ES2517925T3 - Utilización de activadores de canales potásicos K2P como analgésicos - Google Patents
Utilización de activadores de canales potásicos K2P como analgésicos Download PDFInfo
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- ES2517925T3 ES2517925T3 ES10771161.6T ES10771161T ES2517925T3 ES 2517925 T3 ES2517925 T3 ES 2517925T3 ES 10771161 T ES10771161 T ES 10771161T ES 2517925 T3 ES2517925 T3 ES 2517925T3
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- FCTRVTQZOUKUIV-MCDZGGTQSA-M potassium;[[[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate Chemical compound [K+].C1=NC=2C(N)=NC=NC=2N1[C@@H]1O[C@H](COP(O)(=O)OP(O)(=O)OP(O)([O-])=O)[C@@H](O)[C@H]1O FCTRVTQZOUKUIV-MCDZGGTQSA-M 0.000 description 1
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Classifications
-
- G—PHYSICS
- G01—MEASURING; TESTING
- G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
- G01N33/00—Investigating or analysing materials by specific methods not covered by groups G01N1/00 - G01N31/00
- G01N33/48—Biological material, e.g. blood, urine; Haemocytometers
- G01N33/50—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
- G01N33/68—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving proteins, peptides or amino acids
- G01N33/6872—Intracellular protein regulatory factors and their receptors, e.g. including ion channels
Landscapes
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- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
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- Chemical & Material Sciences (AREA)
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- Hematology (AREA)
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- Proteomics, Peptides & Aminoacids (AREA)
- Medicinal Chemistry (AREA)
- Physics & Mathematics (AREA)
- Analytical Chemistry (AREA)
- Microbiology (AREA)
- General Health & Medical Sciences (AREA)
- General Physics & Mathematics (AREA)
- Pathology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Investigating Or Analysing Biological Materials (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0956477 | 2009-09-21 | ||
| FR0956477A FR2950362B1 (fr) | 2009-09-21 | 2009-09-21 | Utilisation d'activateurs de canaux potassiques k2p en tant qu'antalgiques. |
| PCT/FR2010/051968 WO2011033241A1 (fr) | 2009-09-21 | 2010-09-21 | Utilisation d'activateurs de canaux potassiques k2p en tant qu'antalgiques |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2517925T3 true ES2517925T3 (es) | 2014-11-04 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES10771161.6T Active ES2517925T3 (es) | 2009-09-21 | 2010-09-21 | Utilización de activadores de canales potásicos K2P como analgésicos |
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| Country | Link |
|---|---|
| US (1) | US9448242B2 (enExample) |
| EP (1) | EP2480893B1 (enExample) |
| CN (1) | CN102597780B (enExample) |
| CA (1) | CA2774861C (enExample) |
| DK (1) | DK2480893T3 (enExample) |
| ES (1) | ES2517925T3 (enExample) |
| FR (1) | FR2950362B1 (enExample) |
| IN (1) | IN2012DN02433A (enExample) |
| WO (1) | WO2011033241A1 (enExample) |
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| US10214476B2 (en) | 2011-12-30 | 2019-02-26 | Ecole Nationale Superieure De Chimie De Clermont Ferrand | Pain relief compounds |
| WO2024126778A1 (en) * | 2022-12-16 | 2024-06-20 | Centre National De La Recherche Scientifique | Process for reversibly inhibiting two-pore potassium channels and inducing nociception, with light spatiotemporal resolution |
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| GB1192126A (en) * | 1967-10-05 | 1970-05-20 | Centre Nat Rech Scient | Indole Derivatives and their production |
| FR2623498B1 (fr) * | 1987-11-24 | 1990-04-06 | Bioprojet Soc Civ | Nouveaux composes enantiomeres derives d'amino-acides, leur procede de preparation et leurs applications therapeutiques |
| US20030165806A1 (en) * | 1997-03-11 | 2003-09-04 | Mark H. Pausch | Potassium channels, nucleotide sequences encoding them, and methods of using same |
| US5919473A (en) * | 1997-05-12 | 1999-07-06 | Elkhoury; George F. | Methods and devices for delivering opioid analgesics to wounds via a subdermal implant |
| US7112403B1 (en) * | 1998-09-01 | 2006-09-26 | Centre National De La Recherche Scientifique | Method for the identification of anesthetics |
| US7955616B2 (en) * | 2003-09-23 | 2011-06-07 | Orthocon, Inc. | Absorbable implants and methods for their use in hemostasis and in the treatment of osseous defects |
| GB0329310D0 (en) * | 2003-12-18 | 2004-01-21 | Univ Keele | Method |
| EP2077126A1 (en) * | 2008-01-07 | 2009-07-08 | Graftys | Analgesic apatitic calcium-phosphate cement |
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2009
- 2009-09-21 FR FR0956477A patent/FR2950362B1/fr not_active Expired - Fee Related
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2010
- 2010-09-21 EP EP10771161.6A patent/EP2480893B1/fr active Active
- 2010-09-21 WO PCT/FR2010/051968 patent/WO2011033241A1/fr not_active Ceased
- 2010-09-21 IN IN2433DEN2012 patent/IN2012DN02433A/en unknown
- 2010-09-21 ES ES10771161.6T patent/ES2517925T3/es active Active
- 2010-09-21 DK DK10771161.6T patent/DK2480893T3/da active
- 2010-09-21 US US13/497,353 patent/US9448242B2/en not_active Expired - Fee Related
- 2010-09-21 CA CA2774861A patent/CA2774861C/fr active Active
- 2010-09-21 CN CN201080050386.7A patent/CN102597780B/zh not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| CA2774861A1 (fr) | 2011-03-24 |
| CN102597780A (zh) | 2012-07-18 |
| EP2480893A1 (fr) | 2012-08-01 |
| DK2480893T3 (da) | 2014-09-29 |
| US9448242B2 (en) | 2016-09-20 |
| WO2011033241A1 (fr) | 2011-03-24 |
| EP2480893B1 (fr) | 2014-08-27 |
| IN2012DN02433A (enExample) | 2015-08-21 |
| FR2950362B1 (fr) | 2011-10-21 |
| CA2774861C (fr) | 2017-08-08 |
| US20120260354A1 (en) | 2012-10-11 |
| FR2950362A1 (fr) | 2011-03-25 |
| CN102597780B (zh) | 2014-11-12 |
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