ES2656938T3 - Composición que fluye inyectable que comprende buprenorfina - Google Patents
Composición que fluye inyectable que comprende buprenorfina Download PDFInfo
- Publication number
- ES2656938T3 ES2656938T3 ES11728037.0T ES11728037T ES2656938T3 ES 2656938 T3 ES2656938 T3 ES 2656938T3 ES 11728037 T ES11728037 T ES 11728037T ES 2656938 T3 ES2656938 T3 ES 2656938T3
- Authority
- ES
- Spain
- Prior art keywords
- buprenorphine
- polymer
- composition
- implant
- release
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- 239000007943 implant Substances 0.000 abstract description 52
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Landscapes
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- Psychiatry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Materials For Medical Uses (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
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| GB1009549.5A GB2481018B (en) | 2010-06-08 | 2010-06-08 | Injectable flowable composition comprising buprenorphine |
| GB201009549 | 2010-06-08 | ||
| PCT/GB2011/051057 WO2011154724A2 (en) | 2010-06-08 | 2011-06-06 | Compositions |
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| ES2656938T3 true ES2656938T3 (es) | 2018-03-01 |
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| ES11728037.0T Active ES2656938T3 (es) | 2010-06-08 | 2011-06-06 | Composición que fluye inyectable que comprende buprenorfina |
| ES17205986T Active ES2939612T3 (es) | 2010-06-08 | 2011-06-06 | Composición fluyente inyectable que comprende buprenorfina |
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| ES17205986T Active ES2939612T3 (es) | 2010-06-08 | 2011-06-06 | Composición fluyente inyectable que comprende buprenorfina |
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| US8470359B2 (en) * | 2000-11-13 | 2013-06-25 | Qlt Usa, Inc. | Sustained release polymer |
| GB2481018B (en) | 2010-06-08 | 2015-03-18 | Rb Pharmaceuticals Ltd | Injectable flowable composition comprising buprenorphine |
| GB2481017B (en) | 2010-06-08 | 2015-01-07 | Rb Pharmaceuticals Ltd | Microparticle buprenorphine suspension |
| US9272044B2 (en) | 2010-06-08 | 2016-03-01 | Indivior Uk Limited | Injectable flowable composition buprenorphine |
| WO2013126552A1 (en) | 2012-02-21 | 2013-08-29 | Auburn University | Buprenorphine nanoparticle composition and methods thereof |
| NZ631539A (en) | 2012-04-17 | 2016-10-28 | Purdue Pharma Lp | Systems and methods for treating an opioid-induced adverse pharmacodynamic response |
| MX387722B (es) | 2012-07-26 | 2025-03-18 | Camurus Ab | Formulaciones de opioides. |
| SI2877155T1 (sl) | 2012-07-26 | 2021-04-30 | Camurus Ab | Opioidne formulacije |
| EP2931253A1 (en) * | 2012-12-13 | 2015-10-21 | Heron Therapeutics, Inc. | Pharmaceutical composition comprising antiemetic compounds and polyorthoester |
| US9393211B2 (en) * | 2013-03-15 | 2016-07-19 | Oakwood Laboratories LLC | High drug load buprenorphine microspheres and method of producing same |
| KR102505642B1 (ko) * | 2013-03-15 | 2023-03-06 | 헤론 테라퓨틱스 인코포레이티드 | 폴리오르토에스테르 및 비프로톤성 용매의 조성물 |
| US9636308B2 (en) | 2013-03-15 | 2017-05-02 | Oakwood Laboratories LLC | High drug load buprenorphine microspheres and method of producing same |
| GB201404139D0 (en) | 2014-03-10 | 2014-04-23 | Rb Pharmaceuticals Ltd | Sustained release buprenorphine solution formulations |
| EP3509601A1 (en) | 2014-04-21 | 2019-07-17 | Heron Therapeutics, Inc. | A pharmaceutical composition comprising a delivery system, an amide-type local anesthetic, and meloxicam |
| EP3785700A1 (en) * | 2014-04-21 | 2021-03-03 | Heron Therapeutics, Inc. | Compositions of a polyorthoester and an organic acid excipient |
| KR20220138419A (ko) | 2014-04-21 | 2022-10-12 | 헤론 테라퓨틱스 인코포레이티드 | 장기간 작용하는 중합체 전달 시스템 |
| US9801945B2 (en) | 2014-04-21 | 2017-10-31 | Heron Therapeutics, Inc. | Long-acting polymeric delivery systems |
| JP6568102B2 (ja) | 2014-04-28 | 2019-08-28 | オーフォームド，インコーポレイティド | ブプレノルフィン二量体及び消化管疾患の治療におけるその使用 |
| GB201419091D0 (en) | 2014-10-27 | 2014-12-10 | Camurus Ab | Formulations |
| ES2808150T3 (es) * | 2014-11-07 | 2021-02-25 | Indivior Uk Ltd | Regímenes de dosificación de buprenorfina |
| KR102696721B1 (ko) * | 2015-08-03 | 2024-08-19 | 톨마 인터내셔날 리미티드 | 약물의 장기간 지속적인 투여를 위한 액체 폴리머 전달 시스템 |
| AU2016355236C1 (en) | 2015-11-16 | 2022-09-22 | Medincell | A method for morselizing and/or targeting pharmaceutically active principles to synovial tissue |
| FI3512518T3 (fi) * | 2016-09-13 | 2023-01-31 | Hitaasti vapautuvia buprenorfiiniformulaatioita | |
| US10646484B2 (en) | 2017-06-16 | 2020-05-12 | Indivior Uk Limited | Methods to treat opioid use disorder |
| AU2018283724B2 (en) | 2017-06-16 | 2021-08-19 | Indivior Uk Limited | Methods to treat opioid use disorder |
| CN112236142A (zh) | 2018-01-22 | 2021-01-15 | 逸达生物科技股份有限公司 | 用于缓释递送丁丙诺啡的药物组合物 |
| NZ766474A (en) * | 2018-05-11 | 2023-03-31 | Alar Pharmaceuticals Inc | Long-acting injectable formulations and crystalline forms of buprenorphine derivatives |
| AU2019357036B2 (en) | 2018-10-11 | 2024-11-14 | Indivior Uk Limited | Buprenorphine to treat respiratory depression |
| US12403291B2 (en) | 2019-08-30 | 2025-09-02 | Intersect Ent, Inc. | Submucosal bioresorbable drug eluting platform |
| CN118831057A (zh) * | 2023-04-25 | 2024-10-25 | 深圳善康医药科技股份有限公司 | 丁丙诺啡植入剂及其制备方法 |
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| US5702716A (en) | 1988-10-03 | 1997-12-30 | Atrix Laboratories, Inc. | Polymeric compositions useful as controlled release implants |
| US4938763B1 (en) | 1988-10-03 | 1995-07-04 | Atrix Lab Inc | Biodegradable in-situ forming implants and method of producing the same |
| US5324519A (en) | 1989-07-24 | 1994-06-28 | Atrix Laboratories, Inc. | Biodegradable polymer composition |
| CA2582666C (en) | 1994-04-08 | 2010-05-25 | Qlt Usa, Inc. | Controlled release implant |
| US20030211157A1 (en) * | 1996-05-06 | 2003-11-13 | Simon David Lew | Semi-sol delivery blend for water soluble molecules |
| US6143314A (en) * | 1998-10-28 | 2000-11-07 | Atrix Laboratories, Inc. | Controlled release liquid delivery compositions with low initial drug burst |
| US6565874B1 (en) | 1998-10-28 | 2003-05-20 | Atrix Laboratories | Polymeric delivery formulations of leuprolide with improved efficacy |
| US6461631B1 (en) | 1999-11-16 | 2002-10-08 | Atrix Laboratories, Inc. | Biodegradable polymer composition |
| NZ536965A (en) * | 2002-05-31 | 2007-02-23 | Titan Pharmaceuticals Inc | Nonerodible polymeric matrix with buprenorphine encapsulated for the treatment of opiate addiction and pain |
| PL377333A1 (pl) * | 2002-11-06 | 2006-01-23 | Alza Corporation | Preparaty depot o kontrolowanym uwalnianiu |
| EP1622540A4 (en) * | 2003-03-11 | 2009-12-30 | Qlt Usa Inc | PREPARATIONS OF ANTI-CANCER AGENTS DEPENDENT ON THE CELLULAR PROGRAM |
| MX2007003789A (es) * | 2004-10-04 | 2007-07-20 | Qlt Usa Inc | Suministro ocular de formulaciones polimericas para suministro. |
| RS53890B1 (sr) * | 2004-11-10 | 2015-08-31 | Tolmar Therapeutics, Inc. | Stabilizovan polimerni sistem za isporuku |
| ES2550014T3 (es) | 2007-02-15 | 2015-11-03 | Tolmar Therapeutics, Inc. | Poli-(lactida/glicolida) de descarga lenta y métodos para producir polímeros |
| US20090181068A1 (en) * | 2008-01-14 | 2009-07-16 | Dunn Richard L | Low Viscosity Liquid Polymeric Delivery System |
| GB2481018B (en) | 2010-06-08 | 2015-03-18 | Rb Pharmaceuticals Ltd | Injectable flowable composition comprising buprenorphine |
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- 2011-06-06 SM SM20180038T patent/SMT201800038T1/it unknown
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