ES8203368A1 - Procedimiento de producir amidas ciclicas - Google Patents
Procedimiento de producir amidas ciclicasInfo
- Publication number
- ES8203368A1 ES8203368A1 ES502064A ES502064A ES8203368A1 ES 8203368 A1 ES8203368 A1 ES 8203368A1 ES 502064 A ES502064 A ES 502064A ES 502064 A ES502064 A ES 502064A ES 8203368 A1 ES8203368 A1 ES 8203368A1
- Authority
- ES
- Spain
- Prior art keywords
- lower alkyl
- integer
- cyclic amides
- hydrogen
- independently
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
- C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D223/16—Benzazepines; Hydrogenated benzazepines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
- C07D217/26—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D279/04—1,3-Thiazines; Hydrogenated 1,3-thiazines
- C07D279/08—1,3-Thiazines; Hydrogenated 1,3-thiazines condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Hydrogenated Pyridines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
Abstract
PROCEDIMIENTO PARA PRODUCIR AMIDAS CICLICAS. CONSISTE EN ACILAR UNA AMINA DE FORMULA GENERAL (I) CON UN ACIDO MERCAPTO O DERIVADO ACILANTE EQUIVALENTE (II). OPCIONALMENTE SE CONVIERTE EL GRUPO -COY EN EL ACIDO LIBRE (Y=OH) O BIEN SE OXIDA EL PRODUCTO EN QUE R5 ES H PARA OBTENER EL BISULFURO O BIEN SE DERIVA EL PRODUCTO EN QUE R5 ES H PARA INTRODUCIR SUSTITUYENTES REPRESENTATIVOS DE R5 DIFERENTES DE H. SE OBTIENE EL COMPUESTO (III).
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US06/148,083 US5200416A (en) | 1980-05-12 | 1980-05-12 | Cyclic amides |
Publications (2)
Publication Number | Publication Date |
---|---|
ES502064A0 ES502064A0 (es) | 1982-04-01 |
ES8203368A1 true ES8203368A1 (es) | 1982-04-01 |
Family
ID=22524186
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES502064A Expired ES8203368A1 (es) | 1980-05-12 | 1981-05-09 | Procedimiento de producir amidas ciclicas |
Country Status (18)
Country | Link |
---|---|
US (1) | US5200416A (es) |
EP (1) | EP0039804B1 (es) |
JP (1) | JPS577470A (es) |
KR (1) | KR850001088B1 (es) |
AT (1) | ATE21511T1 (es) |
AU (1) | AU546218B2 (es) |
DE (1) | DE3175150D1 (es) |
DK (1) | DK206881A (es) |
ES (1) | ES8203368A1 (es) |
FI (1) | FI811424L (es) |
IL (1) | IL62782A0 (es) |
IN (1) | IN152326B (es) |
NO (1) | NO811599L (es) |
NZ (1) | NZ197048A (es) |
SU (1) | SU1304748A3 (es) |
YU (1) | YU120481A (es) |
ZA (1) | ZA812941B (es) |
ZW (1) | ZW10881A1 (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2672598A1 (fr) * | 1991-02-11 | 1992-08-14 | Adir | Nouveaux inhibiteurs de n-myristoyltransferase, leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
AU7724496A (en) * | 1995-11-09 | 1997-05-29 | Monsanto Company | An improved method for preparation of substituted tetrahydroisoquinolines |
US5627282A (en) * | 1996-01-03 | 1997-05-06 | Yukong Limited | Process for the preparation of optically pure 1,2,3,4-tetrahydro-3-isoquinolinecarboxylic acid and its derivatives |
EP2518070A1 (en) * | 2011-04-29 | 2012-10-31 | Almirall, S.A. | Pyrrolotriazinone derivatives as PI3K inhibitors |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5572169A (en) * | 1978-11-27 | 1980-05-30 | Tanabe Seiyaku Co Ltd | Isoquinoline derivative and its preparation |
EP0018104B1 (en) * | 1979-03-26 | 1983-05-25 | Takeda Chemical Industries, Ltd. | Tetrahydroisoquinolines, their production and the compounds and pharmaceutical compositions containing them for use in the prevention or treatment of hypertension |
GB2048863B (en) * | 1979-05-16 | 1983-06-15 | Morton Norwich Products Inc | Tetrahydroisoquinoline-3-carboxylic acids |
DE2937779A1 (de) * | 1979-09-19 | 1981-04-09 | Hoechst Ag, 6000 Frankfurt | Aminosaeurederivate und verfahren zu ihrer herstellung |
FR2487829A2 (fr) * | 1979-12-07 | 1982-02-05 | Science Union & Cie | Nouveaux imino acides substitues, leurs procedes de preparation et leur emploi comme inhibiteur d'enzyme |
US4251444A (en) * | 1980-04-07 | 1981-02-17 | American Home Products Corporation | Thiazepino-[4,3-b]-isoquinoline-1,5-dione derivatives and precursors |
-
1980
- 1980-05-12 US US06/148,083 patent/US5200416A/en not_active Expired - Lifetime
-
1981
- 1981-04-23 AT AT81103072T patent/ATE21511T1/de not_active IP Right Cessation
- 1981-04-23 EP EP81103072A patent/EP0039804B1/en not_active Expired
- 1981-04-23 DE DE8181103072T patent/DE3175150D1/de not_active Expired
- 1981-05-04 IL IL62782A patent/IL62782A0/xx unknown
- 1981-05-04 ZA ZA00812941A patent/ZA812941B/xx unknown
- 1981-05-06 IN IN473/CAL/81A patent/IN152326B/en unknown
- 1981-05-07 ZW ZW108/81A patent/ZW10881A1/xx unknown
- 1981-05-08 FI FI811424A patent/FI811424L/fi not_active Application Discontinuation
- 1981-05-09 ES ES502064A patent/ES8203368A1/es not_active Expired
- 1981-05-11 AU AU70450/81A patent/AU546218B2/en not_active Ceased
- 1981-05-11 DK DK206881A patent/DK206881A/da not_active Application Discontinuation
- 1981-05-11 NZ NZ197048A patent/NZ197048A/en unknown
- 1981-05-11 NO NO811599A patent/NO811599L/no unknown
- 1981-05-11 SU SU813282548A patent/SU1304748A3/ru active
- 1981-05-12 KR KR1019810001634A patent/KR850001088B1/ko active IP Right Grant
- 1981-05-12 JP JP7024181A patent/JPS577470A/ja active Pending
- 1981-05-12 YU YU01204/81A patent/YU120481A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
ATE21511T1 (de) | 1986-09-15 |
FI811424L (fi) | 1981-11-13 |
JPS577470A (en) | 1982-01-14 |
ES502064A0 (es) | 1982-04-01 |
KR830006210A (ko) | 1983-09-20 |
NO811599L (no) | 1981-11-13 |
YU120481A (en) | 1983-12-31 |
IL62782A0 (en) | 1981-07-31 |
KR850001088B1 (ko) | 1985-07-27 |
SU1304748A3 (ru) | 1987-04-15 |
AU546218B2 (en) | 1985-08-22 |
DE3175150D1 (en) | 1986-09-25 |
DK206881A (da) | 1981-11-13 |
IN152326B (es) | 1983-12-17 |
EP0039804B1 (en) | 1986-08-20 |
NZ197048A (en) | 1984-04-27 |
EP0039804A1 (en) | 1981-11-18 |
AU7045081A (en) | 1981-11-19 |
ZA812941B (en) | 1982-05-26 |
US5200416A (en) | 1993-04-06 |
ZW10881A1 (en) | 1981-07-29 |
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