ES423178A1 - Procedimiento para la preparacion de esteres acilamidometi-licos de penicilinas y cefalosporinas. - Google Patents
Procedimiento para la preparacion de esteres acilamidometi-licos de penicilinas y cefalosporinas.Info
- Publication number
- ES423178A1 ES423178A1 ES423178A ES423178A ES423178A1 ES 423178 A1 ES423178 A1 ES 423178A1 ES 423178 A ES423178 A ES 423178A ES 423178 A ES423178 A ES 423178A ES 423178 A1 ES423178 A1 ES 423178A1
- Authority
- ES
- Spain
- Prior art keywords
- see formula
- hydrogen
- formula
- chosen
- group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 229930186147 Cephalosporin Natural products 0.000 title abstract 2
- 229930182555 Penicillin Natural products 0.000 title abstract 2
- 229940124587 cephalosporin Drugs 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- 150000002960 penicillins Chemical class 0.000 title abstract 2
- HOKIDJSKDBPKTQ-GLXFQSAKSA-N cephalosporin C Chemical compound S1CC(COC(=O)C)=C(C(O)=O)N2C(=O)[C@@H](NC(=O)CCC[C@@H](N)C(O)=O)[C@@H]12 HOKIDJSKDBPKTQ-GLXFQSAKSA-N 0.000 title 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 6
- 239000001257 hydrogen Substances 0.000 abstract 6
- 239000002253 acid Substances 0.000 abstract 3
- 150000002148 esters Chemical class 0.000 abstract 3
- HSHGZXNAXBPPDL-HZGVNTEJSA-N 7beta-aminocephalosporanic acid Chemical compound S1CC(COC(=O)C)=C(C([O-])=O)N2C(=O)[C@@H]([NH3+])[C@@H]12 HSHGZXNAXBPPDL-HZGVNTEJSA-N 0.000 abstract 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
- 125000004432 carbon atom Chemical group C* 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 150000002431 hydrogen Chemical class 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
- 229910052740 iodine Inorganic materials 0.000 abstract 2
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical compound [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 abstract 1
- QDHHCQZDFGDHMP-UHFFFAOYSA-N Chloramine Chemical group ClN QDHHCQZDFGDHMP-UHFFFAOYSA-N 0.000 abstract 1
- ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 abstract 1
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical group FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 abstract 1
- 150000007513 acids Chemical class 0.000 abstract 1
- 229910052783 alkali metal Inorganic materials 0.000 abstract 1
- 150000001340 alkali metals Chemical class 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 150000001412 amines Chemical group 0.000 abstract 1
- GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Substances BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 abstract 1
- 229910052794 bromium Inorganic materials 0.000 abstract 1
- 150000001768 cations Chemical group 0.000 abstract 1
- 150000001780 cephalosporins Chemical class 0.000 abstract 1
- 229910052801 chlorine Inorganic materials 0.000 abstract 1
- 239000000460 chlorine Substances 0.000 abstract 1
- 229910052731 fluorine Chemical group 0.000 abstract 1
- 239000011737 fluorine Chemical group 0.000 abstract 1
- 125000002541 furyl group Chemical group 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 125000004076 pyridyl group Chemical group 0.000 abstract 1
- 125000000168 pyrrolyl group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 150000003512 tertiary amines Chemical class 0.000 abstract 1
- 125000001544 thienyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT2035873 | 1973-02-14 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES423178A1 true ES423178A1 (es) | 1976-05-01 |
Family
ID=11166010
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES423178A Expired ES423178A1 (es) | 1973-02-14 | 1974-02-13 | Procedimiento para la preparacion de esteres acilamidometi-licos de penicilinas y cefalosporinas. |
Country Status (9)
| Country | Link |
|---|---|
| JP (1) | JPS5418277B2 (enrdf_load_stackoverflow) |
| AT (1) | AT329179B (enrdf_load_stackoverflow) |
| BE (1) | BE810969A (enrdf_load_stackoverflow) |
| CH (1) | CH592670A5 (enrdf_load_stackoverflow) |
| DE (1) | DE2406817A1 (enrdf_load_stackoverflow) |
| ES (1) | ES423178A1 (enrdf_load_stackoverflow) |
| FR (1) | FR2216995B1 (enrdf_load_stackoverflow) |
| GB (1) | GB1421526A (enrdf_load_stackoverflow) |
| NL (1) | NL7401782A (enrdf_load_stackoverflow) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4428935A (en) * | 1982-05-24 | 1984-01-31 | Pfizer Inc. | Penicillanic acid dioxide prodrug |
| GB8300295D0 (en) * | 1983-01-06 | 1983-02-09 | Erba Farmitalia | Penem esters |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1491583A (fr) * | 1965-07-22 | 1967-08-11 | Bristol Myers Co | Production de nouveaux esters activés de l'acide 6-aminopénicillanique |
| US3873521A (en) * | 1970-09-17 | 1975-03-25 | Astra Laekemedel Ab | Esters of {60 -amino penicillins |
| GB1425933A (en) * | 1972-03-13 | 1976-02-25 | Astra Laekemedel Ab | Cephalosporins |
| GB1426869A (en) * | 1972-03-13 | 1976-03-03 | Astra Laekemedel Ab | Penicillins |
-
1974
- 1974-02-08 NL NL7401782A patent/NL7401782A/xx not_active Application Discontinuation
- 1974-02-11 GB GB611574A patent/GB1421526A/en not_active Expired
- 1974-02-11 AT AT105874A patent/AT329179B/de not_active IP Right Cessation
- 1974-02-12 JP JP1751374A patent/JPS5418277B2/ja not_active Expired
- 1974-02-12 FR FR7404609A patent/FR2216995B1/fr not_active Expired
- 1974-02-13 BE BE140855A patent/BE810969A/xx unknown
- 1974-02-13 ES ES423178A patent/ES423178A1/es not_active Expired
- 1974-02-13 CH CH196074A patent/CH592670A5/xx not_active IP Right Cessation
- 1974-02-13 DE DE19742406817 patent/DE2406817A1/de not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| FR2216995A1 (enrdf_load_stackoverflow) | 1974-09-06 |
| CH592670A5 (enrdf_load_stackoverflow) | 1977-10-31 |
| DE2406817A1 (de) | 1974-08-22 |
| NL7401782A (enrdf_load_stackoverflow) | 1974-08-16 |
| GB1421526A (en) | 1976-01-21 |
| JPS49116093A (enrdf_load_stackoverflow) | 1974-11-06 |
| AT329179B (de) | 1976-04-26 |
| JPS5418277B2 (enrdf_load_stackoverflow) | 1979-07-06 |
| BE810969A (fr) | 1974-08-13 |
| ATA105874A (de) | 1975-07-15 |
| FR2216995B1 (enrdf_load_stackoverflow) | 1978-07-28 |
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