ES8306727A1 - Un procedimiento para la preparacion de fenilaminoimidazolidinas. - Google Patents

Un procedimiento para la preparacion de fenilaminoimidazolidinas.

Info

Publication number
ES8306727A1
ES8306727A1 ES511665A ES511665A ES8306727A1 ES 8306727 A1 ES8306727 A1 ES 8306727A1 ES 511665 A ES511665 A ES 511665A ES 511665 A ES511665 A ES 511665A ES 8306727 A1 ES8306727 A1 ES 8306727A1
Authority
ES
Spain
Prior art keywords
alkyl
hydrogen
alkoxy
halogen
imidazoline derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES511665A
Other languages
English (en)
Other versions
ES511665A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Beecham Group PLC
Original Assignee
Beecham Group PLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beecham Group PLC filed Critical Beecham Group PLC
Publication of ES8306727A1 publication Critical patent/ES8306727A1/es
Publication of ES511665A0 publication Critical patent/ES511665A0/es
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12—Antidiarrhoeals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/44—Nitrogen atoms not forming part of a nitro radical
    • C07D233/50—Nitrogen atoms not forming part of a nitro radical with carbocyclic radicals directly attached to said nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Abstract

UN PROCEDIMIENTO PARA LA PREPARACION DE FENILAMINOIMIDAZOLIDINAS. CONSTA DE ALGUNA DE LAS SIGUIENTES ETAPAS: 1 ) SOMETER A REACCION A UN COMPUESTO (II) CON R -X. 2 ) SOMETER A REACCION UN COMPUESTO (II) CON H N-CH -CH -NHR . 3 ) SOMETER A REACCION UN COMPUESTO (IV) CON EL (V). 4 ) SOMETER A REACCION UN COMPUESTO (VI) CON R -(CH )M-COZ. SE OBTIENE EL COMPUESTO (I) O UNA SAL DE ADICION DEL MISMO. R ES HALOGENO, ALQUILO O ALCOXI; R ES HIDROGENO, HALOGENO ALQUILO O ALCOXI; R 3 ES UN GRUPO CARBO O HETERO, MONO O BICICLICO; R ES HIDROGENO C O ALQUILO.
ES511665A 1981-04-24 1982-04-23 Un procedimiento para la preparacion de fenilaminoimidazolidinas. Granted ES511665A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8112692 1981-04-24

Publications (2)

Publication Number Publication Date
ES8306727A1 true ES8306727A1 (es) 1983-06-01
ES511665A0 ES511665A0 (es) 1983-06-01

Family

ID=10521338

Family Applications (1)

Application Number Title Priority Date Filing Date
ES511665A Granted ES511665A0 (es) 1981-04-24 1982-04-23 Un procedimiento para la preparacion de fenilaminoimidazolidinas.

Country Status (6)

Country Link
EP (1) EP0070084A3 (es)
JP (1) JPS57181060A (es)
AU (1) AU8293682A (es)
DK (1) DK180182A (es)
ES (1) ES511665A0 (es)
ZA (1) ZA822780B (es)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4461904A (en) * 1981-11-20 1984-07-24 Alcon Laboratories, Inc. 2-(Trisubstituted phenylimino)-imidazolines
EP0107306B1 (en) * 1982-09-16 1986-04-30 Beecham Group Plc Imidazoline derivatives
GB8304593D0 (en) * 1983-02-18 1983-03-23 Beecham Group Plc Amidines
GB8333835D0 (en) * 1983-12-20 1984-02-01 Beecham Group Plc Compounds
US4588737A (en) * 1984-12-20 1986-05-13 Usv Pharmaceutical Corp. Antiallergic bis-imidazolinoamino derivatives
GB8903592D0 (en) * 1989-02-16 1989-04-05 Boots Co Plc Therapeutic agents
CA2196792A1 (en) 1994-08-04 1996-02-15 Yoon T. Jeon Novel benzimidazole derivatives
DE19514579A1 (de) * 1995-04-20 1996-10-24 Boehringer Ingelheim Kg Verwendung von alpha¶1¶¶L¶-Agonisten zur Behandlung der Harninkontinenz
US6495583B1 (en) 1997-03-25 2002-12-17 Synaptic Pharmaceutical Corporation Benzimidazole derivatives
DE10163239A1 (de) * 2001-12-21 2003-07-10 Aventis Pharma Gmbh Substituierte Imidazolidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie enthaltendes Medikament
JP2012227306A (ja) 2011-04-19 2012-11-15 Ngk Insulators Ltd セラミック基板の製造方法
WO2016043260A1 (ja) * 2014-09-19 2016-03-24 塩野義製薬株式会社 環状グアニジンまたはアミジン化合物

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2806775A1 (de) * 1978-02-17 1979-08-30 Boehringer Sohn Ingelheim Neue substituierte 2-phenylimino- imidazolidine deren saeureadditionssalze, diese enthaltende arzneimittel und verfahren zur herstellung derselben
US4287201A (en) * 1980-03-03 1981-09-01 Merck & Co., Inc. Anovulatory method and chicken feed compositions
DE3168754D1 (en) * 1980-07-09 1985-03-21 Beecham Group Plc Clonidine derivatives useful in the treatment of diarrhoea

Also Published As

Publication number Publication date
EP0070084A3 (en) 1983-02-16
JPS57181060A (en) 1982-11-08
ES511665A0 (es) 1983-06-01
AU8293682A (en) 1983-10-27
DK180182A (da) 1982-10-25
EP0070084A2 (en) 1983-01-19
ZA822780B (en) 1983-02-23

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