ES531530A0 - Un procedimiento para la preparacion de nuevas cefalosporinas. - Google Patents

Un procedimiento para la preparacion de nuevas cefalosporinas.

Info

Publication number
ES531530A0
ES531530A0 ES531530A ES531530A ES531530A0 ES 531530 A0 ES531530 A0 ES 531530A0 ES 531530 A ES531530 A ES 531530A ES 531530 A ES531530 A ES 531530A ES 531530 A0 ES531530 A0 ES 531530A0
Authority
ES
Spain
Prior art keywords
procedure
preparation
new cephalosporins
cephalosporins
new
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES531530A
Other languages
English (en)
Spanish (es)
Other versions
ES8600307A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/484,128 external-priority patent/US4490370A/en
Priority claimed from US06/516,220 external-priority patent/US4474780A/en
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of ES8600307A1 publication Critical patent/ES8600307A1/es
Publication of ES531530A0 publication Critical patent/ES531530A0/es
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/227-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with radicals containing only hydrogen and carbon atoms, attached in position 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/26Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group
    • C07D501/28Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group with the 7-amino radical acylated by an aliphatic carboxylic acid, which is substituted by hetero atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/59Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3 with hetero atoms directly attached in position 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Peptides Or Proteins (AREA)
ES531530A 1983-04-12 1984-04-11 Un procedimiento para la preparacion de nuevas cefalosporinas. Granted ES531530A0 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US06/484,128 US4490370A (en) 1983-04-12 1983-04-12 Naphthylglycyl cephalosporin derivatives
US06/516,220 US4474780A (en) 1983-07-22 1983-07-22 Crystalline cephalosporin
US53805083A 1983-09-30 1983-09-30

Publications (2)

Publication Number Publication Date
ES8600307A1 ES8600307A1 (es) 1985-10-01
ES531530A0 true ES531530A0 (es) 1985-10-01

Family

ID=27413675

Family Applications (1)

Application Number Title Priority Date Filing Date
ES531530A Granted ES531530A0 (es) 1983-04-12 1984-04-11 Un procedimiento para la preparacion de nuevas cefalosporinas.

Country Status (12)

Country Link
DD (1) DD216240A5 (enrdf_load_html_response)
DK (1) DK187484A (enrdf_load_html_response)
ES (1) ES531530A0 (enrdf_load_html_response)
FI (1) FI841438A7 (enrdf_load_html_response)
GR (1) GR79909B (enrdf_load_html_response)
HU (1) HUT34497A (enrdf_load_html_response)
IL (1) IL71500A0 (enrdf_load_html_response)
MA (1) MA20094A1 (enrdf_load_html_response)
NO (1) NO841442L (enrdf_load_html_response)
OA (1) OA07702A (enrdf_load_html_response)
PT (1) PT78405A (enrdf_load_html_response)
ZW (1) ZW4484A1 (enrdf_load_html_response)

Also Published As

Publication number Publication date
DD216240A5 (de) 1984-12-05
ZW4484A1 (en) 1984-10-03
PT78405A (en) 1984-05-01
GR79909B (enrdf_load_html_response) 1984-10-31
OA07702A (fr) 1985-08-30
NO841442L (no) 1984-10-15
DK187484A (da) 1984-11-23
IL71500A0 (en) 1984-07-31
ES8600307A1 (es) 1985-10-01
HUT34497A (en) 1985-03-28
FI841438A0 (fi) 1984-04-11
MA20094A1 (fr) 1984-12-31
FI841438A7 (fi) 1984-10-13
DK187484D0 (da) 1984-04-11

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