ZA80922B - Pyrazole derivatives pharmaceutical formulations containing these derivatives and processes for their preparation - Google Patents

Pyrazole derivatives pharmaceutical formulations containing these derivatives and processes for their preparation

Info

Publication number
ZA80922B
ZA80922B ZA00800922A ZA80922A ZA80922B ZA 80922 B ZA80922 B ZA 80922B ZA 00800922 A ZA00800922 A ZA 00800922A ZA 80922 A ZA80922 A ZA 80922A ZA 80922 B ZA80922 B ZA 80922B
Authority
ZA
South Africa
Prior art keywords
derivatives
processes
preparation
pharmaceutical formulations
formulations containing
Prior art date
Application number
ZA00800922A
Other languages
English (en)
Inventor
Klockow
H Radunz
J Gante
K Minck
D Orth
A Wild
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of ZA80922B publication Critical patent/ZA80922B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
ZA00800922A 1979-02-19 1980-02-18 Pyrazole derivatives pharmaceutical formulations containing these derivatives and processes for their preparation ZA80922B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19792906252 DE2906252A1 (de) 1979-02-19 1979-02-19 Pyrazolderivate, diese enthaltende pharmazeutische zubereitungen und verfahren zu ihrer herstellung

Publications (1)

Publication Number Publication Date
ZA80922B true ZA80922B (en) 1981-02-25

Family

ID=6063264

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA00800922A ZA80922B (en) 1979-02-19 1980-02-18 Pyrazole derivatives pharmaceutical formulations containing these derivatives and processes for their preparation

Country Status (8)

Country Link
US (1) US4258047A (es)
EP (1) EP0014847A1 (es)
JP (1) JPS55120583A (es)
AU (1) AU5556280A (es)
DE (1) DE2906252A1 (es)
ES (1) ES8102120A1 (es)
IL (1) IL59410A0 (es)
ZA (1) ZA80922B (es)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4826868A (en) * 1986-05-29 1989-05-02 Ortho Pharmaceutical Corporation 1,5-Diaryl-3-substituted pyrazoles pharmaceutical compositions and use
AU611437B2 (en) * 1987-05-29 1991-06-13 Ortho Pharmaceutical Corporation Pharmacologically active 2- and 3-substituted (1',5'-diaryl-3-pyrazolyl)-n-hydroxypropanamides and method for synthesizing the same
PH27357A (en) * 1989-09-22 1993-06-21 Fujisawa Pharmaceutical Co Pyrazole derivatives and pharmaceutical compositions comprising the same
GB9714303D0 (en) * 1997-07-07 1997-09-10 Pharmacia & Upjohn Spa 5-(3-phenyl-3-oxo-propyl)-1H-tetrazole derivatives
DE10149370A1 (de) * 2001-10-06 2003-04-10 Merck Patent Gmbh Pyrazolderivate
AU2003275637A1 (en) * 2002-10-24 2004-05-13 Wakamoto Pharmaceutical Co., Ltd. Pyrazole-4-alkanoate derivatives inhibiting cyclooxygenase and 5-lipoxygenase
DE10315572A1 (de) * 2003-04-05 2004-10-14 Merck Patent Gmbh Substituierte Pyrazole
DE10315571A1 (de) 2003-04-05 2004-10-14 Merck Patent Gmbh Pyrazolverbindungen
DE10315569A1 (de) 2003-04-05 2004-10-14 Merck Patent Gmbh Substituierte Pyrazolverbindungen
DE10315573A1 (de) 2003-04-05 2004-10-14 Merck Patent Gmbh Substituierte Pyrazole
CN101528740B (zh) * 2006-09-29 2012-09-19 株式会社绿十字 作为大麻素cb1受体拮抗剂的杂芳基-吡唑衍生物
WO2009078498A1 (en) * 2007-12-17 2009-06-25 Green Cross Corporation Biarylpyrazole 4-carboxamides as cannabinoid cb1 receptor ligands

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE663344A (es) * 1964-05-04
DE1595920B2 (de) * 1964-11-04 1978-08-10 Merck Patent Gmbh, 6100 Darmstadt 4-(co-Piperazinoalkyl)-pyrazole, ihre Salze und Verfahren zu ihrer Herstellung
CH535777A (de) * 1967-03-01 1973-04-15 Ciba Geigy Ag Verfahren zur Herstellung neuer azacycloaliphatischer Verbindungen
BE755924A (fr) * 1969-09-12 1971-02-15 Byk Gulden Lomberg Chem Fab Derives d'acide pyrazole-4-acetique, leur procede de preparation et medicaments en contenant
DE2526469A1 (de) * 1975-06-13 1976-12-30 Bayer Ag 1-substituierte pyrazolderivate, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel

Also Published As

Publication number Publication date
EP0014847A1 (de) 1980-09-03
IL59410A0 (en) 1980-05-30
ES488717A0 (es) 1980-12-16
ES8102120A1 (es) 1980-12-16
JPS55120583A (en) 1980-09-17
US4258047A (en) 1981-03-24
AU5556280A (en) 1980-08-28
DE2906252A1 (de) 1980-08-28

Similar Documents

Publication Publication Date Title
IL60129A0 (en) Phenylsulphonamide derivatives,their preparation and pharmaceutical compositions containing them
MY8700186A (en) 3-aminopropoxyaryl derivatives their preparation and pharmaceutical compositions containing them
SG20887G (en) Trans-quinazoline derivatives processes for their preparation intermediates and medicaments containing these derivatives
IL61481A0 (en) Piperidylbenzimidazolinone derivatives,their preparation and pharmaceutical compositions containing them
IL60470A0 (en) Imidazole derivatives,their preparation and pharmaceutical compositions containing them
ZA80922B (en) Pyrazole derivatives pharmaceutical formulations containing these derivatives and processes for their preparation
GB2043644B (en) 3-phosphonocephalosporanic acid derivatives process for preparation thereof and pharmaceutical composition comprising the same
GB2063874B (en) Triazole derivatives processes for the preparation thereof and pharmaceutical compositions containing them
NZ193078A (en) Derivatives of 9-aminoalkyl-flyorene medicinal preparations
IL57599A0 (en) Indolealkylamines,pharmaceutical formulations containing these and processes for their preparation
GB2047238B (en) Triazole derivatives processes for their production and pharmaceutical compositions containing them
DE3065460D1 (en) Benzocycloheptapyrrolealkanoic acids and their derivatives, processes for their preparation and pharmaceutical compositions containing them
IL60376A0 (en) 3-methyleneazetidine derivatives and pharmaceutical compositions containing them
GB2063253B (en) Triazole derivatives processes for their production and pharmaceutical compositions containing them
IL60058A0 (en) Hydroxyamino-eburnane derivatives,their preparation and pharmaceutical compositions containing them
IL60359A (en) Dialkylaminoalkoxyiminocycloalkane derivatives,their preparation and pharmaceutical compositions containing them
ZA793131B (en) Indolealkylamines,pharmaceutical formulations containing these,and processes for their preparation
DE3173933D1 (en) Pyrazoline derivatives, processes for their preparation and pharmaceutical formulations containing them
DE3062972D1 (en) Pyridazopyridazine derivatives, processes for their preparation and pharmaceutical compositions containing these pyridazopyridazine derivatives
DE3062531D1 (en) Pyrrolidine derivatives, processes for their preparation and pharmaceutical compositions containing them
IL60927A (en) Amino-propanoloxytetrahydroquinoline derivatives,their preparation and pharmaceutical compositions containing them
DE2860796D1 (en) Tantomeric arylaminoimidazoline derivatives, their preparation and pharmaceutical formulations for analgetic application containing them
IL60548A0 (en) Ergol-8-ene and ergolin derivatives,their preparation and pharmaceutical compositions containing them
IL61675A0 (en) N-substituted -amino acids and derivatives thereof,their preparation and pharmaceutical compositions containing them
IL60040A0 (en) Imidazole derivatives and pharmaceutical compositions containing them