ES349316A1 - Procedimiento para la preparacion de 4,5,6,7-tetrahidro - tiazolo (5,4-c) piridinas. - Google Patents

Procedimiento para la preparacion de 4,5,6,7-tetrahidro - tiazolo (5,4-c) piridinas.

Info

Publication number
ES349316A1
ES349316A1 ES349316A ES349316A ES349316A1 ES 349316 A1 ES349316 A1 ES 349316A1 ES 349316 A ES349316 A ES 349316A ES 349316 A ES349316 A ES 349316A ES 349316 A1 ES349316 A1 ES 349316A1
Authority
ES
Spain
Prior art keywords
alkenyl
aryl
alkyl
cycloalkyl
aralkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES349316A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Pharma GmbH and Co KG
Original Assignee
Dr Karl Thomae GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dr Karl Thomae GmbH filed Critical Dr Karl Thomae GmbH
Publication of ES349316A1 publication Critical patent/ES349316A1/es
Expired legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/485—Morphinan derivatives, e.g. morphine, codeine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/02—Preparation by ring-closure or hydrogenation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D211/74—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/80—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D211/84—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
    • C07D211/86—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/80—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D211/84—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
    • C07D211/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/44—Acylated amino or imino radicals
    • C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • E—FIXED CONSTRUCTIONS
    • E02—HYDRAULIC ENGINEERING; FOUNDATIONS; SOIL SHIFTING
    • E02F—DREDGING; SOIL-SHIFTING
    • E02F9/00—Component parts of dredgers or soil-shifting machines, not restricted to one of the kinds covered by groups E02F3/00 - E02F7/00
    • E02F9/20—Drives; Control devices

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Mining & Mineral Resources (AREA)
  • Civil Engineering (AREA)
  • Structural Engineering (AREA)
  • General Engineering & Computer Science (AREA)
  • Emergency Medicine (AREA)
  • Molecular Biology (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
ES349316A 1965-07-23 1968-01-15 Procedimiento para la preparacion de 4,5,6,7-tetrahidro - tiazolo (5,4-c) piridinas. Expired ES349316A1 (es)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
DET0029055 1965-07-23
DET0032992 1967-01-16
DET0032993 1967-01-16
DET0032990 1967-01-16
DET0032991 1967-01-16
DET0032994 1967-01-16

Publications (1)

Publication Number Publication Date
ES349316A1 true ES349316A1 (es) 1969-04-01

Family

ID=27512321

Family Applications (9)

Application Number Title Priority Date Filing Date
ES329299A Expired ES329299A1 (es) 1965-07-23 1966-07-20 Procedimiento para la obtencion de nuevas 4,5,6,7-tetrahi- dro - tiazolo, 5,4-c piridinas.
ES349321A Expired ES349321A1 (es) 1965-07-23 1968-01-15 Procedimiento para la preparacion de 4,5,6,7-tetrahidro - tiazolo (5,4-c) piridinas.
ES349317A Expired ES349317A1 (es) 1965-07-23 1968-01-15 Procedimiento para la preparacion de 4,5,6,7-tetrahidro - tiazolo (5,4-c) piridinas.
ES349314A Expired ES349314A1 (es) 1965-07-23 1968-01-15 Procedimiento para la preparacion de 4,5,6,7-tetrahidro - tiazolo (5,4-c) piridinas.
ES349319A Expired ES349319A1 (es) 1965-07-23 1968-01-15 Procedimiento para la preparacion de 4,5,6,7-tetrahidro - tiazolo (5,4-c) piridinas.
ES349322A Expired ES349322A1 (es) 1965-07-23 1968-01-15 Procedimiento para la preparacion de 4,5,6,7-tetrahidro - tiazolo (5,4-c) piridinas.
ES349316A Expired ES349316A1 (es) 1965-07-23 1968-01-15 Procedimiento para la preparacion de 4,5,6,7-tetrahidro - tiazolo (5,4-c) piridinas.
ES349318A Expired ES349318A1 (es) 1965-07-23 1968-01-15 Procedimiento para la preparacion de 4,5,6,7-tetrahidro - tiazolo (5,4-c) piridinas.
ES349320A Expired ES349320A1 (es) 1965-07-23 1968-01-15 Procedimiento para la preparacion de 4,5,6,7-tetrahidro - tiazolo (5,4-c) piridinas.

Family Applications Before (6)

Application Number Title Priority Date Filing Date
ES329299A Expired ES329299A1 (es) 1965-07-23 1966-07-20 Procedimiento para la obtencion de nuevas 4,5,6,7-tetrahi- dro - tiazolo, 5,4-c piridinas.
ES349321A Expired ES349321A1 (es) 1965-07-23 1968-01-15 Procedimiento para la preparacion de 4,5,6,7-tetrahidro - tiazolo (5,4-c) piridinas.
ES349317A Expired ES349317A1 (es) 1965-07-23 1968-01-15 Procedimiento para la preparacion de 4,5,6,7-tetrahidro - tiazolo (5,4-c) piridinas.
ES349314A Expired ES349314A1 (es) 1965-07-23 1968-01-15 Procedimiento para la preparacion de 4,5,6,7-tetrahidro - tiazolo (5,4-c) piridinas.
ES349319A Expired ES349319A1 (es) 1965-07-23 1968-01-15 Procedimiento para la preparacion de 4,5,6,7-tetrahidro - tiazolo (5,4-c) piridinas.
ES349322A Expired ES349322A1 (es) 1965-07-23 1968-01-15 Procedimiento para la preparacion de 4,5,6,7-tetrahidro - tiazolo (5,4-c) piridinas.

Family Applications After (2)

Application Number Title Priority Date Filing Date
ES349318A Expired ES349318A1 (es) 1965-07-23 1968-01-15 Procedimiento para la preparacion de 4,5,6,7-tetrahidro - tiazolo (5,4-c) piridinas.
ES349320A Expired ES349320A1 (es) 1965-07-23 1968-01-15 Procedimiento para la preparacion de 4,5,6,7-tetrahidro - tiazolo (5,4-c) piridinas.

Country Status (7)

Country Link
BE (1) BE684415A (es)
BR (1) BR6681517D0 (es)
DE (1) DE1620508A1 (es)
ES (9) ES329299A1 (es)
FR (3) FR6013M (es)
GB (1) GB1140387A (es)
NL (2) NL6610324A (es)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4847264A (en) * 1982-07-21 1989-07-11 Rorer Pharmaceutical Corporation Bicyclic nitrogen heterocyclic ethers and thioethers, and their pharmaceutical uses
GB8333514D0 (en) * 1983-12-16 1984-01-25 Erba Farmitalia Tetrahydrothiazolo(5 4-c)pyridine derivatives
EP0192098B1 (de) 1985-02-06 1991-08-21 Boehringer Ingelheim Kg Verwendung des 2-Amino-6-allyl-5,6,7,8-tetrahydro-4H-thiazolo[4,5-d]azepins zur Herstellung eines zur Behandlung der Parkinsonschen Erkrankung bzw. des Parkinsonismus geeigneten Arzneimittels
GB2173187B (en) * 1985-03-23 1988-05-18 Erba Farmitalia Condensed 2-substituted thiazole derivatives
US5060904A (en) * 1987-05-01 1991-10-29 David Hegarty Multi-positionable support stand with movable center of gravity and article holding means
ATE249219T1 (de) * 1997-12-11 2003-09-15 Iaf Biochem Int Antivirale verbindungen
SE0001899D0 (sv) * 2000-05-22 2000-05-22 Pharmacia & Upjohn Ab New compounds
EA200400707A1 (ru) 2001-11-22 2004-10-28 Биовитрум Аб Ингибиторы 11-бета-гидроксистероиддегидрогеназы типа 1
AR041952A1 (es) 2002-11-14 2005-06-01 Novartis Ag N-sulfonilaminotiazol
CL2004000553A1 (es) 2003-03-20 2005-02-04 Actelion Pharmaceuticals Ltd Uso de compuestos derivados de guanidina como antagonistas del receptor de neuropeptido ff; compuestos derivados de guanidina; procedimientos de preparacion; y composicion farmaceutica que los comprende.
JP4759388B2 (ja) 2003-11-12 2011-08-31 第一三共株式会社 チアゾール誘導体の製造法
CA2630718A1 (en) 2005-11-22 2007-05-31 Amgen Inc. Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
WO2010071822A1 (en) * 2008-12-19 2010-06-24 Schering Corporation Piperidine and piperazine derivatives and methods of use thereof
US20120029190A1 (en) * 2009-04-03 2012-02-02 Douglas Burdi Compounds for treating disorders mediated by metabotropic glutamate receptor 5, and methods of use thereof
US11071721B2 (en) 2016-12-02 2021-07-27 Genentech, Inc. Bicyclic amide compounds and methods of use thereof
DK3652178T3 (da) 2017-07-14 2024-03-25 Hoffmann La Roche Bicykliske ketonforbindelser og fremgangsmåder til anvendelse deraf
RU2020115915A (ru) * 2017-10-31 2021-12-01 Ф. Хоффманн-Ля Рош Аг Бициклические сульфоны и сульфоксиды и способы их применения
CN109134510A (zh) * 2018-11-13 2019-01-04 井冈山大学 制备2-氨基-5-cbz-4,5,6,7-四氢噻唑并[5，4-c]吡啶的新方法

Also Published As

Publication number Publication date
ES349322A1 (es) 1969-04-01
ES349317A1 (es) 1969-04-01
ES329299A1 (es) 1968-02-16
FR6013M (es) 1968-05-06
ES349320A1 (es) 1969-04-01
FR1498465A (fr) 1967-10-20
BR6681517D0 (pt) 1973-12-27
ES349318A1 (es) 1969-04-01
ES349321A1 (es) 1969-04-01
BE684415A (es) 1967-01-20
ES349314A1 (es) 1969-04-01
FR94123E (fr) 1969-07-04
DE1620508A1 (de) 1969-09-18
ES349319A1 (es) 1969-04-01
GB1140387A (en) 1969-01-15
NL6610324A (es) 1967-01-24
NL6800589A (es) 1968-07-17

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