ES458740A1 - Procedimiento para la preparacion de bencenosulfonilureas. - Google Patents
Procedimiento para la preparacion de bencenosulfonilureas.Info
- Publication number
- ES458740A1 ES458740A1 ES458740A ES458740A ES458740A1 ES 458740 A1 ES458740 A1 ES 458740A1 ES 458740 A ES458740 A ES 458740A ES 458740 A ES458740 A ES 458740A ES 458740 A1 ES458740 A1 ES 458740A1
- Authority
- ES
- Spain
- Prior art keywords
- treatment
- diabetes mellitus
- benzenesulfonyl ureas
- benzenesulfonyl
- ureas
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
- C07D213/82—Amides; Imides in position 3
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pain & Pain Management (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Quinoline Compounds (AREA)
Abstract
Procedimiento para la preparación de bencenosulfonilurea de la fórmula *** ver imagen 01 en la cual R significa alcohilo, alcoxialcohilo, alquenilo con hasta 6 átomos en cada caso, cicloalcohilo, cicloalquenilo, alcohilcicloalcohilo, alcohilcicloalquenilo, cicloalcohilalquenilo, cicloalquenilalcohilo, alcohilcicloalcohilalcohilo, alcohilcicloalquenilalcohilo, con 5 a 9 átomos de carbono en cada caso, fenilo el cual está eventualmente mono- o disustituido con alcohilo o alcoxi, con hasta 4 átomos de carbono, en cada caso o con halógeno; R1, R2, R3 significan hidrógeno, alcohilo, alcoxi con hasta 2 átomos de carbono en cada caso, halógeno, R1 y R2 significan conjuntamente también *** ver imagen 02 5, 6, eventualmente sustituidos con halógeno o metilo, e Y significa alcohileno de 2 a 3 átomos de carbono preferentemente ¿CH2-CH2-;
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19762621958 DE2621958A1 (de) | 1976-05-18 | 1976-05-18 | Benzolsulfonylharnstoffe und verfahren zu ihrer herstellung |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES458740A1 true ES458740A1 (es) | 1978-03-01 |
Family
ID=5978221
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES458740A Expired ES458740A1 (es) | 1976-05-18 | 1977-05-12 | Procedimiento para la preparacion de bencenosulfonilureas. |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US4132795A (es) |
| JP (1) | JPS52142075A (es) |
| AT (1) | AT357558B (es) |
| AU (1) | AU509768B2 (es) |
| BE (1) | BE854812A (es) |
| CH (4) | CH628887A5 (es) |
| DE (1) | DE2621958A1 (es) |
| DK (1) | DK214577A (es) |
| EG (1) | EG12586A (es) |
| ES (1) | ES458740A1 (es) |
| FI (1) | FI771548A (es) |
| FR (1) | FR2351965A1 (es) |
| GB (1) | GB1581593A (es) |
| HU (1) | HU173606B (es) |
| IL (1) | IL52100A0 (es) |
| IT (1) | IT1085546B (es) |
| NL (1) | NL7705323A (es) |
| NO (1) | NO771728L (es) |
| NZ (1) | NZ184102A (es) |
| PT (1) | PT66561B (es) |
| SE (1) | SE7705873L (es) |
| ZA (1) | ZA772950B (es) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2948472A1 (de) * | 1979-12-01 | 1981-06-11 | Hoechst Ag, 6000 Frankfurt | Benzolsulfonylharnstoffe und verfahren zu ihrer herstellung |
| DE2948522A1 (de) * | 1979-12-01 | 1981-06-11 | Hoechst Ag, 6000 Frankfurt | Benzolsulfonylharnstoffe und verfahren zu ihrer herstellung |
| DE2948434A1 (de) * | 1979-12-01 | 1981-06-11 | Hoechst Ag, 6000 Frankfurt | 1-piperidinsulfonylharnstoffe und verfahren zu ihrer herstellung |
| EP0031088A1 (de) * | 1979-12-19 | 1981-07-01 | Hoechst Aktiengesellschaft | Benzolsulfonylharnstoffe, Verfahren zu ihrer Herstellung, pharmazeutische Präparate auf Basis dieser Verbindungen sowie ihre Verwendung |
| DE2951135A1 (de) * | 1979-12-19 | 1981-06-25 | Hoechst Ag, 6230 Frankfurt | Sulfonylharnstoffe, verfahren zu ihrer herstellung, pharmazeutische praeparate auf basis dieser verbindungen und ihre verwendung |
| DE3134780A1 (de) * | 1981-09-02 | 1983-03-10 | Hoechst Ag, 6000 Frankfurt | "sulfonylharnstoffe, verfahren zu ihrer herstellung, pharmazeutische praeparate auf basis dieser verbindungen und ihre verwendung" |
| DE3210063A1 (de) * | 1982-03-19 | 1983-09-22 | Hoechst Ag, 6230 Frankfurt | Sulfonylharnstoffe, verfahren zu ihrer herstellung, pharmazeutische praeparate auf basis dieser verbindungen und ihre verwendung |
| ES2333214T3 (es) * | 2002-02-19 | 2010-02-18 | SHIONOGI & CO., LTD. | Antipruriticos. |
| WO2008005457A2 (en) | 2006-06-30 | 2008-01-10 | Sunesis Pharmaceuticals | Pyridinonyl pdk1 inhibitors |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4066639A (en) * | 1965-05-06 | 1978-01-03 | Hoechst Aktiengesellschaft | Benzene-sulfonyl semicarbazides and process for preparing them |
| DE2238870C3 (de) * | 1972-08-07 | 1978-09-28 | Hoechst Ag, 6000 Frankfurt | Benzolsulfonylharnstoffe |
-
1976
- 1976-05-18 DE DE19762621958 patent/DE2621958A1/de not_active Withdrawn
-
1977
- 1977-05-12 ES ES458740A patent/ES458740A1/es not_active Expired
- 1977-05-13 NL NL7705323A patent/NL7705323A/xx not_active Application Discontinuation
- 1977-05-14 EG EG290/77A patent/EG12586A/xx active
- 1977-05-16 IL IL52100A patent/IL52100A0/xx unknown
- 1977-05-16 CH CH607777A patent/CH628887A5/de not_active IP Right Cessation
- 1977-05-16 NZ NZ184102A patent/NZ184102A/xx unknown
- 1977-05-16 FI FI771548A patent/FI771548A/fi not_active Application Discontinuation
- 1977-05-16 US US05/797,132 patent/US4132795A/en not_active Expired - Lifetime
- 1977-05-16 NO NO771728A patent/NO771728L/no unknown
- 1977-05-16 IT IT23615/77A patent/IT1085546B/it active
- 1977-05-17 HU HU77HO1985A patent/HU173606B/hu unknown
- 1977-05-17 ZA ZA00772950A patent/ZA772950B/xx unknown
- 1977-05-17 SE SE7705873A patent/SE7705873L/xx unknown
- 1977-05-17 PT PT66561A patent/PT66561B/pt unknown
- 1977-05-17 AT AT353377A patent/AT357558B/de not_active IP Right Cessation
- 1977-05-17 AU AU25191/77A patent/AU509768B2/en not_active Expired
- 1977-05-17 GB GB20668/77A patent/GB1581593A/en not_active Expired
- 1977-05-17 DK DK214577A patent/DK214577A/da not_active Application Discontinuation
- 1977-05-18 FR FR7715360A patent/FR2351965A1/fr active Granted
- 1977-05-18 JP JP5650477A patent/JPS52142075A/ja active Pending
- 1977-05-18 BE BE177721A patent/BE854812A/xx unknown
-
1981
- 1981-06-15 CH CH393781A patent/CH629781A5/de not_active IP Right Cessation
- 1981-06-15 CH CH393581A patent/CH629780A5/de not_active IP Right Cessation
- 1981-06-15 CH CH393381A patent/CH629779A5/de not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| AU2519177A (en) | 1978-11-23 |
| CH629781A5 (de) | 1982-05-14 |
| PT66561B (de) | 1979-01-22 |
| CH629779A5 (de) | 1982-05-14 |
| DK214577A (da) | 1977-11-19 |
| IT1085546B (it) | 1985-05-28 |
| US4132795A (en) | 1979-01-02 |
| HU173606B (hu) | 1979-06-28 |
| BE854812A (fr) | 1977-11-18 |
| FI771548A (es) | 1977-11-19 |
| NL7705323A (nl) | 1977-11-22 |
| CH628887A5 (de) | 1982-03-31 |
| GB1581593A (en) | 1980-12-17 |
| DE2621958A1 (de) | 1977-12-08 |
| FR2351965B1 (es) | 1980-02-08 |
| ZA772950B (en) | 1978-04-26 |
| AU509768B2 (en) | 1980-05-22 |
| CH629780A5 (de) | 1982-05-14 |
| AT357558B (de) | 1980-07-25 |
| ATA353377A (de) | 1979-12-15 |
| FR2351965A1 (fr) | 1977-12-16 |
| NZ184102A (en) | 1979-03-28 |
| JPS52142075A (en) | 1977-11-26 |
| IL52100A0 (en) | 1977-07-31 |
| SE7705873L (sv) | 1977-11-19 |
| PT66561A (de) | 1977-06-01 |
| EG12586A (en) | 1981-06-30 |
| NO771728L (no) | 1977-11-21 |
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