ES8104299A1 - Un procedimiento para oxidar una penicilina a sulfoxido de penicilina - Google Patents

Un procedimiento para oxidar una penicilina a sulfoxido de penicilina

Info

Publication number
ES8104299A1
ES8104299A1 ES489909A ES489909A ES8104299A1 ES 8104299 A1 ES8104299 A1 ES 8104299A1 ES 489909 A ES489909 A ES 489909A ES 489909 A ES489909 A ES 489909A ES 8104299 A1 ES8104299 A1 ES 8104299A1
Authority
ES
Spain
Prior art keywords
penicillin sulfoxides
preparing penicillin
preparing
sulfoxides
nucleus
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES489909A
Other languages
English (en)
Other versions
ES489909A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of ES8104299A1 publication Critical patent/ES8104299A1/es
Publication of ES489909A0 publication Critical patent/ES489909A0/es
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/04—Preparation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

PROCEDIMIENTO PARA OXIDAR UNA PENICILINA A SULFOXIDO DE PENICILINA, DE FORMULA GENERAL: *FORMULA* DONDE R ELEVADO A 1 SE SELECCIONA DEL GRUPO FORMADO POR FENOXIACETILO, BENZOILO, TIENIL-2-ACETILO, FENILGLICILO E HIDROGENO, UN CATION DE METAL ALCALINO Y UN GRUPO PROTECTOR DE ACIDO CARBOXILICO. COMPRENDE HACER REACCIONAR LA PENICILINA EN UN MEDIO ACUOSO A UNA TEMPERATURA COMPRENDIDA ENTRE 0 Y 50GC CON UN PEROXIMONOSULFATO.
ES489909A 1979-03-26 1980-03-25 Un procedimiento para oxidar una penicilina a sulfoxido de penicilina Granted ES489909A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/023,875 US4230620A (en) 1979-03-26 1979-03-26 Process for preparing penicillin sulfoxides

Publications (2)

Publication Number Publication Date
ES8104299A1 true ES8104299A1 (es) 1981-04-16
ES489909A0 ES489909A0 (es) 1981-04-16

Family

ID=21817696

Family Applications (1)

Application Number Title Priority Date Filing Date
ES489909A Granted ES489909A0 (es) 1979-03-26 1980-03-25 Un procedimiento para oxidar una penicilina a sulfoxido de penicilina

Country Status (23)

Country Link
US (1) US4230620A (es)
EP (1) EP0017419A1 (es)
JP (1) JPS55130982A (es)
KR (1) KR830001968B1 (es)
AR (1) AR225170A1 (es)
AU (1) AU5672980A (es)
BE (1) BE882356A (es)
CS (1) CS212343B2 (es)
DD (1) DD149668A5 (es)
DK (1) DK127680A (es)
ES (1) ES489909A0 (es)
FI (1) FI800872A (es)
FR (1) FR2452492A1 (es)
GB (1) GB2047245A (es)
GR (1) GR68012B (es)
IL (1) IL59685A0 (es)
IT (1) IT1130076B (es)
LU (1) LU82290A1 (es)
PH (1) PH14454A (es)
PL (1) PL222865A1 (es)
PT (1) PT70982A (es)
YU (1) YU81180A (es)
ZA (1) ZA801621B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL70221A0 (en) * 1982-11-16 1984-02-29 Lilly Co Eli Process for sulfones
US4502988A (en) * 1983-08-08 1985-03-05 Eli Lilly And Company Oxidation process
DE3432365A1 (de) * 1984-09-03 1986-03-13 Deutsche Bp Ag, 2000 Hamburg Brennstoff auf basis von kohle
CA1256426A (en) * 1985-09-06 1989-06-27 Jacobus J. Bos Process for the preparation of 6-amino-penicillanic acid 1,1 dioxide by oxidation of 6-amino penicillanic acid,
US5604222A (en) * 1993-12-27 1997-02-18 Lupin Laboratories, Ltd. Method for the preparation of 2-chloro sulfinyl azetidinones
US5578721A (en) * 1994-07-11 1996-11-26 Lupin Laboratories Limited Process for preparation of 3-exomethylene cepham sulfoxide esters
CN102964355B (zh) * 2012-12-17 2015-07-01 华北制药河北华民药业有限责任公司 一种青霉素g亚砜的制备方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3197466A (en) * 1961-10-30 1965-07-27 Smith Kline French Lab Penicillin sulfoxides and process
US3544581A (en) * 1965-07-22 1970-12-01 Bristol Myers Co Production of 6-amino-penicillanic acid sulfoxide
US3586667A (en) * 1967-12-22 1971-06-22 Lilly Co Eli Penicillin esterification process
GB1442993A (en) * 1972-07-18 1976-07-21 Gist Brocades Nv Penicillin and cephalosporin r-sulphoxides
US4052387A (en) * 1974-12-24 1977-10-04 Eli Lilly And Company Method of preparation of 3-methylenecephams
CA1069126A (en) * 1974-12-24 1980-01-01 Eli Lilly And Company Sulfinyl halides and their preparation from penicillin sulfoxides
PL95709B1 (pl) * 1975-01-28 1977-11-30 Sposob wytwarzania selfotlenkow estrow penicylin

Also Published As

Publication number Publication date
BE882356A (fr) 1980-09-22
YU81180A (en) 1983-02-28
FI800872A (fi) 1980-09-27
IT1130076B (it) 1986-06-11
EP0017419A1 (en) 1980-10-15
DD149668A5 (de) 1981-07-22
CS212343B2 (en) 1982-03-26
KR830001948A (ko) 1983-05-21
JPS55130982A (en) 1980-10-11
US4230620A (en) 1980-10-28
PT70982A (en) 1980-04-01
AU5672980A (en) 1980-10-02
IL59685A0 (en) 1980-06-30
ZA801621B (en) 1981-10-28
PH14454A (en) 1981-07-23
AR225170A1 (es) 1982-02-26
DK127680A (da) 1980-09-27
FR2452492A1 (fr) 1980-10-24
ES489909A0 (es) 1981-04-16
GR68012B (es) 1981-10-26
GB2047245A (en) 1980-11-26
IT8020873A0 (it) 1980-03-24
LU82290A1 (fr) 1980-07-01
KR830001968B1 (ko) 1983-09-29
PL222865A1 (es) 1980-12-01

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