ES8304986A1 - "un procedimiento para la preparacion de pirrolo (3,4-d)(2)benzacipinas". - Google Patents

"un procedimiento para la preparacion de pirrolo (3,4-d)(2)benzacipinas".

Info

Publication number
ES8304986A1
ES8304986A1 ES513623A ES513623A ES8304986A1 ES 8304986 A1 ES8304986 A1 ES 8304986A1 ES 513623 A ES513623 A ES 513623A ES 513623 A ES513623 A ES 513623A ES 8304986 A1 ES8304986 A1 ES 8304986A1
Authority
ES
Spain
Prior art keywords
radicals
reaction
formula
benzazepines
pyrrolo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES513623A
Other languages
English (en)
Other versions
ES513623A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of ES513623A0 publication Critical patent/ES513623A0/es
Publication of ES8304986A1 publication Critical patent/ES8304986A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyrrole Compounds (AREA)

Abstract

PROCEDIMIENTO PARA LA OBTENCION DE PIRROLO 3,4-D 2 / BENZACEPINAS Y DE SUS SALES DE ADICION DE ACIDO FISIOLOGICAMENTE COMPATIBLES, DE FORMULA (I), EN LA QUE R ES HIDROGENO, FLUOR O CLORO; Y A, R Y R PUEDEN SER VARIOS TIPOS DE RADICALES. CONSISTE EN LA REACCION DE ALQUILACION, ALQUENILACION DE C <- O ALQUINILACION DE C <- EN LAS POSICIONES 1 Y/O 3, UN COMPUESTO DE FORMULA (II), EN LA QUE R , R , R Y R PUEDEN SER VARIOS TIPOS DE RADICALES. LA REACCION SE LLEVA A CABO EN PRESENCIA DE UN EQUIVALENTE DE UNA BASE FUERTE, A UNA TEMPERATURA ENTRE -78 C Y 0 C. ESTOS COMPUESTOS TIENEN APLICACIONES FARMACOLOGICAS COMO AGENTES SEDANTES Y ANXIOLITICOS.
ES513623A 1980-08-05 1982-07-01 "un procedimiento para la preparacion de pirrolo (3,4-d)(2)benzacipinas". Expired ES8304986A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17555580A 1980-08-05 1980-08-05

Publications (2)

Publication Number Publication Date
ES513623A0 ES513623A0 (es) 1983-04-01
ES8304986A1 true ES8304986A1 (es) 1983-04-01

Family

ID=22640700

Family Applications (1)

Application Number Title Priority Date Filing Date
ES513623A Expired ES8304986A1 (es) 1980-08-05 1982-07-01 "un procedimiento para la preparacion de pirrolo (3,4-d)(2)benzacipinas".

Country Status (6)

Country Link
JP (1) JPS5758684A (es)
KR (5) KR850000198B1 (es)
BR (1) BR8105021A (es)
ES (1) ES8304986A1 (es)
GR (1) GR78315B (es)
ZA (1) ZA815193B (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2017357329A1 (en) * 2016-11-10 2019-06-13 Luoxin Pharmaceutical (Shanghai) Co., Ltd. Nitrogenous macrocyclic compound, preparation method therefor, pharmaceutical composition and application thereof

Also Published As

Publication number Publication date
ES513623A0 (es) 1983-04-01
KR850000195B1 (ko) 1985-03-05
KR830006291A (ko) 1983-09-20
KR850000197B1 (ko) 1985-03-05
ZA815193B (en) 1982-07-28
GR78315B (es) 1984-09-26
JPS5758684A (en) 1982-04-08
KR850000194B1 (ko) 1985-03-05
KR850000198B1 (ko) 1985-03-05
BR8105021A (pt) 1982-04-20
KR850000196B1 (ko) 1985-03-05

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