ES8203334A1 - Procedimiento para la obtencion de dehidropeptidos - Google Patents

Procedimiento para la obtencion de dehidropeptidos

Info

Publication number
ES8203334A1
ES8203334A1 ES488301A ES488301A ES8203334A1 ES 8203334 A1 ES8203334 A1 ES 8203334A1 ES 488301 A ES488301 A ES 488301A ES 488301 A ES488301 A ES 488301A ES 8203334 A1 ES8203334 A1 ES 8203334A1
Authority
ES
Spain
Prior art keywords
preparation
compositions containing
phenylalanyl
pharmaceutical compositions
tryptophan derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES488301A
Other languages
English (en)
Other versions
ES488301A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Troponwerke GmbH
Original Assignee
Troponwerke GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Troponwerke GmbH filed Critical Troponwerke GmbH
Publication of ES8203334A1 publication Critical patent/ES8203334A1/es
Publication of ES488301A0 publication Critical patent/ES488301A0/es
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Ultra Sonic Daignosis Equipment (AREA)
  • Measuring Pulse, Heart Rate, Blood Pressure Or Blood Flow (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
  • Indole Compounds (AREA)
  • Flanged Joints, Insulating Joints, And Other Joints (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Liquid Crystal Substances (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)

Abstract

PROCEDIMIENTO PARA LA OBTENCION DE DEHIDROPEPTIDOS. CONSISTE EN HACER REACCIONAR OXAZOLES DE FORMULA GENERAL (I) CON DERIVADOS DE TRIPTOFANO (II) EN PRESENCIA DE DISOLVENTES ORGANICOS, AGUA O MEZCLAS DE AMBOS, A TEMPERATURAS COMPRENDIDAS ENTRE 0 Y 80C. SE OBTIENE EL COMPUESTO (III), EN QUE R1 ES HIDROGENO, ALQUILO U OTROS; R2 ES UN RESTO FENILO; R3 Y R4 SON HIDROGENO; R5 ES HIDROXI O ALCOXI; N VALE 1 O 0; C* ES CENTRO DE ASIMETRIA.
ES488301A 1979-02-07 1980-02-06 Procedimiento para la obtencion de dehidropeptidos Granted ES488301A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19792904512 DE2904512A1 (de) 1979-02-07 1979-02-07 Dehydropeptide, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel

Publications (2)

Publication Number Publication Date
ES8203334A1 true ES8203334A1 (es) 1980-08-01
ES488301A0 ES488301A0 (es) 1980-08-01

Family

ID=6062317

Family Applications (1)

Application Number Title Priority Date Filing Date
ES488301A Granted ES488301A0 (es) 1979-02-07 1980-02-06 Procedimiento para la obtencion de dehidropeptidos

Country Status (13)

Country Link
US (1) US4285935A (es)
EP (1) EP0017705B1 (es)
JP (1) JPS55105654A (es)
AT (1) ATE1352T1 (es)
CA (1) CA1147725A (es)
DE (2) DE2904512A1 (es)
DK (1) DK52080A (es)
ES (1) ES488301A0 (es)
FI (1) FI800350A (es)
GR (1) GR73033B (es)
HU (1) HU181052B (es)
IL (1) IL59295A (es)
NO (1) NO149103B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4350628A (en) * 1979-10-01 1982-09-21 Research Corporation Preparation of dehydropeptides
US4906615A (en) * 1980-12-18 1990-03-06 Schering Corporation Substituted dipeptides as inhibitors of enkephalinases
US4610816A (en) * 1980-12-18 1986-09-09 Schering Corporation Substituted dipeptides as inhibitors of enkephalinases
US4757151A (en) * 1985-11-14 1988-07-12 Warner-Lambert Company 2-substituted-[2-substituted-amino]-N-arylalkyl-3-[indol-3-yl]
DE3823464A1 (de) * 1988-07-11 1990-01-18 Asta Pharma Ag Neue tryptophandipeptide
GB9508195D0 (en) * 1995-04-20 1995-06-07 Univ British Columbia Novel biologically active compounds and compositions,their use and derivation
DE19943508A1 (de) * 1999-09-10 2001-03-15 Morphochem Ag 3-Vinylpyrol-Derivate, Verfahren zu ihrer Herstellung sowie ihre Verwendung als Arzneimittel

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1570140A (en) * 1976-12-28 1980-06-25 Troponwerke Gmbh & Co Kg Tumour-resolving and histolytic medicaments comprising dehydrooligropeptides
NO774303L (no) * 1976-12-28 1978-06-29 Troponwerke Gmbh & Co Kg Nye dehydrooligopeptider, fremgangsmaate til deres fremstilling samt deres anvendelse som legemiddel

Also Published As

Publication number Publication date
IL59295A (en) 1982-12-31
DE3060669D1 (en) 1982-09-09
CA1147725A (en) 1983-06-07
EP0017705A1 (de) 1980-10-29
IL59295A0 (en) 1980-05-30
NO149103B (no) 1983-11-07
ES488301A0 (es) 1980-08-01
NO800151L (no) 1980-08-08
DK52080A (da) 1980-08-08
GR73033B (es) 1984-01-26
JPS55105654A (en) 1980-08-13
HU181052B (en) 1983-05-30
US4285935A (en) 1981-08-25
EP0017705B1 (de) 1982-07-21
DE2904512A1 (de) 1980-08-28
ATE1352T1 (de) 1982-08-15
FI800350A (fi) 1980-08-08

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