ES8201169A1 - Un procedimiento para la preparacion de derivados de quina- zolina - Google Patents
Un procedimiento para la preparacion de derivados de quina- zolinaInfo
- Publication number
- ES8201169A1 ES8201169A1 ES495865A ES495865A ES8201169A1 ES 8201169 A1 ES8201169 A1 ES 8201169A1 ES 495865 A ES495865 A ES 495865A ES 495865 A ES495865 A ES 495865A ES 8201169 A1 ES8201169 A1 ES 8201169A1
- Authority
- ES
- Spain
- Prior art keywords
- intermediates
- preparation
- pharmaceutical use
- quinazoline derivatives
- medicaments containing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pulmonology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Immunology (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
PROCEDIMIENTO PARA LA OBTENCION DE DERIVADOS DE QUINAZOLINA, DE FORMULA (I), Y SUS SALES, DONDE R1 ES METILTIO O METILSULFINILO. CONSISTE EN HIDROLIZAR UN COMPUESTO DE FORMULA (II), DONDE R'' ES UN ALQUILO INFERIOR. LA HIDROLISIS SE LLEVA A CABO EN UN EXCESO DE HIDROXIDO DE METAL ALCALINO, A UNA TEMPERATURA COMPRENDIDA ENTRE 0 Y 30 C, Y MEDIANTE REFLUJO CON UN ACIDO CARBOXILICO ORGANICO. OPCIONALMENTE, PUEDE OXIDARSE EL ACIDO OBTENIDO PARA PRODUCIR LA SAL DEL MISMO. DE APLICACION EN LA PREVENCION DE REACCIONES ALERGICAS.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US06/084,471 US4282360A (en) | 1979-10-12 | 1979-10-12 | 7-Methylthio or methylsulfinyl-5-oxo-5H-thiazolo[2,3-b]quinazoline-2-carboxylic acid |
Publications (2)
Publication Number | Publication Date |
---|---|
ES495865A0 ES495865A0 (es) | 1981-12-01 |
ES8201169A1 true ES8201169A1 (es) | 1981-12-01 |
Family
ID=22185170
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES495865A Expired ES8201169A1 (es) | 1979-10-12 | 1980-10-11 | Un procedimiento para la preparacion de derivados de quina- zolina |
Country Status (17)
Country | Link |
---|---|
US (1) | US4282360A (es) |
EP (1) | EP0027268A3 (es) |
JP (1) | JPS5677288A (es) |
KR (1) | KR830004320A (es) |
AU (1) | AU6319080A (es) |
CA (1) | CA1122216A (es) |
DK (1) | DK426980A (es) |
ES (1) | ES8201169A1 (es) |
FI (1) | FI803214L (es) |
GR (1) | GR70307B (es) |
HU (1) | HU179391B (es) |
IL (1) | IL61240A0 (es) |
MC (1) | MC1356A1 (es) |
NO (1) | NO803058L (es) |
PH (1) | PH15743A (es) |
PT (1) | PT71902B (es) |
ZA (1) | ZA805920B (es) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3142728A1 (de) * | 1981-10-28 | 1983-05-05 | Basf Ag, 6700 Ludwigshafen | Herbizide, enthaltend thiazolo(2,3-b)-chinazolone als wirkstoffe, und ihre verwendung zur beeinflussung des pflanzenwachstums |
DE3142727A1 (de) * | 1981-10-28 | 1983-05-05 | Basf Ag, 6700 Ludwigshafen | Thiazolo (2,3-b)-chinazolone, verfahren zu ihrer herstellung und ihre verwendung zur beeinflussung des pflanzenwachstums |
GB8300728D0 (en) * | 1983-01-12 | 1983-02-16 | Erba Farmitalia | Substituted carboxy-thiazolo / 3 2 - a / pyrimidine derivatives |
US4579132A (en) * | 1983-02-04 | 1986-04-01 | Windmere Corporation | Flocked hair curling roller |
EP0142057A3 (en) * | 1983-11-04 | 1988-03-30 | F. Hoffmann-La Roche Ag | Thiazoloquinazoline derivatives, their preparation and pharmaceutical compositions containing same |
US4738964A (en) * | 1984-05-30 | 1988-04-19 | Pennwalt Corporation | Method of suppressing the immune system comprising administering 5H-thiazolo[2,3-b]quinazoline-3(2H)-one |
US4588812A (en) * | 1984-05-30 | 1986-05-13 | Pennwalt Corporation | Substituted 2,3-dihydro-5H-thiazolo[2,3,-b]quinazoline derivatives |
DE3634532A1 (de) * | 1986-10-10 | 1988-04-14 | Basf Ag | Verfahren zur herstellung von thiazolo-(2,3-b)chinazolonen |
DE10046728C1 (de) * | 2000-09-21 | 2001-09-27 | Ibfb Gmbh Privates Inst Fuer B | Tricyclische mercaptomethylsubstituierte 2,3-Dihydro-chinazolin-5-one und 2,3-Dihydro-benzo[1,2,4,]-thiadiazin-5,5-dioxide als Matrix Metalloproteinase (MMP) Inhibitoren |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2557425A1 (de) * | 1975-12-19 | 1977-06-30 | Boehringer Sohn Ingelheim | Chinazolonderivate |
US4041163A (en) * | 1976-03-29 | 1977-08-09 | Pfizer Inc. | N-(5-Tetrazolyl)-4-oxo-4H-pyrimido(2,1-b)benzothiazole-3-carboxamide antiallergy agents |
US4122274A (en) * | 1977-05-25 | 1978-10-24 | Bristol-Myers Company | 3-Tetrazolo-5,6,7,8-substituted-pyrido[1,2-a]pyrimidin-4-ones |
US4168380A (en) * | 1978-04-21 | 1979-09-18 | Hoffmann-La Roche Inc. | 7-Methoxy-5-oxo-5H-thiazolo[2,3-b]quinazoline-2-carboxylic acid |
-
1979
- 1979-10-12 US US06/084,471 patent/US4282360A/en not_active Expired - Lifetime
-
1980
- 1980-09-24 ZA ZA00805920A patent/ZA805920B/xx unknown
- 1980-10-09 MC MC801478A patent/MC1356A1/xx unknown
- 1980-10-09 GR GR63093A patent/GR70307B/el unknown
- 1980-10-09 PH PH24691A patent/PH15743A/en unknown
- 1980-10-09 IL IL61240A patent/IL61240A0/xx unknown
- 1980-10-09 CA CA000362072A patent/CA1122216A/en not_active Expired
- 1980-10-09 DK DK426980A patent/DK426980A/da unknown
- 1980-10-10 KR KR1019800003887A patent/KR830004320A/ko unknown
- 1980-10-10 FI FI803214A patent/FI803214L/fi not_active Application Discontinuation
- 1980-10-10 HU HU80802470A patent/HU179391B/hu unknown
- 1980-10-10 EP EP80106183A patent/EP0027268A3/de not_active Withdrawn
- 1980-10-10 NO NO803058A patent/NO803058L/no unknown
- 1980-10-10 PT PT71902A patent/PT71902B/pt unknown
- 1980-10-11 JP JP14114880A patent/JPS5677288A/ja active Pending
- 1980-10-11 ES ES495865A patent/ES8201169A1/es not_active Expired
- 1980-10-13 AU AU63190/80A patent/AU6319080A/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
NO803058L (no) | 1981-04-13 |
US4282360A (en) | 1981-08-04 |
EP0027268A3 (de) | 1981-06-17 |
ES495865A0 (es) | 1981-12-01 |
CA1122216A (en) | 1982-04-20 |
IL61240A0 (en) | 1980-12-31 |
PT71902A (en) | 1980-10-31 |
PT71902B (en) | 1982-03-31 |
JPS5677288A (en) | 1981-06-25 |
EP0027268A2 (de) | 1981-04-22 |
KR830004320A (ko) | 1983-07-09 |
HU179391B (en) | 1982-10-28 |
DK426980A (da) | 1981-04-13 |
PH15743A (en) | 1983-03-18 |
ZA805920B (en) | 1981-09-30 |
GR70307B (es) | 1982-09-08 |
MC1356A1 (fr) | 1981-08-10 |
FI803214L (fi) | 1981-04-13 |
AU6319080A (en) | 1981-04-16 |
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