ES440901A1 - 6-isocyanato-2,2-dimethyl-3-(5-tetrazolyl)penams - Google Patents

6-isocyanato-2,2-dimethyl-3-(5-tetrazolyl)penams

Info

Publication number
ES440901A1
ES440901A1 ES440901A ES440901A ES440901A1 ES 440901 A1 ES440901 A1 ES 440901A1 ES 440901 A ES440901 A ES 440901A ES 440901 A ES440901 A ES 440901A ES 440901 A1 ES440901 A1 ES 440901A1
Authority
ES
Spain
Prior art keywords
carbon atoms
formula
phenyl
alkyl
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES440901A
Other languages
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of ES440901A1 publication Critical patent/ES440901A1/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

A method of producing new, substituted amino-3-tetrazolylpenams of the formula **(See formula)** where Y3 is the acyl radical of an organic, carbamyl or substituted carbamyl acid acylating agent, Y1 is **(See formula)** wherein R1 is R2 or a nitrogen protecting group from tetrazozolylpenam; R2 is hydrogen, trialkylsilyl having 1 to 4 carbon atoms per alkyl group, alkanoyloxymethyl having three to eight carbon atoms, 1-alkanoyloxyethyl having four to nine carbon atoms, phthalidyl or **(See formula)** wherein each of R3, R4, and R5 is hydrogen, chlorine, bromine, fluorine, alkyl having one to four carbon atoms, alkoxy having one to four carbon atoms, or phenyl, characterized by reacting in a solvent inert organic, a compound of the formula **(See formula)** with an isocyanate conversion reagent which is (a) an organic acid acylating agent, (b) ammonia or (c) an amine of the formula X3'NH2, where Y3'is alkyl of 1 to 6 carbon atoms, phenyl, substituted phenyl, naphthyl, or substituted naphthyl, wherein the phenyl or naphthyl substituent is hydroxy, C 1 -C 4 -alkoxy, C 1 -C 4 -alkyl, chlorine, bromine, fluorine, trifluoromethyl, carboxy or carboalkoxy of 2 to 5 carbon atoms. (Machine-translation by Google Translate, not legally binding)
ES440901A 1974-10-07 1975-09-12 6-isocyanato-2,2-dimethyl-3-(5-tetrazolyl)penams Expired ES440901A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US51242674A 1974-10-07 1974-10-07

Publications (1)

Publication Number Publication Date
ES440901A1 true ES440901A1 (en) 1977-06-16

Family

ID=24039029

Family Applications (2)

Application Number Title Priority Date Filing Date
ES440901A Expired ES440901A1 (en) 1974-10-07 1975-09-12 6-isocyanato-2,2-dimethyl-3-(5-tetrazolyl)penams
ES451529A Expired ES451529A1 (en) 1974-10-07 1976-09-15 6-isocyanato-2,2-dimethyl-3-(5-tetrazolyl)penams

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES451529A Expired ES451529A1 (en) 1974-10-07 1976-09-15 6-isocyanato-2,2-dimethyl-3-(5-tetrazolyl)penams

Country Status (15)

Country Link
JP (1) JPS5159894A (en)
AR (1) AR213165A1 (en)
BE (1) BE833781A (en)
DD (1) DD123470A5 (en)
DE (1) DE2543703A1 (en)
ES (2) ES440901A1 (en)
FI (1) FI752673A (en)
FR (2) FR2313388A1 (en)
GB (1) GB1479099A (en)
IE (1) IE41585B1 (en)
IL (1) IL47987A0 (en)
LU (1) LU73473A1 (en)
NL (1) NL7510696A (en)
RO (1) RO68718B (en)
SE (1) SE7509000L (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11251075B2 (en) * 2018-08-06 2022-02-15 Mattson Technology, Inc. Systems and methods for workpiece processing using neutral atom beams

Also Published As

Publication number Publication date
FI752673A (en) 1976-04-08
FR2327248B1 (en) 1979-04-20
FR2313388B1 (en) 1978-04-07
DE2543703A1 (en) 1976-04-08
GB1479099A (en) 1977-07-06
AR213165A1 (en) 1978-12-29
FR2327248A1 (en) 1977-05-06
ES451529A1 (en) 1977-12-01
LU73473A1 (en) 1976-08-19
NL7510696A (en) 1976-04-09
IL47987A0 (en) 1975-11-25
BE833781A (en) 1976-03-25
JPS5159894A (en) 1976-05-25
RO68718A (en) 1983-04-29
IE41585B1 (en) 1980-02-13
AU8479875A (en) 1976-10-28
FR2313388A1 (en) 1976-12-31
IE41585L (en) 1976-04-07
SE7509000L (en) 1976-04-08
DD123470A5 (en) 1976-12-20
RO68718B (en) 1983-04-30

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