ES8102120A1 - Procedimiento para la obtencion de derivados de pirazol - Google Patents
Procedimiento para la obtencion de derivados de pirazolInfo
- Publication number
- ES8102120A1 ES8102120A1 ES488717A ES488717A ES8102120A1 ES 8102120 A1 ES8102120 A1 ES 8102120A1 ES 488717 A ES488717 A ES 488717A ES 488717 A ES488717 A ES 488717A ES 8102120 A1 ES8102120 A1 ES 8102120A1
- Authority
- ES
- Spain
- Prior art keywords
- pyrazole derivatives
- production
- pharmaceutical preparations
- preparations containing
- phenylpiperazino
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pain & Pain Management (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Rheumatology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
PROCEDIMIENTO PARA LA OBTENCION DE DERIVADOS DE PIRAZOL, DE FORMULA (I): EN LA QUE R ELEVADO A 1 SIGNIFICA H O C1; R ELEVADO A 2 SIGNIFICA 1-METIL-4-PIPERIDILOXICARBONILO, 2-(4-FENILPIPERAZINO). CARACTERIZADO PORQUE SE HACE REACCIONAR UN COMPUESTO DE FORMULA GENERAL (II): *FORMULA* O UNO DE SUS DERIVADOS REACTIVOS, CON FENILHIDRAZINA O UNA DE SUS SALES; TAMBIEN SE REVINDICAN OTROS PROCEDIMIENTOS DE OBTENCION. ESTOS DERIVADOS SE EMPLEAN EN LA MEDICINA HUMANA O ANIMAL.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19792906252 DE2906252A1 (de) | 1979-02-19 | 1979-02-19 | Pyrazolderivate, diese enthaltende pharmazeutische zubereitungen und verfahren zu ihrer herstellung |
Publications (2)
Publication Number | Publication Date |
---|---|
ES488717A0 ES488717A0 (es) | 1980-12-16 |
ES8102120A1 true ES8102120A1 (es) | 1980-12-16 |
Family
ID=6063264
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES488717A Expired ES8102120A1 (es) | 1979-02-19 | 1980-02-18 | Procedimiento para la obtencion de derivados de pirazol |
Country Status (8)
Country | Link |
---|---|
US (1) | US4258047A (es) |
EP (1) | EP0014847A1 (es) |
JP (1) | JPS55120583A (es) |
AU (1) | AU5556280A (es) |
DE (1) | DE2906252A1 (es) |
ES (1) | ES8102120A1 (es) |
IL (1) | IL59410A0 (es) |
ZA (1) | ZA80922B (es) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4826868A (en) * | 1986-05-29 | 1989-05-02 | Ortho Pharmaceutical Corporation | 1,5-Diaryl-3-substituted pyrazoles pharmaceutical compositions and use |
AU611437B2 (en) * | 1987-05-29 | 1991-06-13 | Ortho Pharmaceutical Corporation | Pharmacologically active 2- and 3-substituted (1',5'-diaryl-3-pyrazolyl)-n-hydroxypropanamides and method for synthesizing the same |
PH27357A (en) * | 1989-09-22 | 1993-06-21 | Fujisawa Pharmaceutical Co | Pyrazole derivatives and pharmaceutical compositions comprising the same |
GB9714303D0 (en) * | 1997-07-07 | 1997-09-10 | Pharmacia & Upjohn Spa | 5-(3-phenyl-3-oxo-propyl)-1H-tetrazole derivatives |
DE10149370A1 (de) * | 2001-10-06 | 2003-04-10 | Merck Patent Gmbh | Pyrazolderivate |
AU2003275637A1 (en) * | 2002-10-24 | 2004-05-13 | Wakamoto Pharmaceutical Co., Ltd. | Pyrazole-4-alkanoate derivatives inhibiting cyclooxygenase and 5-lipoxygenase |
DE10315572A1 (de) * | 2003-04-05 | 2004-10-14 | Merck Patent Gmbh | Substituierte Pyrazole |
DE10315571A1 (de) | 2003-04-05 | 2004-10-14 | Merck Patent Gmbh | Pyrazolverbindungen |
DE10315569A1 (de) | 2003-04-05 | 2004-10-14 | Merck Patent Gmbh | Substituierte Pyrazolverbindungen |
DE10315573A1 (de) | 2003-04-05 | 2004-10-14 | Merck Patent Gmbh | Substituierte Pyrazole |
CN101528740B (zh) * | 2006-09-29 | 2012-09-19 | 株式会社绿十字 | 作为大麻素cb1受体拮抗剂的杂芳基-吡唑衍生物 |
WO2009078498A1 (en) * | 2007-12-17 | 2009-06-25 | Green Cross Corporation | Biarylpyrazole 4-carboxamides as cannabinoid cb1 receptor ligands |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE663344A (es) * | 1964-05-04 | |||
DE1595920B2 (de) * | 1964-11-04 | 1978-08-10 | Merck Patent Gmbh, 6100 Darmstadt | 4-(co-Piperazinoalkyl)-pyrazole, ihre Salze und Verfahren zu ihrer Herstellung |
CH535777A (de) * | 1967-03-01 | 1973-04-15 | Ciba Geigy Ag | Verfahren zur Herstellung neuer azacycloaliphatischer Verbindungen |
BE755924A (fr) * | 1969-09-12 | 1971-02-15 | Byk Gulden Lomberg Chem Fab | Derives d'acide pyrazole-4-acetique, leur procede de preparation et medicaments en contenant |
DE2526469A1 (de) * | 1975-06-13 | 1976-12-30 | Bayer Ag | 1-substituierte pyrazolderivate, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel |
-
1979
- 1979-02-19 DE DE19792906252 patent/DE2906252A1/de not_active Withdrawn
-
1980
- 1980-01-22 EP EP80100294A patent/EP0014847A1/de not_active Withdrawn
- 1980-02-14 AU AU55562/80A patent/AU5556280A/en not_active Abandoned
- 1980-02-18 IL IL59410A patent/IL59410A0/xx unknown
- 1980-02-18 ES ES488717A patent/ES8102120A1/es not_active Expired
- 1980-02-18 ZA ZA00800922A patent/ZA80922B/xx unknown
- 1980-02-19 US US06/122,795 patent/US4258047A/en not_active Expired - Lifetime
- 1980-02-19 JP JP1862280A patent/JPS55120583A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
EP0014847A1 (de) | 1980-09-03 |
IL59410A0 (en) | 1980-05-30 |
ES488717A0 (es) | 1980-12-16 |
JPS55120583A (en) | 1980-09-17 |
ZA80922B (en) | 1981-02-25 |
US4258047A (en) | 1981-03-24 |
AU5556280A (en) | 1980-08-28 |
DE2906252A1 (de) | 1980-08-28 |
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