ES469952A1 - Un procedimiento para la preparacion de aminoalquiltiofenos - Google Patents
Un procedimiento para la preparacion de aminoalquiltiofenosInfo
- Publication number
- ES469952A1 ES469952A1 ES469952A ES469952A ES469952A1 ES 469952 A1 ES469952 A1 ES 469952A1 ES 469952 A ES469952 A ES 469952A ES 469952 A ES469952 A ES 469952A ES 469952 A1 ES469952 A1 ES 469952A1
- Authority
- ES
- Spain
- Prior art keywords
- image
- lower alkyl
- hydrogen
- compounds
- arylsulphonyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 150000001875 compounds Chemical class 0.000 title abstract 4
- 125000000217 alkyl group Chemical group 0.000 abstract 5
- 239000001257 hydrogen Substances 0.000 abstract 4
- 229910052739 hydrogen Inorganic materials 0.000 abstract 4
- 125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 4
- 125000003342 alkenyl group Chemical group 0.000 abstract 2
- 125000004390 alkyl sulfonyl group Chemical group 0.000 abstract 2
- 125000004391 aryl sulfonyl group Chemical group 0.000 abstract 2
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 2
- 101100244083 Arabidopsis thaliana PKL gene Proteins 0.000 abstract 1
- 125000004183 alkoxy alkyl group Chemical group 0.000 abstract 1
- 125000002947 alkylene group Chemical group 0.000 abstract 1
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 125000005842 heteroatom Chemical group 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 150000004677 hydrates Chemical class 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 125000004430 oxygen atom Chemical group O* 0.000 abstract 1
- 150000003141 primary amines Chemical class 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
- C07D333/20—Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB20659/77A GB1601459A (en) | 1977-05-17 | 1977-05-17 | Aminoalkyl thiophene derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES469952A1 true ES469952A1 (es) | 1979-09-16 |
Family
ID=10149541
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES469952A Expired ES469952A1 (es) | 1977-05-17 | 1978-05-17 | Un procedimiento para la preparacion de aminoalquiltiofenos |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US4239769A (OSRAM) |
| JP (2) | JPS53144568A (OSRAM) |
| AU (1) | AU519277B2 (OSRAM) |
| BE (1) | BE867105A (OSRAM) |
| DE (1) | DE2821409A1 (OSRAM) |
| DK (1) | DK214778A (OSRAM) |
| ES (1) | ES469952A1 (OSRAM) |
| FI (1) | FI781386A7 (OSRAM) |
| FR (1) | FR2391209A1 (OSRAM) |
| GB (1) | GB1601459A (OSRAM) |
| IE (1) | IE46811B1 (OSRAM) |
| NL (1) | NL7805278A (OSRAM) |
| NZ (1) | NZ187145A (OSRAM) |
| SE (1) | SE7805590L (OSRAM) |
| ZA (1) | ZA782478B (OSRAM) |
Families Citing this family (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4233302A (en) | 1977-12-23 | 1980-11-11 | Glaxo Group Limited | Amine derivatives and pharmaceutical compositions containing them |
| US4539207A (en) * | 1978-02-13 | 1985-09-03 | Smith Kline & French Laboratories Limited | Pyrimidine compounds |
| IN151188B (OSRAM) | 1978-02-13 | 1983-03-05 | Smith Kline French Lab | |
| AR228941A1 (es) * | 1978-04-26 | 1983-05-13 | Glaxo Group Ltd | Procedimiento para preparar nuevos derivados de 3,5-diamino-1,2,4-triazol que son activos contra receptores histaminicos |
| NZ193009A (en) * | 1979-03-02 | 1983-07-15 | Glaxo Group Ltd | 3-n-(( -aminoalkyl)(furyl thiophenyl or phenyl)(alkyl))-amino-1h-1,2,4-triazoles |
| JPS55120571A (en) * | 1979-03-02 | 1980-09-17 | Glaxo Group Ltd | Heterocyclic derivative |
| PH18379A (en) * | 1979-03-02 | 1985-06-19 | Glaxo Group Ltd | Triazole acylamines and pharmaceutical compositions thereof |
| JPS568352A (en) * | 1979-07-03 | 1981-01-28 | Shionogi & Co Ltd | Aminoalkylvenzene derivative |
| AU539189B2 (en) * | 1979-10-22 | 1984-09-13 | Glaxo Group Limited | 1h-1,2,4-triazole derivatives |
| DE3067019D1 (en) * | 1979-10-23 | 1984-04-19 | Glaxo Group Ltd | Thiophene derivatives, processes for the production thereof and pharmaceutical compositions containing them |
| US4382929A (en) * | 1979-10-23 | 1983-05-10 | Glaxo Group Limited | Thiophene derivatives and their pharmaceutical compositions and method of use |
| JPS5681578A (en) * | 1979-12-07 | 1981-07-03 | Shionogi & Co Ltd | Novel thioalkyl amide derivative |
| US4431802A (en) * | 1979-12-10 | 1984-02-14 | G. D. Searle & Co. | N-Heterocyclyl-N-cyano-N-(heterocyclythioalkyl)-guanidines |
| US4491586A (en) * | 1980-06-05 | 1985-01-01 | Glaxo Group Limited | Amine derivatives |
| EP0057981A3 (en) * | 1981-02-09 | 1982-08-25 | Beecham Group Plc | Aromatic compounds, processes for their preparation and their use |
| DE3108753A1 (de) * | 1981-03-07 | 1982-09-16 | Degussa Ag, 6000 Frankfurt | Neue substituierte alkyl-phenylsulfonylguanidine miteinem heterocyclischen rest |
| US4390701A (en) * | 1981-05-18 | 1983-06-28 | Bristol-Myers Company | 1-Amino-2-[3-(3-piperidinomethylphenoxy)propylamino]cyclobutene-3,4-dione |
| US4788184A (en) * | 1981-05-18 | 1988-11-29 | Bristol-Myers Company | Substituted 3-cyclobutene-1,2-diones as anti-ulcer agents |
| WO1983002113A1 (fr) * | 1981-12-17 | 1983-06-23 | Yuki, Hiroshi | Derives de propenylamine et medicaments les contenant |
| DE3238867A1 (de) * | 1982-10-20 | 1984-04-26 | Ludwig Heumann & Co GmbH, 8500 Nürnberg | Heterocyclische verbindungen, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
| JPS5988458A (ja) * | 1982-11-12 | 1984-05-22 | Toyama Chem Co Ltd | アミン誘導体およびその塩 |
| NL8303965A (nl) * | 1982-12-08 | 1984-07-02 | Degussa | Nieuwe etheendiamine- en guanidine-derivaten; werkwijze voor het bereiden daarvan; geneesmiddelen die ze bevatten; werkwijze voor het bereiden van dergelijke geneesmiddelen; toepassing van de verbindingen voor het bereiden van geneesmiddelen en in de geneeskunde. |
| DE3343884A1 (de) * | 1982-12-08 | 1984-06-14 | Degussa Ag, 6000 Frankfurt | Neue ethendiamin- und guanidin-derivate |
| DE3404786A1 (de) * | 1984-02-10 | 1985-08-14 | Ludwig Heumann & Co GmbH, 8500 Nürnberg | Neue alkanolderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltendes arzneimittel |
| FR2571723B1 (fr) * | 1984-10-12 | 1988-08-26 | Lipha | Derives de thieno et furo-(2,3-c) pyrroles, procedes de preparation et medicaments les contenant |
| DE3568374D1 (en) * | 1985-12-20 | 1989-03-30 | Litef Gmbh | Method to determine heading by using and automatically calibrating a 3-axis magnetometer rigidly fitted in an aircraft |
| JPS6370615U (OSRAM) * | 1986-10-28 | 1988-05-12 | ||
| JPH05236847A (ja) * | 1992-02-28 | 1993-09-17 | Reishii:Kk | 熱交換装置 |
| US6291514B1 (en) * | 1998-02-09 | 2001-09-18 | 3-Dimensional Pharmaceuticals, Inc. | Heteroaryl amidines, methylamidines and guanidines, preparation thereof, and use thereof as protease inhibitors |
| WO2022034121A1 (en) | 2020-08-11 | 2022-02-17 | Université De Strasbourg | H2 blockers targeting liver macrophages for the prevention and treatment of liver disease and cancer |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2519325A (en) * | 1947-01-04 | 1950-08-15 | White Lab Inc | Antihistamine compounds |
| US2556636A (en) * | 1948-06-23 | 1951-06-12 | Schering Corp | gamma-substituted propylamine type antihistamines |
| US2604473A (en) * | 1950-07-17 | 1952-07-22 | Schering Corp | Propylamine type antihistamines |
| GB1307539A (en) | 1970-06-25 | 1973-02-21 | Smith Kline French Lab | Thiourea derivatives |
| GB1338169A (en) | 1971-03-09 | 1973-11-21 | Smith Kline French Lab | Ureas thioureas and guanidines |
| GB1397436A (en) | 1972-09-05 | 1975-06-11 | Smith Kline French Lab | Heterocyclic n-cyanoguinidines |
| GB1421792A (en) | 1973-05-17 | 1976-01-21 | Smith Kline French Lab | Heterocyclic substituted-1, 1-diamino-ethylene derivatives methods for their preparation and compositions containing them |
| GB1565966A (en) * | 1976-08-04 | 1980-04-23 | Allen & Hanburys Ltd | Aminoalkyl furan derivatives |
-
1977
- 1977-05-17 GB GB20659/77A patent/GB1601459A/en not_active Expired
-
1978
- 1978-04-28 IE IE853/78A patent/IE46811B1/en unknown
- 1978-05-01 ZA ZA00782478A patent/ZA782478B/xx unknown
- 1978-05-02 AU AU35673/78A patent/AU519277B2/en not_active Expired
- 1978-05-02 NZ NZ187145A patent/NZ187145A/xx unknown
- 1978-05-04 FI FI781386A patent/FI781386A7/fi not_active Application Discontinuation
- 1978-05-05 US US05/903,116 patent/US4239769A/en not_active Expired - Lifetime
- 1978-05-16 BE BE187721A patent/BE867105A/xx not_active IP Right Cessation
- 1978-05-16 DE DE19782821409 patent/DE2821409A1/de not_active Withdrawn
- 1978-05-16 DK DK214778A patent/DK214778A/da unknown
- 1978-05-16 SE SE7805590A patent/SE7805590L/xx unknown
- 1978-05-16 NL NL7805278A patent/NL7805278A/xx not_active Application Discontinuation
- 1978-05-17 FR FR7814593A patent/FR2391209A1/fr active Granted
- 1978-05-17 ES ES469952A patent/ES469952A1/es not_active Expired
- 1978-05-17 JP JP5870578A patent/JPS53144568A/ja active Granted
-
1979
- 1979-10-26 JP JP13860479A patent/JPS55113776A/ja active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| US4239769A (en) | 1980-12-16 |
| BE867105A (fr) | 1978-11-16 |
| FR2391209A1 (fr) | 1978-12-15 |
| GB1601459A (en) | 1981-10-28 |
| DK214778A (da) | 1978-11-18 |
| DE2821409A1 (de) | 1978-11-30 |
| AU3567378A (en) | 1979-11-08 |
| IE46811B1 (en) | 1983-10-05 |
| NZ187145A (en) | 1980-10-24 |
| JPS53144568A (en) | 1978-12-15 |
| IE780853L (en) | 1978-11-17 |
| NL7805278A (nl) | 1978-11-21 |
| JPS6312069B2 (OSRAM) | 1988-03-17 |
| JPS5510591B2 (OSRAM) | 1980-03-17 |
| ZA782478B (en) | 1979-04-25 |
| FR2391209B1 (OSRAM) | 1982-05-14 |
| JPS55113776A (en) | 1980-09-02 |
| FI781386A7 (fi) | 1978-11-18 |
| AU519277B2 (en) | 1981-11-19 |
| SE7805590L (sv) | 1978-11-18 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 19980202 |