ES8305714A1 - Procedimiento para la produccion de derivados de piperidile-no - Google Patents
Procedimiento para la produccion de derivados de piperidile-noInfo
- Publication number
- ES8305714A1 ES8305714A1 ES505106A ES505106A ES8305714A1 ES 8305714 A1 ES8305714 A1 ES 8305714A1 ES 505106 A ES505106 A ES 505106A ES 505106 A ES505106 A ES 505106A ES 8305714 A1 ES8305714 A1 ES 8305714A1
- Authority
- ES
- Spain
- Prior art keywords
- production
- pharmaceutical compositions
- compositions containing
- piperidylidene
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/14—Antitussive agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Pulmonology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Immunology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
PROCEDIMIENTO PARA LA PRODUCCION DE UN COMPUESTO DE FORMULA (I), EN LA QUE N ES 2 O 3; R ES UN NUCLEO TRICICLICO; Y R ES HIDROGENO O UN RESIDUO DE ACIDO FISIOLOGICAMENTE ACEPTABLE E HIDROLIZABLE, Y SUS SALES FARMACEUTICAMENTE ACEPTABLES. CONSISTE EN INTRODUCIR UN GRUPO DE FORMULA (II), EN DONDE N TIENE EL SIGNIFICADO YA INDICADO, EN UN COMPUESTO DE FORMULA (III), EN DONDE R ES UN NUCLEO TRICICLICO. DE APLICACION COMO FARMACO PARA EL TRATAMIENTO DEL ASMA ALERGICA Y DE OTROS DESORDENES ALERGICOS.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH660680 | 1980-09-02 |
Publications (2)
Publication Number | Publication Date |
---|---|
ES505106A0 ES505106A0 (es) | 1983-05-01 |
ES8305714A1 true ES8305714A1 (es) | 1983-05-01 |
Family
ID=4312212
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES505106A Expired ES8305714A1 (es) | 1980-09-02 | 1981-09-01 | Procedimiento para la produccion de derivados de piperidile-no |
Country Status (16)
Country | Link |
---|---|
US (1) | US4609664A (es) |
EP (1) | EP0047226B1 (es) |
JP (1) | JPS5777673A (es) |
AT (1) | ATE13297T1 (es) |
AU (1) | AU547111B2 (es) |
CA (1) | CA1166245A (es) |
DE (1) | DE3170504D1 (es) |
DK (1) | DK385681A (es) |
ES (1) | ES8305714A1 (es) |
FI (1) | FI75160C (es) |
IE (1) | IE52182B1 (es) |
IL (1) | IL63698A (es) |
NZ (1) | NZ198220A (es) |
PH (1) | PH16317A (es) |
PT (1) | PT73601B (es) |
ZA (1) | ZA816103B (es) |
Families Citing this family (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4777177A (en) * | 1984-10-19 | 1988-10-11 | Ciba-Geigy Corporation | Pesticidal thioxanthen-9-ylidenepiperidines |
US5089496A (en) * | 1986-10-31 | 1992-02-18 | Schering Corporation | Benzo[5,6]cycloheptapyridine compounds, compositions and method of treating allergies |
US5665726A (en) * | 1986-10-31 | 1997-09-09 | Schering Corporation | Benzo[5,6]cycloheptapyridines, compositions and methods of use |
US5438062A (en) * | 1986-10-31 | 1995-08-01 | Schering Corporation | Benzo(5,6)cycloheptapyridines, compositions and methods of use |
US5104876A (en) * | 1988-04-28 | 1992-04-14 | Schering Corporation | Benzopyrido piperidine, piperidylidene and piperazine compounds, compositions, methods of manufacture and methods of use |
US5231104A (en) * | 1988-07-08 | 1993-07-27 | Pfizer Inc. | 1-arylethyl-3-substituted piperidines |
US5095022A (en) * | 1989-07-04 | 1992-03-10 | Hokuriku Pharmaceutical Co., Ltd. | Piperidine derivatives and pharmaceutical compositions comprising the same |
IL98572A (en) * | 1990-06-22 | 1995-07-31 | Schering Corp | Bite-benzo or benzopyrido compounds Cyclohepta piperidine, piperidylidene and piperazine, preparations and methods of use. |
CA2093797C (en) * | 1990-10-10 | 1998-09-22 | Richard J. Friary | Substituted imidazobenzazepines and imidazopyridoazepines |
WO1992020681A1 (en) * | 1991-05-23 | 1992-11-26 | Schering Corporation | Novel benzopyrido piperidylidene compounds, compositions, methods of manufacture and methods of use |
CA2114009A1 (en) * | 1991-07-23 | 1993-02-04 | Jesse K. Wong | Novel benzopyrido piperidylidene compounds, compositions, methods of manufacture and methods of use |
US5679692A (en) * | 1992-03-27 | 1997-10-21 | Schering Corporation | Unbridged bis-aryl carbinol derivatives, compositions and methods of use |
WO1993020080A1 (en) * | 1992-03-27 | 1993-10-14 | Schering Corporation | Bridged bis-aryl carbinol derivatives, compositions and methods of use |
MX2010005813A (es) * | 2007-11-28 | 2010-06-15 | Nektar Therapeutics | Conjugados oligomero-triciclicos. |
CN101932575B (zh) | 2008-01-30 | 2013-06-12 | 日本脏器制药株式会社 | 哌啶衍生物 |
JP5083989B2 (ja) * | 2008-11-20 | 2012-11-28 | 日本臓器製薬株式会社 | ピペリジン誘導体を含有する医薬 |
WO2011091050A1 (en) * | 2010-01-19 | 2011-07-28 | Nektar Therapeutics | Oligomer-tricyclic conjugates |
ES2624271T3 (es) * | 2010-04-21 | 2017-07-13 | General Electric Technology Gmbh | Método para separar dióxido de carbono de gas de humo de plantas de combustión |
EP2727919B1 (en) * | 2011-06-28 | 2019-05-08 | Fujian Mindong Rejuvenation Pharmaceutical Co., Ltd. | Benzocycloheptanethiophene derivatives for anti-allergic reactions |
CN115960135A (zh) * | 2022-07-21 | 2023-04-14 | 华创合成制药股份有限公司 | 抗组胺类化合物及其制备方法和用途 |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA780441A (en) * | 1968-03-12 | Sandoz Patents Limited | 4 h-benzo (4,5) cyclohepta (1,2-b) thiophene derivatives | |
CA746508A (en) * | 1966-11-15 | D. Marcus Arnold | Dibenzocycloheptenes | |
GB801710A (en) * | 1956-07-02 | 1958-09-17 | Dow Chemical Co | N-polyoxyalkylene derivatives of heterocyclic amines |
FR1488972A (fr) * | 1965-05-25 | 1967-07-21 | Rhone Poulenc Sa | Nouveaux dérivés du dibenzocycloheptatriene et leur préparation |
GB1242169A (en) * | 1969-04-09 | 1971-08-11 | Ucb Sa | Piperidine derivatives |
BE791699A (fr) * | 1971-11-22 | 1973-05-21 | Sandoz Sa | Nouveaux derives du thioxanthene, leur preparation et leur application comme medicaments |
DE2626583A1 (de) * | 1975-06-24 | 1977-01-13 | Sandoz Ag | Neue benzocycloheptathiophenderivate ihre herstellung und ihre verwendung als heilmittel |
GB1570500A (en) * | 1976-01-02 | 1980-07-02 | Sandoz Ltd | Anti-9,10-dihydro-4-(1-methyl-4-piperidylidene)-4h-benzo(4,5) cyclohepta (1,2-b)thiophen-10(9h)-one oxime |
US4128549A (en) * | 1976-02-27 | 1978-12-05 | Sandoz Ltd. | Precursors of 4-(1-alkyl-4-piperidylidene-4H-benzo[4,5]cyclohepta-[1,2-b]thiophen-10(9H)-ones |
US4132796A (en) * | 1977-12-01 | 1979-01-02 | Merck & Co., Inc. | Antipsychotic 3-trifluoromethylsulfinyl analogs of cyproheptadine |
-
1981
- 1981-08-19 AT AT81810337T patent/ATE13297T1/de active
- 1981-08-19 DE DE8181810337T patent/DE3170504D1/de not_active Expired
- 1981-08-19 EP EP81810337A patent/EP0047226B1/en not_active Expired
- 1981-08-26 FI FI812635A patent/FI75160C/fi not_active IP Right Cessation
- 1981-08-31 IL IL63698A patent/IL63698A/xx unknown
- 1981-08-31 AU AU74782/81A patent/AU547111B2/en not_active Ceased
- 1981-08-31 CA CA000384939A patent/CA1166245A/en not_active Expired
- 1981-08-31 PT PT73601A patent/PT73601B/pt unknown
- 1981-08-31 DK DK385681A patent/DK385681A/da not_active Application Discontinuation
- 1981-08-31 NZ NZ198220A patent/NZ198220A/en unknown
- 1981-09-01 JP JP56138298A patent/JPS5777673A/ja active Pending
- 1981-09-01 ES ES505106A patent/ES8305714A1/es not_active Expired
- 1981-09-01 PH PH26131A patent/PH16317A/en unknown
- 1981-09-01 IE IE2012/81A patent/IE52182B1/en unknown
- 1981-09-02 ZA ZA816103A patent/ZA816103B/xx unknown
-
1984
- 1984-07-16 US US06/631,221 patent/US4609664A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
US4609664A (en) | 1986-09-02 |
CA1166245A (en) | 1984-04-24 |
ES505106A0 (es) | 1983-05-01 |
ZA816103B (en) | 1983-04-27 |
PT73601B (en) | 1983-02-28 |
PH16317A (en) | 1983-09-05 |
NZ198220A (en) | 1984-04-27 |
EP0047226A2 (en) | 1982-03-10 |
IL63698A0 (en) | 1981-11-30 |
IL63698A (en) | 1985-06-30 |
DK385681A (da) | 1982-03-03 |
FI75160C (fi) | 1988-05-09 |
FI75160B (fi) | 1988-01-29 |
EP0047226A3 (en) | 1982-05-05 |
AU7478281A (en) | 1982-03-11 |
IE812012L (en) | 1982-03-02 |
FI812635L (fi) | 1982-03-03 |
IE52182B1 (en) | 1987-08-05 |
AU547111B2 (en) | 1985-10-10 |
PT73601A (en) | 1981-09-01 |
DE3170504D1 (en) | 1985-06-20 |
JPS5777673A (en) | 1982-05-15 |
ATE13297T1 (de) | 1985-06-15 |
EP0047226B1 (en) | 1985-05-15 |
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