ES399347A1 - Substituted beta-lactams and their preparation - Google Patents
Substituted beta-lactams and their preparationInfo
- Publication number
- ES399347A1 ES399347A1 ES399347A ES399347A ES399347A1 ES 399347 A1 ES399347 A1 ES 399347A1 ES 399347 A ES399347 A ES 399347A ES 399347 A ES399347 A ES 399347A ES 399347 A1 ES399347 A1 ES 399347A1
- Authority
- ES
- Spain
- Prior art keywords
- formula
- group
- hydrogen
- halogen
- lactams
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
- C07D205/09—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
- C07D205/09—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4
- C07D205/095—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4 and with a nitrogen atom directly attached in position 3
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Hydrogenated Pyridines (AREA)
- Pyrrole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
A procedure for the preparation of new substituted β-lactams of formula (I) **(See formula)** where X represents hydrogen or halogen or a substituted anino or amino group; Y represents hydrogen or, in cases where X is hydrogen or halogen, Y can be halogen; R3 represents hydrogen or a group of formula (II) **(See formula)** where R4 represents a carboxylic acid group or a salt, ester, thioester or amide derived from a carboxylic acid group and A represents a group of formula (III) **(See formula)** where R1 represents hydrogen or an alkyl, alkenyl, alkynyl or aryl group and R2 represents an acyl group whose process is characterized by reacting a compound of formula (VI) **(See formula)** where X, Y and R3 are as defined above and Z is hydrogen or an alkyl, alkenyl, alkynyl or aryl group, with a lead tetracarboxylate of formula (VIA) Pb (OR2) 4 (VIA) where R2 is acyl. (Machine-translation by Google Translate, not legally binding)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB388371A GB1368074A (en) | 1971-02-04 | 1971-02-04 | Substituted beta-lactams and their preparation |
Publications (1)
Publication Number | Publication Date |
---|---|
ES399347A1 true ES399347A1 (en) | 1975-06-01 |
Family
ID=9766672
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES399347A Expired ES399347A1 (en) | 1971-02-04 | 1972-01-31 | Substituted beta-lactams and their preparation |
ES427900A Expired ES427900A1 (en) | 1971-02-04 | 1974-07-01 | Substituted beta-lactams and their preparation |
ES427901A Expired ES427901A1 (en) | 1971-02-04 | 1974-07-01 | Substituted beta-lactams and their preparation |
Family Applications After (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES427900A Expired ES427900A1 (en) | 1971-02-04 | 1974-07-01 | Substituted beta-lactams and their preparation |
ES427901A Expired ES427901A1 (en) | 1971-02-04 | 1974-07-01 | Substituted beta-lactams and their preparation |
Country Status (8)
Country | Link |
---|---|
AU (1) | AU3837272A (en) |
BE (1) | BE779016A (en) |
DE (1) | DE2205123A1 (en) |
ES (3) | ES399347A1 (en) |
FR (1) | FR2124251A1 (en) |
GB (1) | GB1368074A (en) |
NL (1) | NL7201386A (en) |
ZA (1) | ZA72166B (en) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
LU77306A1 (en) * | 1977-05-09 | 1979-01-18 | ||
EP0000636A1 (en) * | 1977-07-13 | 1979-02-07 | Glaxo Group Limited | Penem compounds, processes for their preparation, their use in pharmaceutical compositions and azetidinones used in their preparation |
EP0003960B1 (en) * | 1978-02-02 | 1983-06-29 | Ciba-Geigy Ag | 6-substituted thia-aza-compounds, their preparation and pharmaceutical compositions containing them |
JPS55133355A (en) * | 1979-04-03 | 1980-10-17 | Shionogi & Co Ltd | Inversion of 3-amino group of beta-lactam ring |
EP0023887B1 (en) * | 1979-08-01 | 1984-11-07 | Ciba-Geigy Ag | 3-substituted bicyclic azetidinone derivatives, process for their preparation, and intermediates as well as their preparation |
EP0232966B1 (en) * | 1986-01-17 | 1997-10-08 | Beecham Group Plc | Process for the preparation of penem compounds and intermediates for this preparation |
-
1971
- 1971-02-04 GB GB388371A patent/GB1368074A/en not_active Expired
-
1972
- 1972-01-11 ZA ZA720166A patent/ZA72166B/en unknown
- 1972-01-21 FR FR7202006A patent/FR2124251A1/fr not_active Withdrawn
- 1972-01-26 AU AU38372/72A patent/AU3837272A/en not_active Expired
- 1972-01-31 ES ES399347A patent/ES399347A1/en not_active Expired
- 1972-02-02 NL NL7201386A patent/NL7201386A/xx unknown
- 1972-02-03 DE DE19722205123 patent/DE2205123A1/en active Pending
- 1972-02-04 BE BE779016A patent/BE779016A/en unknown
-
1974
- 1974-07-01 ES ES427900A patent/ES427900A1/en not_active Expired
- 1974-07-01 ES ES427901A patent/ES427901A1/en not_active Expired
Also Published As
Publication number | Publication date |
---|---|
GB1368074A (en) | 1974-09-25 |
AU3837272A (en) | 1973-08-02 |
DE2205123A1 (en) | 1972-08-10 |
ES427901A1 (en) | 1976-12-16 |
ZA72166B (en) | 1972-09-27 |
NL7201386A (en) | 1972-08-08 |
BE779016A (en) | 1972-08-04 |
ES427900A1 (en) | 1976-12-16 |
FR2124251A1 (en) | 1972-09-22 |
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