BE867105A - Aminoalkyl thiophenes, leur preparation et compositions en contenant - Google Patents

Aminoalkyl thiophenes, leur preparation et compositions en contenant

Info

Publication number
BE867105A
BE867105A BE187721A BE187721A BE867105A BE 867105 A BE867105 A BE 867105A BE 187721 A BE187721 A BE 187721A BE 187721 A BE187721 A BE 187721A BE 867105 A BE867105 A BE 867105A
Authority
BE
Belgium
Prior art keywords
thiophens
aminoalkyl
preparation
compositions containing
compositions
Prior art date
Application number
BE187721A
Other languages
English (en)
Original Assignee
Allen & Hanburys Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Allen & Hanburys Ltd filed Critical Allen & Hanburys Ltd
Publication of BE867105A publication Critical patent/BE867105A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
    • C07D333/20—Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
BE187721A 1977-05-17 1978-05-16 Aminoalkyl thiophenes, leur preparation et compositions en contenant BE867105A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB20659/77A GB1601459A (en) 1977-05-17 1977-05-17 Aminoalkyl thiophene derivatives

Publications (1)

Publication Number Publication Date
BE867105A true BE867105A (fr) 1978-11-16

Family

ID=10149541

Family Applications (1)

Application Number Title Priority Date Filing Date
BE187721A BE867105A (fr) 1977-05-17 1978-05-16 Aminoalkyl thiophenes, leur preparation et compositions en contenant

Country Status (15)

Country Link
US (1) US4239769A (fr)
JP (2) JPS53144568A (fr)
AU (1) AU519277B2 (fr)
BE (1) BE867105A (fr)
DE (1) DE2821409A1 (fr)
DK (1) DK214778A (fr)
ES (1) ES469952A1 (fr)
FI (1) FI781386A (fr)
FR (1) FR2391209A1 (fr)
GB (1) GB1601459A (fr)
IE (1) IE46811B1 (fr)
NL (1) NL7805278A (fr)
NZ (1) NZ187145A (fr)
SE (1) SE7805590L (fr)
ZA (1) ZA782478B (fr)

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4304780A (en) 1977-12-23 1981-12-08 Glaxo Group Limited Aminoalkylthiophene derivatives as histamine H2 -antagonists
US4323566A (en) * 1979-03-02 1982-04-06 Glaxo Group Limited Triazole acylamines, pharmaceutical compositions thereof and method of use thereof
US4382929A (en) * 1979-10-23 1983-05-10 Glaxo Group Limited Thiophene derivatives and their pharmaceutical compositions and method of use
DE3343884A1 (de) * 1982-12-08 1984-06-14 Degussa Ag, 6000 Frankfurt Neue ethendiamin- und guanidin-derivate
US4491586A (en) * 1980-06-05 1985-01-01 Glaxo Group Limited Amine derivatives
US4536508A (en) * 1979-03-02 1985-08-20 Glaxo Group Limited Triazoleamine derivatives having histamine H2 -antagonist properties
US4539207A (en) * 1978-02-13 1985-09-03 Smith Kline & French Laboratories Limited Pyrimidine compounds
US4649141A (en) * 1978-02-13 1987-03-10 Smith Kline & French Laboratories Limited Pyrimidine compounds

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR228941A1 (es) * 1978-04-26 1983-05-13 Glaxo Group Ltd Procedimiento para preparar nuevos derivados de 3,5-diamino-1,2,4-triazol que son activos contra receptores histaminicos
IE49528B1 (en) * 1979-03-02 1985-10-16 Glaxo Group Ltd Substituted aminotriazoles
JPS568352A (en) * 1979-07-03 1981-01-28 Shionogi & Co Ltd Aminoalkylvenzene derivative
AU539189B2 (en) * 1979-10-22 1984-09-13 Glaxo Group Limited 1h-1,2,4-triazole derivatives
AU539733B2 (en) * 1979-10-23 1984-10-11 Glaxo Group Limited Thiophen derivatives
JPS5681578A (en) * 1979-12-07 1981-07-03 Shionogi & Co Ltd Novel thioalkyl amide derivative
US4431802A (en) * 1979-12-10 1984-02-14 G. D. Searle & Co. N-Heterocyclyl-N-cyano-N-(heterocyclythioalkyl)-guanidines
EP0057981A3 (fr) * 1981-02-09 1982-08-25 Beecham Group Plc Composés aromatiques, procédés pour leur préparation et leur application
DE3108753A1 (de) * 1981-03-07 1982-09-16 Degussa Ag, 6000 Frankfurt Neue substituierte alkyl-phenylsulfonylguanidine miteinem heterocyclischen rest
US4390701A (en) * 1981-05-18 1983-06-28 Bristol-Myers Company 1-Amino-2-[3-(3-piperidinomethylphenoxy)propylamino]cyclobutene-3,4-dione
US4788184A (en) * 1981-05-18 1988-11-29 Bristol-Myers Company Substituted 3-cyclobutene-1,2-diones as anti-ulcer agents
WO1983002113A1 (fr) * 1981-12-17 1983-06-23 Yuki, Hiroshi Derives de propenylamine et medicaments les contenant
DE3238867A1 (de) * 1982-10-20 1984-04-26 Ludwig Heumann & Co GmbH, 8500 Nürnberg Heterocyclische verbindungen, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
JPS5988458A (ja) * 1982-11-12 1984-05-22 Toyama Chem Co Ltd アミン誘導体およびその塩
NL8303965A (nl) * 1982-12-08 1984-07-02 Degussa Nieuwe etheendiamine- en guanidine-derivaten; werkwijze voor het bereiden daarvan; geneesmiddelen die ze bevatten; werkwijze voor het bereiden van dergelijke geneesmiddelen; toepassing van de verbindingen voor het bereiden van geneesmiddelen en in de geneeskunde.
DE3404786A1 (de) * 1984-02-10 1985-08-14 Ludwig Heumann & Co GmbH, 8500 Nürnberg Neue alkanolderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltendes arzneimittel
FR2571723B1 (fr) * 1984-10-12 1988-08-26 Lipha Derives de thieno et furo-(2,3-c) pyrroles, procedes de preparation et medicaments les contenant
EP0226653B1 (fr) * 1985-12-20 1989-02-22 LITEF GmbH Procédé pour la détermination du cap magnétique par l'utilisation et le calibrage automatique d'un magnétomètre à trois axes installé dans un avion
JPS6370615U (fr) * 1986-10-28 1988-05-12
JPH05236847A (ja) * 1992-02-28 1993-09-17 Reishii:Kk 熱交換装置
US6291514B1 (en) 1998-02-09 2001-09-18 3-Dimensional Pharmaceuticals, Inc. Heteroaryl amidines, methylamidines and guanidines, preparation thereof, and use thereof as protease inhibitors
WO2022034121A1 (fr) 2020-08-11 2022-02-17 Université De Strasbourg Bloqueurs de h2 ciblant des macrophages du foie pour la prévention et le traitement d'une maladie du foie et du cancer

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2519325A (en) * 1947-01-04 1950-08-15 White Lab Inc Antihistamine compounds
US2556636A (en) * 1948-06-23 1951-06-12 Schering Corp gamma-substituted propylamine type antihistamines
US2604473A (en) * 1950-07-17 1952-07-22 Schering Corp Propylamine type antihistamines
GB1307539A (en) 1970-06-25 1973-02-21 Smith Kline French Lab Thiourea derivatives
GB1338169A (en) 1971-03-09 1973-11-21 Smith Kline French Lab Ureas thioureas and guanidines
GB1397436A (en) 1972-09-05 1975-06-11 Smith Kline French Lab Heterocyclic n-cyanoguinidines
GB1421792A (en) 1973-05-17 1976-01-21 Smith Kline French Lab Heterocyclic substituted-1, 1-diamino-ethylene derivatives methods for their preparation and compositions containing them
GB1565966A (en) * 1976-08-04 1980-04-23 Allen & Hanburys Ltd Aminoalkyl furan derivatives

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4304780A (en) 1977-12-23 1981-12-08 Glaxo Group Limited Aminoalkylthiophene derivatives as histamine H2 -antagonists
US4539207A (en) * 1978-02-13 1985-09-03 Smith Kline & French Laboratories Limited Pyrimidine compounds
US4649141A (en) * 1978-02-13 1987-03-10 Smith Kline & French Laboratories Limited Pyrimidine compounds
US4323566A (en) * 1979-03-02 1982-04-06 Glaxo Group Limited Triazole acylamines, pharmaceutical compositions thereof and method of use thereof
US4536508A (en) * 1979-03-02 1985-08-20 Glaxo Group Limited Triazoleamine derivatives having histamine H2 -antagonist properties
US4382929A (en) * 1979-10-23 1983-05-10 Glaxo Group Limited Thiophene derivatives and their pharmaceutical compositions and method of use
US4491586A (en) * 1980-06-05 1985-01-01 Glaxo Group Limited Amine derivatives
DE3343884A1 (de) * 1982-12-08 1984-06-14 Degussa Ag, 6000 Frankfurt Neue ethendiamin- und guanidin-derivate

Also Published As

Publication number Publication date
DK214778A (da) 1978-11-18
GB1601459A (en) 1981-10-28
SE7805590L (sv) 1978-11-18
FI781386A (fi) 1978-11-18
IE780853L (en) 1978-11-17
ZA782478B (en) 1979-04-25
ES469952A1 (es) 1979-09-16
FR2391209A1 (fr) 1978-12-15
IE46811B1 (en) 1983-10-05
JPS6312069B2 (fr) 1988-03-17
AU519277B2 (en) 1981-11-19
NL7805278A (nl) 1978-11-21
NZ187145A (en) 1980-10-24
JPS53144568A (en) 1978-12-15
US4239769A (en) 1980-12-16
FR2391209B1 (fr) 1982-05-14
DE2821409A1 (de) 1978-11-30
JPS55113776A (en) 1980-09-02
AU3567378A (en) 1979-11-08
JPS5510591B2 (fr) 1980-03-17

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: ALLEN & HANBURYS LTD

Effective date: 19860531