ES8308568A1 - Un procedimiento para la preparacion de nuevos derivados del 1,1-dioxido del acido penicilanico. - Google Patents
Un procedimiento para la preparacion de nuevos derivados del 1,1-dioxido del acido penicilanico.Info
- Publication number
- ES8308568A1 ES8308568A1 ES515577A ES515577A ES8308568A1 ES 8308568 A1 ES8308568 A1 ES 8308568A1 ES 515577 A ES515577 A ES 515577A ES 515577 A ES515577 A ES 515577A ES 8308568 A1 ES8308568 A1 ES 8308568A1
- Authority
- ES
- Spain
- Prior art keywords
- amino
- group
- antibacterial
- penicillanoyloxymethyl
- acetamido
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 230000000844 anti-bacterial effect Effects 0.000 title abstract 2
- 125000000738 acetamido group Chemical group [H]C([H])([H])C(=O)N([H])[*] 0.000 title 1
- 150000002148 esters Chemical class 0.000 title 1
- 239000002253 acid Substances 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- -1 AMINO Chemical class 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 230000001012 protector Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/78—Compounds with an amino radical, acylated by carbonic acid, or by nitrogen or sulfur analogues thereof, attached in position 6
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Cephalosporin Compounds (AREA)
Abstract
UN PROCEDIMIENTO PARA LA PREPARACION DE NUEVOS DERIVADOS DE 1,1-DIOXIDO DEL ACIDO PENICILANICO. COMPRENDE SOMETER A REACCION DE ESCISION DEL GRUPO PROTECTOR X DE AMINO Y EL GRUPO PRETECTOR DE CARBOXI EN R>7 SI ESTA PRESENTE, DE UN COMPUESTO (II). SE OBTIENE EL COMPUESTO (I), UNA SAL DE ADICION DE ACIDO FARMACEUTICAMENTE ACEPTABLE O LA SAL DE BASE CORRESPONDIENTE; R>2 SE SELECCIONA DEL GRUPO FORMADO POR ALQUILO CON 1 A 6 CARBONOS, ALCOXI, HOOC-(CH<2)<N-, HOOC-C(CH<3)<2-, CARBOXICICLOPENTILO, 4-CARBOXICICLOHEXILO, R>8R>9N- Y EL GRUPO (III). ACTIVIDAD ANTIBACTERIANA.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US30042181A | 1981-09-09 | 1981-09-09 | |
| US39213982A | 1982-06-28 | 1982-06-28 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES8308568A1 true ES8308568A1 (es) | 1983-09-16 |
| ES515577A0 ES515577A0 (es) | 1983-09-16 |
Family
ID=26971775
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES515577A Granted ES515577A0 (es) | 1981-09-09 | 1982-09-08 | Un procedimiento para la preparacion de nuevos derivados del 1,1-dioxido del acido penicilanico. |
Country Status (16)
| Country | Link |
|---|---|
| EP (1) | EP0074777B1 (es) |
| KR (1) | KR860001363B1 (es) |
| AU (1) | AU535033B2 (es) |
| CA (1) | CA1203797A (es) |
| DE (1) | DE3277456D1 (es) |
| DK (1) | DK162843C (es) |
| ES (1) | ES515577A0 (es) |
| FI (1) | FI77038C (es) |
| GR (1) | GR77006B (es) |
| HU (1) | HU187574B (es) |
| IE (1) | IE53817B1 (es) |
| IL (1) | IL66750A (es) |
| PH (1) | PH18096A (es) |
| PL (1) | PL136237B1 (es) |
| PT (1) | PT75524B (es) |
| YU (1) | YU43278B (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS59502063A (ja) * | 1982-10-26 | 1984-12-13 | ビ−チヤム・グル−プ・ピ−エルシ− | 化学化合物 |
| EP2906661B1 (de) * | 2012-10-11 | 2016-10-26 | Merck Patent GmbH | Materialien für organische elektrolumineszenzvorrichtungen |
| CN112724162B (zh) * | 2020-12-28 | 2022-06-10 | 华南农业大学 | 一种阿莫西林-舒巴坦杂合分子的合成方法及应用 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IE49881B1 (en) * | 1979-02-13 | 1986-01-08 | Leo Pharm Prod Ltd | B-lactam intermediates |
-
1982
- 1982-09-07 EP EP82304673A patent/EP0074777B1/en not_active Expired
- 1982-09-07 DE DE8282304673T patent/DE3277456D1/de not_active Expired
- 1982-09-07 PL PL1982238164A patent/PL136237B1/pl unknown
- 1982-09-08 IE IE2190/82A patent/IE53817B1/en not_active IP Right Cessation
- 1982-09-08 ES ES515577A patent/ES515577A0/es active Granted
- 1982-09-08 GR GR69229A patent/GR77006B/el unknown
- 1982-09-08 AU AU88117/82A patent/AU535033B2/en not_active Expired
- 1982-09-08 CA CA000410940A patent/CA1203797A/en not_active Expired
- 1982-09-08 HU HU822867A patent/HU187574B/hu unknown
- 1982-09-08 IL IL66750A patent/IL66750A/xx not_active IP Right Cessation
- 1982-09-08 DK DK401382A patent/DK162843C/da not_active IP Right Cessation
- 1982-09-08 YU YU2026/82A patent/YU43278B/xx unknown
- 1982-09-08 PT PT75524A patent/PT75524B/pt unknown
- 1982-09-08 FI FI823108A patent/FI77038C/fi not_active IP Right Cessation
- 1982-09-09 KR KR8204087A patent/KR860001363B1/ko not_active Expired
- 1982-09-09 PH PH27841A patent/PH18096A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IE822190L (en) | 1983-03-09 |
| IL66750A (en) | 1985-12-31 |
| FI823108L (fi) | 1983-03-10 |
| IL66750A0 (en) | 1982-12-31 |
| EP0074777B1 (en) | 1987-10-14 |
| CA1203797A (en) | 1986-04-29 |
| FI823108A0 (fi) | 1982-09-08 |
| GR77006B (es) | 1984-09-04 |
| AU8811782A (en) | 1983-03-17 |
| YU43278B (en) | 1989-06-30 |
| DK401382A (da) | 1983-03-10 |
| YU202682A (en) | 1984-12-31 |
| PT75524A (en) | 1982-10-01 |
| DK162843B (da) | 1991-12-16 |
| FI77038B (fi) | 1988-09-30 |
| KR860001363B1 (ko) | 1986-09-16 |
| DE3277456D1 (de) | 1987-11-19 |
| KR840001580A (ko) | 1984-05-07 |
| FI77038C (fi) | 1989-01-10 |
| PH18096A (en) | 1985-03-20 |
| PL238164A1 (en) | 1984-05-07 |
| DK162843C (da) | 1992-05-04 |
| IE53817B1 (en) | 1989-03-01 |
| PL136237B1 (en) | 1986-02-28 |
| EP0074777A1 (en) | 1983-03-23 |
| AU535033B2 (en) | 1984-03-01 |
| PT75524B (en) | 1985-11-25 |
| ES515577A0 (es) | 1983-09-16 |
| HU187574B (en) | 1986-01-28 |
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