ES8103053A1 - Un procedimiento para preparar derivados de 2-imidazolina - Google Patents

Un procedimiento para preparar derivados de 2-imidazolina

Info

Publication number
ES8103053A1
ES8103053A1 ES490292A ES490292A ES8103053A1 ES 8103053 A1 ES8103053 A1 ES 8103053A1 ES 490292 A ES490292 A ES 490292A ES 490292 A ES490292 A ES 490292A ES 8103053 A1 ES8103053 A1 ES 8103053A1
Authority
ES
Spain
Prior art keywords
preparation
same
pharmaceutical composition
imidazoline derivatives
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES490292A
Other languages
English (en)
Other versions
ES490292A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Fujisawa Pharmaceutical Co Ltd
Original Assignee
Fujisawa Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fujisawa Pharmaceutical Co Ltd filed Critical Fujisawa Pharmaceutical Co Ltd
Publication of ES8103053A1 publication Critical patent/ES8103053A1/es
Publication of ES490292A0 publication Critical patent/ES490292A0/es
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/44—Nitrogen atoms not forming part of a nitro radical
    • C07D233/50—Nitrogen atoms not forming part of a nitro radical with carbocyclic radicals directly attached to said nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

PROCEDIMIENTO PARA PREPARAR DERIVDOS DE 2-IMIDAZOLINA DE FORMULA *FORMULA* DONDE R1, R2 Y R3 SON DISTINTOS TIPOS DE ATOMOS O RADICALES SE OBTIENE HACIENDO REACCIOAR DISTINTOS COMPUESTOS DE FORMULA GENERAL: *FORMULA* CON ETILENDIAMINA O UNA SAL DE LA MISMA, CON UN COMPUESTO DE FORMULA: CON NITRO O CON AMINO, SIENDO R1 Y X DISTINTOS TIPOS RADICALES. ESTOS DERIVADOS POSEEN ACTIVIDADES ANTIHIPERTENSORAS, ANTIINFLAMATORIAS, ANALGESICAS Y ANTIULCERA. M
ES490292A 1979-04-03 1980-04-02 Un procedimiento para preparar derivados de 2-imidazolina Granted ES490292A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7911537 1979-04-03

Publications (2)

Publication Number Publication Date
ES8103053A1 true ES8103053A1 (es) 1981-02-16
ES490292A0 ES490292A0 (es) 1981-02-16

Family

ID=10504284

Family Applications (1)

Application Number Title Priority Date Filing Date
ES490292A Granted ES490292A0 (es) 1979-04-03 1980-04-02 Un procedimiento para preparar derivados de 2-imidazolina

Country Status (13)

Country Link
EP (1) EP0017484B1 (es)
JP (1) JPS55136266A (es)
AR (1) AR227556A1 (es)
AT (1) ATE2953T1 (es)
AU (1) AU535979B2 (es)
CA (1) CA1138451A (es)
DE (1) DE3062586D1 (es)
DK (1) DK142480A (es)
ES (1) ES490292A0 (es)
GR (1) GR66816B (es)
HU (1) HU184259B (es)
PH (1) PH15980A (es)
ZA (1) ZA801680B (es)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2521140A1 (fr) * 1982-02-05 1983-08-12 Synthelabo Derives d'imidazolidine, leur preparation et leur application en therapeutique
US4880838A (en) * 1982-06-30 1989-11-14 Rhone-Poulenc Pesticidal 1-(4-Phenoxyphenyl)-5-Benzoyl urea compounds and process for preparation
US4665097A (en) * 1983-03-31 1987-05-12 Union Carbide Corporation Novel bicyclooxyaryl thioureas and process for preparation
US4873264A (en) * 1983-05-20 1989-10-10 Rhone-Poulenc Nederlands B.V. Novel pesticidal 1-(alkyl-phenoxy-aryl)-3-benzoyl ureas and process for preparation
US4638088A (en) * 1984-11-15 1987-01-20 Union Carbide Corporation Pesticidal biphenylyloxy and biphenylylalkoxy aryl acyl urea compounds
GB8827152D0 (en) * 1988-11-21 1988-12-29 Wellcome Found Anti-atherosclerotic diaryl compounds
US5290814A (en) * 1988-11-21 1994-03-01 Burroughs Wellcome Co. Anti-atherosclerotic diaryl compounds
GB8903592D0 (en) * 1989-02-16 1989-04-05 Boots Co Plc Therapeutic agents
US5001157A (en) * 1989-02-02 1991-03-19 American Cyanamid Company Substituted N-[[2-(aminocarbonyl)phenylamino]thioxomethyl]benzamides
IN172842B (es) * 1990-05-17 1993-12-11 Boots Pharmaceuticals Limited
JPH0440953A (ja) * 1990-06-05 1992-02-12 Kyodo Sekkei:Kk 注射針処理方法及びその装置
CN1037346C (zh) * 1990-06-29 1998-02-11 布茨公司 降血糖的脒类和胍类的制备方法
SG72827A1 (en) * 1997-06-23 2000-05-23 Hoffmann La Roche Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives
NZ331480A (en) * 1997-09-04 2000-02-28 F 2-(Arylphenyl)amino-imidazoline derivatives and pharmaceutical compositions
US6184242B1 (en) 1997-09-04 2001-02-06 Syntex Usa (Llc) 2-(substituted-phenyl)amino-imidazoline derivatives
US6417186B1 (en) 2000-11-14 2002-07-09 Syntex (U.S.A.) Llc Substituted-phenyl ketone derivatives as IP antagonists
EP1622611A1 (en) 2003-05-01 2006-02-08 F. Hoffmann-La Roche Ag Imidazolin-2-ylaminophenyl amides as ip antagonists
EP1656350A2 (en) * 2003-07-09 2006-05-17 F.Hoffmann-La Roche Ag Thiophenylaminoimidazolines as prostaglandin i2 antagonists
JP2007523868A (ja) * 2003-07-10 2007-08-23 アキリオン ファーマシューティカルズ，インコーポレーテッド ウイルス複製の阻害薬として有用な置換アリールチオウレア誘導体類
PE20060493A1 (es) * 2004-10-05 2006-09-03 Smithkline Beecham Corp Compuestos derivados de bifenil (di o tri) carboxamidas como inhibidores de serina/treonina quinasa p38
DE102005007160A1 (de) * 2005-02-16 2006-08-24 Basf Ag Pyrazolcarbonsäureanilide, Verfahren zu ihrer Herstellung und sie enthaltende Mittel zur Bekämpfung von Schadpilzen

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB889706A (en) * 1960-07-16 1962-02-21 Thomas Adam Clayton Fungicidal composition
DE2446758C3 (de) * 1974-10-01 1979-01-04 C.H. Boehringer Sohn, 6507 Ingelheim 2-(2-Fluor-6-trifluormethylphenylimino)-imidazolidin, dessen Säureadditionssalze, Verfahren zur Herstellung dieser Verbindungen und deren Verwendung bei der Bekämpfung der Hypertonie

Also Published As

Publication number Publication date
EP0017484B1 (en) 1983-04-06
JPH0210830B2 (es) 1990-03-09
JPS55136266A (en) 1980-10-23
ZA801680B (en) 1981-03-25
DE3062586D1 (en) 1983-05-11
CA1138451A (en) 1982-12-28
AU535979B2 (en) 1984-04-12
PH15980A (en) 1983-05-16
GR66816B (es) 1981-04-30
AU5689280A (en) 1980-10-09
HU184259B (en) 1984-07-30
EP0017484A1 (en) 1980-10-15
AR227556A1 (es) 1982-11-15
DK142480A (da) 1980-10-04
ATE2953T1 (de) 1983-04-15
ES490292A0 (es) 1981-02-16

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