH; Y ES CH O N; Y Z1 ES UN RESIDUO DE ACIDO O UNA SAL DEL MISMO, REALIZANDOSE LA REACCION EN UN DISOLVENTE SELECCIONADO ENTRE ALCOHOL, BENCENO, TETRAHIDROFURANO Y ETER DIETILICO, A TEMPERATURA AMBIENTE O BAJO CALENTAMIENTO MODERADO O INTENSO. DE APLICACION EN TERAPEUTICA POR SU ACTIVIDAD ANTIULCERATIVA.
ES555653A 1985-06-04 1986-06-03 Un procedimiento para preparar compuestos imidazoheterociclicos Expired ES8800943A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB858514080A GB8514080D0 (en) 1985-06-04 1985-06-04 Imidazopyridine compounds
GB858530878A GB8530878D0 (en) 1985-12-16 1985-12-16 Imidazopyridine compounds

Publications (2)

Publication Number Publication Date
ES555653A0 ES555653A0 (es) 1987-12-01
ES8800943A1 true ES8800943A1 (es) 1987-12-01

Family

ID=26289330

Family Applications (1)

Application Number Title Priority Date Filing Date
ES555653A Expired ES8800943A1 (es) 1985-06-04 1986-06-03 Un procedimiento para preparar compuestos imidazoheterociclicos

Country Status (15)

Country Link
US (1) US4725601A (es)
EP (1) EP0204285B1 (es)
KR (1) KR870000332A (es)
CN (1) CN86104313A (es)
AT (1) ATE71625T1 (es)
AU (1) AU593802B2 (es)
CA (1) CA1257264A (es)
DE (1) DE3683403D1 (es)
DK (1) DK250386A (es)
ES (1) ES8800943A1 (es)
FI (1) FI862210A (es)
GR (1) GR861379B (es)
HU (1) HUT40798A (es)
IL (1) IL78923A0 (es)
NO (1) NO862208L (es)

Families Citing this family (44)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4831041A (en) * 1986-11-26 1989-05-16 Fujisawa Pharmaceutical Co., Ltd. Imidazopyridine compounds and processes for preparation thereof
IL86269A0 (en) * 1987-05-08 1988-11-15 Byk Gulden Lomberg Chem Fab Imidazole derivatives,processes for the preparation thereof and pharmaceutical compositions containing the same
KR890701585A (ko) * 1987-07-16 1989-12-21 헤르베르크 슈키·울리히 볼프 새로운 디아졸
GB8722488D0 (en) * 1987-09-24 1987-10-28 Fujisawa Pharmaceutical Co Imidazopyridine compound
AT390438B (de) * 1987-10-08 1990-05-10 Yamanouchi Pharma Co Ltd Neue imidazo(1,2-a)pyridinderivate und deren herstellung und diese enthaltende pharmazeutische zubereitungen
SE8704248D0 (sv) * 1987-10-30 1987-10-30 Haessle Ab Medical use
WO1990005136A1 (de) * 1988-11-07 1990-05-17 Byk Gulden Lomberg Chemische Fabrik Gmbh Neue imidazopyridine
DE3837809A1 (de) * 1988-11-08 1990-05-10 Merck Patent Gmbh Tetralinderivate
GB9201693D0 (en) * 1992-01-27 1992-03-11 Smithkline Beecham Intercredit Compounds
US5574042A (en) * 1992-11-02 1996-11-12 Fujisawa Pharmaceutical Co., Ltd Imidazo [1,2-a] pyridines and their pharmaceutical use
UA48122C2 (uk) * 1993-10-11 2002-08-15 Бік Гульден Ломберг Хеміше Фабрік Гмбх АЛКОКСІАЛКІЛКАРБАМАТИ ІМІДАЗО[1,2-а]ПІРИДИНІВ, СПОСІБ ЇХ ОДЕРЖАННЯ ТА ЛІКАРСЬКИЙ ЗАСІБ НА ЇХ ОСНОВІ
CZ22697A3 (en) * 1994-07-28 1997-07-16 Byk Gulden Lomberg Chem Fab Imidazopyridine-azolidinone derivatives, process of their preparation and pharmaceutical composition containing thereof
CA2218705A1 (en) * 1995-04-21 1996-10-24 Shinnippon Pharmaceutical Inc. Fused imidazo¬1,2-a|pyridines
EP0778277B1 (en) * 1995-12-08 2003-06-25 Pfizer Inc. Substituted heterocyclic derivatives as CRF antagonists
US6992188B1 (en) 1995-12-08 2006-01-31 Pfizer, Inc. Substituted heterocyclic derivatives
WO1997027192A1 (de) * 1996-01-26 1997-07-31 Byk Gulden Lomberg Chemische Fabrik Gmbh 3-methylimidazopyridine
AU1545297A (en) * 1996-01-26 1997-08-20 Byk Gulden Imidazopyridine halides
SE9700661D0 (sv) * 1997-02-25 1997-02-25 Astra Ab New compounds
SE9704404D0 (sv) 1997-11-28 1997-11-28 Astra Ab New compounds
SE9801526D0 (sv) * 1998-04-29 1998-04-29 Astra Ab New compounds
SE9802794D0 (sv) * 1998-08-21 1998-08-21 Astra Ab New compounds
SE9802793D0 (sv) 1998-08-21 1998-08-21 Astra Ab New compounds
CA2311483A1 (en) * 2000-06-12 2001-12-12 Gregory N Beatch IMIDAZO [1,2-A] PYRIDINIC ETHERS AND USES THEREOF
SE0003186D0 (sv) * 2000-09-07 2000-09-07 Astrazeneca Ab New process
US6900324B2 (en) 2000-09-07 2005-05-31 Astrazeneca Ab Process for preparing a substituted imidazopyridine compound
UA80393C2 (uk) 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
SE0102808D0 (sv) * 2001-08-22 2001-08-22 Astrazeneca Ab New compounds
DE10145457A1 (de) 2001-09-14 2003-04-03 Basf Ag Substituierte Imidazo[1,2-a]-5,6,7,8-tetrahydropyridin-8-one, Verfahren zu ihrer Herstellung, sowie deren Verwendung zur Herstellung von Imidazo[1,2,-a]pyridinen
MY140561A (en) * 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
AR043002A1 (es) * 2003-02-18 2005-07-13 Altana Pharma Ag Imidazopirazinas 6-substituidos
CA2517256C (en) 2003-02-26 2013-04-30 Sugen, Inc. Aminoheteroaryl compounds as protein kinase inhibitors
EP1606261B1 (en) 2003-03-10 2009-11-04 Nycomed GmbH Novel process for the preparation of roflumilast
SE0301904D0 (sv) * 2003-06-26 2003-06-26 Astrazeneca Ab Novel imidazopyridine compound II with therapeutic effect
CN1874772A (zh) 2003-11-03 2006-12-06 阿斯利康(瑞典)有限公司 治疗隐匿性胃食管反流的咪唑并[1,2－a]吡啶衍生物
JP2008523139A (ja) * 2004-12-14 2008-07-03 アストラゼネカ・アクチエボラーグ 置換アミノピリジン類及びその使用
EP1861074B1 (en) * 2005-03-16 2013-04-24 Takeda GmbH Taste masked dosage form containing roflumilast
CA2620223A1 (en) 2005-09-02 2007-03-08 Abbott Laboratories Novel imidazo based heterocycles
WO2007066185A2 (en) 2005-12-05 2007-06-14 Pfizer Products Inc. Polymorphs of a c-met/hgfr inhibitor
PL1959955T3 (pl) 2005-12-05 2011-04-29 Pfizer Prod Inc Sposób traktowania nieprawidłowego wzrostu komórek
CA2654202A1 (en) * 2006-06-06 2007-12-21 Schering Corporation Imidazopyrazines as protein kinase inhibitors
US20080051420A1 (en) * 2006-06-14 2008-02-28 Astrazeneca Ab New Compounds 317
TW200815447A (en) * 2006-06-14 2008-04-01 Astrazeneca Ab Novel compounds IV
FI20086158A0 (fi) * 2008-12-03 2008-12-03 Mikael Dahlstroem Imidatsopyridiinijohdannaiset
JP5458813B2 (ja) * 2009-11-10 2014-04-02 オムロン株式会社 光電センサ

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA81219B (en) * 1980-01-23 1982-01-27 Schering Corp Imidazo (1,2-a) pyridines ,process for their preparation and pharmaceutical compositions containing them
US4507294A (en) * 1982-03-08 1985-03-26 Schering Corp. Imidazo[1,2-a]pyrazines
EP0068378B1 (en) * 1981-06-26 1986-03-05 Schering Corporation Novel imidazo(1,2-a)pyridines and pyrazines, processes for their preparation and pharmaceutical compositions containing them
AU7928787A (en) * 1986-10-07 1988-04-14 Yamanouchi Pharmaceutical Co., Ltd. Imidazopyridine derivatives
US4831041A (en) * 1986-11-26 1989-05-16 Fujisawa Pharmaceutical Co., Ltd. Imidazopyridine compounds and processes for preparation thereof

Also Published As

Publication number Publication date
DK250386A (da) 1986-12-05
CA1257264A (en) 1989-07-11
HUT40798A (en) 1987-02-27
DE3683403D1 (de) 1992-02-27
ES555653A0 (es) 1987-12-01
KR870000332A (ko) 1987-02-17
NO862208L (no) 1986-12-05
CN86104313A (zh) 1987-03-04
EP0204285A1 (en) 1986-12-10
ATE71625T1 (de) 1992-02-15
US4725601A (en) 1988-02-16
FI862210A0 (fi) 1986-05-26
NO862208D0 (no) 1986-06-03
DK250386D0 (da) 1986-05-28
IL78923A0 (en) 1986-09-30
EP0204285B1 (en) 1992-01-15
AU5834586A (en) 1986-12-11
FI862210A (fi) 1986-12-05
GR861379B (en) 1986-08-28
AU593802B2 (en) 1990-02-22

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Legal Events

Date Code Title Description
MM4A Patent lapsed

Effective date: 19960401