ES536728A0 - Un procedimiento para la preparacion de nuevos antibioticos de cefalosporina. - Google Patents

Un procedimiento para la preparacion de nuevos antibioticos de cefalosporina.

Info

Publication number
ES536728A0
ES536728A0 ES536728A ES536728A ES536728A0 ES 536728 A0 ES536728 A0 ES 536728A0 ES 536728 A ES536728 A ES 536728A ES 536728 A ES536728 A ES 536728A ES 536728 A0 ES536728 A0 ES 536728A0
Authority
ES
Spain
Prior art keywords
procedure
preparation
cephalosporin antibiotics
new cephalosporin
new
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES536728A
Other languages
English (en)
Other versions
ES8602816A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of ES8602816A1 publication Critical patent/ES8602816A1/es
Publication of ES536728A0 publication Critical patent/ES536728A0/es
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/48Methylene radicals, substituted by hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
ES536728A 1983-10-17 1984-10-11 Un procedimiento para la preparacion de nuevos antibioticos de cefalosporina. Granted ES536728A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US54261983A 1983-10-17 1983-10-17

Publications (2)

Publication Number Publication Date
ES8602816A1 ES8602816A1 (es) 1985-11-16
ES536728A0 true ES536728A0 (es) 1985-11-16

Family

ID=24164603

Family Applications (1)

Application Number Title Priority Date Filing Date
ES536728A Granted ES536728A0 (es) 1983-10-17 1984-10-11 Un procedimiento para la preparacion de nuevos antibioticos de cefalosporina.

Country Status (17)

Country Link
EP (1) EP0138552A3 (es)
JP (1) JPS60105685A (es)
KR (1) KR850002992A (es)
AU (1) AU574107B2 (es)
CA (1) CA1225390A (es)
DK (1) DK489184A (es)
ES (1) ES536728A0 (es)
FI (1) FI844000L (es)
GB (2) GB2148289B (es)
GR (1) GR80670B (es)
HU (1) HU195512B (es)
IL (1) IL73230A0 (es)
NZ (1) NZ209833A (es)
PH (1) PH21040A (es)
PT (1) PT79357B (es)
SU (1) SU1360587A3 (es)
ZA (1) ZA847926B (es)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH22107A (en) * 1984-06-07 1988-06-01 Takeda Chemical Industries Ltd 3-pyrazolo(1,5-a)pyrdinium cephem compounds
US4734408A (en) * 1986-12-17 1988-03-29 Eli Lilly And Company Crystalline cephalosporin antibiotic salts and solvates
EP0304858A3 (en) * 1987-08-25 1989-12-20 Takeda Chemical Industries, Ltd. Cephem compounds, their production and use
TW526202B (en) * 1998-11-27 2003-04-01 Shionogi & Amp Co Broad spectrum cephem having benzo[4,5-b]pyridium methyl group of antibiotic activity
AT412214B (de) * 1999-05-05 2004-11-25 Sandoz Ag Verfahren zur herstellung des dinatrium-hemiheptahydratsalzes von ceftriaxon
GB0215293D0 (en) 2002-07-03 2002-08-14 Rega Foundation Viral inhibitors
US20050222198A1 (en) 2003-12-22 2005-10-06 K.U. Leuven Research & Development, Gerhard Puerstinger And Gilead Sciences, Inc. Imidazo[4,5-c]pyridine compounds and methods of antiviral treatment
AU2005319167B2 (en) 2004-12-21 2011-09-29 Gilead Sciences, Inc. Imidazo[4,5-C]pyridine compound and method of antiviral treatment
EA019452B1 (ru) 2006-07-07 2014-03-31 Джилид Сайэнс, Инк. 5-({6-[2,4-БИС-(ТРИФТОРМЕТИЛ)ФЕНИЛ]ПИРИДАЗИН-3-ИЛ}МЕТИЛ)-2-(2-ФТОРФЕНИЛ)-5Н-ИМИДАЗО[4,5-c]ПИРИДИН, СПОСОБ ЕГО ПОЛУЧЕНИЯ, СПОСОБ ЛЕЧЕНИЯ ИЛИ ПРОФИЛАКТИКИ ИНФЕКЦИОННОГО ВИРУСНОГО ГЕПАТИТА С С ЕГО ПОМОЩЬЮ, КОМПОЗИЦИЯ И ЛЕКАРСТВЕННОЕ СРЕДСТВО НА ЕГО ОСНОВЕ
UA99466C2 (en) 2007-07-06 2012-08-27 Гилиад Сайенсиз, Инк. Crystalline pyridazine compound
US9872906B2 (en) 2013-03-15 2018-01-23 Merck Sharp & Dohme Corp. Ceftolozane antibiotic compositions
US20140275000A1 (en) 2013-03-15 2014-09-18 Cubist Pharmaceuticals, Inc. Ceftolozane pharmaceutical compositions
WO2014144295A1 (en) 2013-03-15 2014-09-18 Cubist Pharmaceuticals, Inc. Ceftolozane antibiotic compositions
WO2015035376A2 (en) 2013-09-09 2015-03-12 Calixa Therapeutics, Inc. Treating infections with ceftolozane/tazobactam in subjects having impaired renal function
US8906898B1 (en) 2013-09-27 2014-12-09 Calixa Therapeutics, Inc. Solid forms of ceftolozane

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3118732A1 (de) * 1981-05-12 1982-12-02 Hoechst Ag, 6000 Frankfurt Cephalosporinderivate und verfahren zu ihrer herstellung
IL66726A0 (en) * 1981-09-08 1982-12-31 Lilly Co Eli Improvements in or relating to thieno and furopyridinium-substituted cephalosporin derivatives
DE3207840A1 (de) * 1982-03-04 1983-09-15 Hoechst Ag, 6230 Frankfurt "cephalosporinderivate und verfahren zu ihrer herstellung"
US4500526A (en) * 1982-06-28 1985-02-19 Bristol-Myers Company Cephalosporin derivatives
ATE30724T1 (de) * 1982-06-28 1987-11-15 Bristol Myers Co Cephalosporinderivate, verfahren zu ihrer herstellung und pharmazeutische zusammensetzungen die sie enthalten.

Also Published As

Publication number Publication date
HUT35687A (en) 1985-07-29
GB2181136A (en) 1987-04-15
IL73230A0 (en) 1985-01-31
FI844000L (fi) 1985-04-18
PH21040A (en) 1987-07-03
AU574107B2 (en) 1988-06-30
SU1360587A3 (ru) 1987-12-15
JPS60105685A (ja) 1985-06-11
NZ209833A (en) 1988-04-29
FI844000A0 (fi) 1984-10-11
GB2148289B (en) 1987-09-23
DK489184A (da) 1985-04-18
GB8425453D0 (en) 1984-11-14
CA1225390A (en) 1987-08-11
ES8602816A1 (es) 1985-11-16
GB8627171D0 (en) 1986-12-10
EP0138552A2 (en) 1985-04-24
GB2148289A (en) 1985-05-30
ZA847926B (en) 1986-05-28
PT79357B (en) 1986-11-20
KR850002992A (ko) 1985-05-28
GB2181136B (en) 1988-05-25
PT79357A (en) 1984-11-01
AU3418984A (en) 1985-04-26
GR80670B (en) 1985-02-18
EP0138552A3 (en) 1986-03-19
HU195512B (en) 1988-05-30
DK489184D0 (da) 1984-10-12

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