ES8307255A1 - Procedimiento para preparar derivados de cefalosporina. - Google Patents

Procedimiento para preparar derivados de cefalosporina.

Info

Publication number
ES8307255A1
ES8307255A1 ES513256A ES513256A ES8307255A1 ES 8307255 A1 ES8307255 A1 ES 8307255A1 ES 513256 A ES513256 A ES 513256A ES 513256 A ES513256 A ES 513256A ES 8307255 A1 ES8307255 A1 ES 8307255A1
Authority
ES
Spain
Prior art keywords
hydrogen atom
formula
image
cephalosporin
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES513256A
Other languages
English (en)
Other versions
ES513256A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Imperial Chemical Industries Ltd
Original Assignee
Imperial Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Imperial Chemical Industries Ltd filed Critical Imperial Chemical Industries Ltd
Publication of ES8307255A1 publication Critical patent/ES8307255A1/es
Publication of ES513256A0 publication Critical patent/ES513256A0/es
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D505/00Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

PROCEDIMIENTO PARA LA OBTENCION DE DERIVADOS DE CEFALOSPORINA Y DE SUS SALES DE ADICION DE ACIDO FISIOLOGICAMENTE COMPATIBLES, DE FORMULA (I), EN LA QUE X ES OXIGENO, AZUFRE O SULFINILO; Y R Y R Y R PUEDEN SER VARIOS TIPOS DE RADICALES. CONSISTE EN LA REACCION DE UN COMPUESTO DE FORMULA (II), O UN DERIVADO DEL MISMO EN EL QUE EL GRUPO CARBONILO ESTA ENMASCARADO, CON UN COMPUESTO DE FORMULA (III), EN LAS QUE R Y R TIENEN UNO DE LOS SIGNIFICADOS DE R Y R ; R ES HIDROGENO O UN GRUPO PROTECTOR, Y X Y R TIENEN EL MISMO SIGNIFICADO QUE EN LA FORMULA (I). LA REACCION SE LLEVA A CABO EN UN DISOLVENTE INERTE, EN PRESENCIA DE UN ACIDO, A UN PH ENTRE 1 Y 4, A UNA TEMPERATURA ENTRE 20 C Y 100 C. ESTOS COMPUESTOS TIENEN APLICACIONES FARMACOLOGICAS COMO ANTIBACTERIALES.
ES513256A 1981-06-19 1982-06-18 Procedimiento para preparar derivados de cefalosporina. Granted ES513256A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8118894 1981-06-19

Publications (2)

Publication Number Publication Date
ES8307255A1 true ES8307255A1 (es) 1983-07-01
ES513256A0 ES513256A0 (es) 1983-07-01

Family

ID=10522636

Family Applications (1)

Application Number Title Priority Date Filing Date
ES513256A Granted ES513256A0 (es) 1981-06-19 1982-06-18 Procedimiento para preparar derivados de cefalosporina.

Country Status (14)

Country Link
US (2) US4497949A (es)
EP (1) EP0072608A3 (es)
JP (1) JPS58985A (es)
AU (1) AU8474382A (es)
CA (1) CA1205465A (es)
DK (1) DK272582A (es)
ES (1) ES513256A0 (es)
FI (1) FI822207L (es)
HU (1) HU187726B (es)
IL (1) IL66080A (es)
NO (1) NO822032L (es)
NZ (1) NZ201012A (es)
PT (1) PT75078B (es)
ZA (1) ZA824094B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA838864B (en) * 1982-12-17 1984-11-28 Ici Pharma Process for the manufacture of cephalosporin derivatives
GB8413152D0 (en) * 1983-06-03 1984-06-27 Ici Pharma Cephalosporin derivatives
US4547573A (en) * 1983-12-02 1985-10-15 Ici Pharma Process for preparing cephalosporin derivatives
JPH09286039A (ja) 1996-04-22 1997-11-04 Komatsu Ltd 板状複合体およびその製造法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2370663A (en) * 1941-11-12 1945-03-06 Koppers Co Inc Organic cyanamide transmissionfluids
US2331671A (en) * 1942-01-31 1943-10-12 American Cyanamid Co Method of preparing monoalkylol cyanamides
US2727068A (en) * 1953-04-10 1955-12-13 Rohm & Haas Vinyloxyalkyl-cyanamides
US3849465A (en) * 1962-11-01 1974-11-19 Du Pont N-cyanoimines and n-cyanoaziridines
NL129625C (es) * 1965-04-14
US4358447A (en) * 1979-04-27 1982-11-09 Merck & Co., Inc. 7-N-Heterocyclyl cephalosporins
FR2472574A1 (fr) * 1979-12-24 1981-07-03 Ici Pharma Derives de cephalosporine et composition pharmaceutique les contenant

Also Published As

Publication number Publication date
JPS58985A (ja) 1983-01-06
EP0072608A2 (en) 1983-02-23
ES513256A0 (es) 1983-07-01
FI822207A0 (fi) 1982-06-18
IL66080A (en) 1986-07-31
EP0072608A3 (en) 1984-04-18
PT75078A (en) 1982-07-01
US4701556A (en) 1987-10-20
ZA824094B (en) 1983-07-27
HU187726B (en) 1986-02-28
DK272582A (da) 1982-12-20
FI822207L (fi) 1982-12-20
CA1205465A (en) 1986-06-03
NO822032L (no) 1982-12-20
PT75078B (en) 1984-10-09
AU8474382A (en) 1982-12-23
US4497949A (en) 1985-02-05
NZ201012A (en) 1986-02-21

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