ES8605516A1 - Procedimiento para preparar derivados de pirazolpiridina - Google Patents
Procedimiento para preparar derivados de pirazolpiridinaInfo
- Publication number
- ES8605516A1 ES8605516A1 ES538957A ES538957A ES8605516A1 ES 8605516 A1 ES8605516 A1 ES 8605516A1 ES 538957 A ES538957 A ES 538957A ES 538957 A ES538957 A ES 538957A ES 8605516 A1 ES8605516 A1 ES 8605516A1
- Authority
- ES
- Spain
- Prior art keywords
- group
- alkylcarbamoyl
- carboxy
- dialkylcarbamoyl
- methyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pain & Pain Management (AREA)
- Pharmacology & Pharmacy (AREA)
- Rheumatology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
PROCEDIMIENTO PARA PREPARAR DERIVADOS DE PIRAZOLPIRIDINA. CONSISTE EN HACER REACCIONAR UN COMPUESTO DE FORMULA (II) CON UN COMPUESTO DE FORMULA (IV), EN UN DISOLVENTE ORGANICO COMO ETANOL, A UNA TEMPERATURA DE 0 A 10JC, PARA OBTENER UN COMPUESTO DE FORMULA (I), Y SUS SALES FARMACEUTICAMENTE ACEPTABLES, CUANDO: R1 ES ALQUILCARBAMOILO, CUANDO N ES 0, O R1 ES DINTINTO DE UN GRUPO DIALQUILCARBAMOILO, CUANDO N ES 1 Y R2 ES METILO. SIENDO: R1 CARBAMOILO, ALQUILCARBAMOILO O DIALQUILCARBAMOILO; R2, HAL, ALQUILO, CIANO, Y OTROS; Q, HAL, FORMULA (III); R4 Y R5, H, ALQUILO DE CADENA RECTA O RAMIFICADA DE C 1 A 6. SE UTILIZA PARA INHIBIR LA EMIGRACION DE CELULAS MACROFAGICAS Y COMO MEDIDA DEL ANTAGONISMO O REDUCCION DE LOS NIVELES DE LINFOCINAS.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB838334001A GB8334001D0 (en) | 1983-12-21 | 1983-12-21 | Compositions of matter |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES8605516A1 true ES8605516A1 (es) | 1986-03-16 |
| ES538957A0 ES538957A0 (es) | 1986-03-16 |
Family
ID=10553616
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES538957A Expired ES8605516A1 (es) | 1983-12-21 | 1984-12-21 | Procedimiento para preparar derivados de pirazolpiridina |
| ES542457A Expired ES8603426A1 (es) | 1983-12-21 | 1985-04-22 | Procedimiento para preparar derivados de pirazolpiridina. |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES542457A Expired ES8603426A1 (es) | 1983-12-21 | 1985-04-22 | Procedimiento para preparar derivados de pirazolpiridina. |
Country Status (18)
| Country | Link |
|---|---|
| JP (1) | JPS60172979A (es) |
| KR (1) | KR850004758A (es) |
| AT (1) | ATA404684A (es) |
| AU (1) | AU3690684A (es) |
| BE (1) | BE901336A (es) |
| DE (1) | DE3447730A1 (es) |
| DK (1) | DK616784A (es) |
| ES (2) | ES8605516A1 (es) |
| FI (1) | FI845022L (es) |
| FR (1) | FR2556723A1 (es) |
| GB (2) | GB8334001D0 (es) |
| GR (1) | GR82507B (es) |
| IL (1) | IL73860A0 (es) |
| IT (1) | IT1178768B (es) |
| LU (1) | LU85690A1 (es) |
| NL (1) | NL8403874A (es) |
| SE (1) | SE8406478L (es) |
| ZA (1) | ZA849903B (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20070155738A1 (en) | 2005-05-20 | 2007-07-05 | Alantos Pharmaceuticals, Inc. | Heterobicyclic metalloprotease inhibitors |
| JP2010533173A (ja) * | 2007-07-11 | 2010-10-21 | オークランド・ユニサーヴィシズ・リミテッド | ピラゾロ［１，５−ａ］ピリジン、及び癌治療におけるその使用 |
| JP6816287B2 (ja) * | 2016-09-07 | 2021-01-20 | シャンハイ ハイヘ ファーマシューティカル カンパニー リミテッドＳｈａｎｇｈａｉ Ｈａｉｈｅ Ｐｈａｒｍａｃｅｕｔｉｃａｌ Ｃｏ．， Ｌｔｄ | ピリジン並びに５員芳香環系化合物、その製造方法及び使用 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5154583A (en) * | 1974-11-01 | 1976-05-13 | Kyorin Seiyaku Kk | Shinkipirazoro * 1 55a * pirijinjudotaino seizoho |
| JPS5610114A (en) * | 1979-07-05 | 1981-02-02 | Grelan Pharmaceut Co Ltd | Novel analgesic and anti-inflammatory agent |
| GB2121799B (en) * | 1982-06-16 | 1985-07-10 | May & Baker Ltd | New pyrazolopyridine derivative |
-
1983
- 1983-12-21 GB GB838334001A patent/GB8334001D0/en active Pending
-
1984
- 1984-12-18 LU LU85690A patent/LU85690A1/fr unknown
- 1984-12-19 SE SE8406478A patent/SE8406478L/xx not_active Application Discontinuation
- 1984-12-19 JP JP59268203A patent/JPS60172979A/ja active Pending
- 1984-12-19 GR GR82507A patent/GR82507B/el unknown
- 1984-12-19 ZA ZA849903A patent/ZA849903B/xx unknown
- 1984-12-19 KR KR1019840008098A patent/KR850004758A/ko not_active Application Discontinuation
- 1984-12-19 FI FI845022A patent/FI845022L/fi not_active Application Discontinuation
- 1984-12-19 GB GB08431986A patent/GB2153818B/en not_active Expired
- 1984-12-19 AU AU36906/84A patent/AU3690684A/en not_active Abandoned
- 1984-12-19 IL IL73860A patent/IL73860A0/xx unknown
- 1984-12-20 DK DK616784A patent/DK616784A/da not_active Application Discontinuation
- 1984-12-20 BE BE0/214208A patent/BE901336A/fr not_active IP Right Cessation
- 1984-12-20 AT AT0404684A patent/ATA404684A/de not_active IP Right Cessation
- 1984-12-20 FR FR8419522A patent/FR2556723A1/fr not_active Withdrawn
- 1984-12-20 NL NL8403874A patent/NL8403874A/nl not_active Application Discontinuation
- 1984-12-21 IT IT24176/84A patent/IT1178768B/it active
- 1984-12-21 ES ES538957A patent/ES8605516A1/es not_active Expired
- 1984-12-21 DE DE19843447730 patent/DE3447730A1/de not_active Withdrawn
-
1985
- 1985-04-22 ES ES542457A patent/ES8603426A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| SE8406478L (sv) | 1985-06-22 |
| IT8424176A0 (it) | 1984-12-21 |
| BE901336A (fr) | 1985-06-20 |
| IL73860A0 (en) | 1985-03-31 |
| FI845022A0 (fi) | 1984-12-19 |
| NL8403874A (nl) | 1985-07-16 |
| ZA849903B (en) | 1985-08-28 |
| FR2556723A1 (fr) | 1985-06-21 |
| LU85690A1 (fr) | 1986-07-17 |
| AU3690684A (en) | 1985-07-04 |
| GB8334001D0 (en) | 1984-02-01 |
| DE3447730A1 (de) | 1985-07-04 |
| ES542457A0 (es) | 1985-12-16 |
| GB2153818A (en) | 1985-08-29 |
| DK616784A (da) | 1985-06-22 |
| GB8431986D0 (en) | 1985-01-30 |
| KR850004758A (ko) | 1985-07-27 |
| GR82507B (en) | 1985-04-22 |
| GB2153818B (en) | 1987-07-29 |
| FI845022L (fi) | 1985-06-22 |
| ES8603426A1 (es) | 1985-12-16 |
| JPS60172979A (ja) | 1985-09-06 |
| SE8406478D0 (sv) | 1984-12-19 |
| ATA404684A (de) | 1987-08-15 |
| DK616784D0 (da) | 1984-12-20 |
| IT1178768B (it) | 1987-09-16 |
| ES538957A0 (es) | 1986-03-16 |
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