ES2484315T3 - Tratamiento de la pérdida del sentido del tacto con derivados de saxitoxina - Google Patents
Tratamiento de la pérdida del sentido del tacto con derivados de saxitoxina Download PDFInfo
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- ES2484315T3 ES2484315T3 ES11707610.9T ES11707610T ES2484315T3 ES 2484315 T3 ES2484315 T3 ES 2484315T3 ES 11707610 T ES11707610 T ES 11707610T ES 2484315 T3 ES2484315 T3 ES 2484315T3
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- treatment
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Classifications
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
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- General Chemical & Material Sciences (AREA)
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- Dermatology (AREA)
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- Biomedical Technology (AREA)
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- Neurology (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Medicines Containing Plant Substances (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US312903P | 2001-08-16 | ||
| EP10153234 | 2010-02-10 | ||
| EP10153234 | 2010-02-10 | ||
| US31290310P | 2010-03-11 | 2010-03-11 | |
| PCT/EP2011/051992 WO2011098539A1 (en) | 2010-02-10 | 2011-02-10 | Treatment of loss of sense of touch with saxitoxin derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2484315T3 true ES2484315T3 (es) | 2014-08-11 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES11707610.9T Active ES2484315T3 (es) | 2010-02-10 | 2011-02-10 | Tratamiento de la pérdida del sentido del tacto con derivados de saxitoxina |
Country Status (6)
| Country | Link |
|---|---|
| US (2) | US9107925B2 (OSRAM) |
| EP (1) | EP2533785B1 (OSRAM) |
| JP (2) | JP6112867B2 (OSRAM) |
| CN (1) | CN102811722A (OSRAM) |
| ES (1) | ES2484315T3 (OSRAM) |
| WO (1) | WO2011098539A1 (OSRAM) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
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| US10512644B2 (en) | 2007-03-12 | 2019-12-24 | Inheris Pharmaceuticals, Inc. | Oligomer-opioid agonist conjugates |
| US8173666B2 (en) | 2007-03-12 | 2012-05-08 | Nektar Therapeutics | Oligomer-opioid agonist conjugates |
| US9107925B2 (en) * | 2010-02-10 | 2015-08-18 | Phytotox Limited | Sodium channel blocker for treatment of loss of superficial sensitivity |
| EP2638908A1 (en) * | 2012-03-16 | 2013-09-18 | Phytotox SpA | Paralytic Shellfish Poison |
| PL2968225T3 (pl) * | 2013-03-15 | 2019-08-30 | The Children's Medical Center Corporation | Preparaty skojarzone neosaksytoksyny do przedłużonego znieczulenia miejscowego |
| CA2944549A1 (en) * | 2014-04-09 | 2015-10-15 | Siteone Therapeutics, Inc. | 10',11'-modified saxitoxin useful for the treatment of pain |
| CA3000708A1 (en) * | 2015-09-30 | 2017-04-06 | Siteone Therapeutics, Inc. | 11,13-modified saxitoxins for the treatment of pain |
| GB201602576D0 (en) | 2016-02-12 | 2016-03-30 | Bergen Teknologioverforing As | Process |
| JP2020515611A (ja) * | 2017-03-29 | 2020-05-28 | サイトワン セラピューティクス， インコーポレイテッド | 疼痛の処置のための１１，１３−修飾サキシトキシン |
| BR112019020111A2 (pt) * | 2017-03-29 | 2020-05-05 | Siteone Therapeutics Inc | saxitoxinas 11,13-modificadas para o tratamento de dor |
| US12162886B2 (en) | 2018-10-03 | 2024-12-10 | Siteone Therapeutics, Inc. | 11,13-modified saxitoxins for the treatment of pain |
| CA3188924A1 (en) * | 2020-08-14 | 2022-02-17 | Hassan Pajouhesh | Non-hydrated ketone inhibitors of nav1.7 for the treatment of pain |
| WO2022112887A1 (en) * | 2020-11-25 | 2022-06-02 | Algenis | Method of treating acute nociceptive pain in mammals |
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| CN1284536C (zh) * | 2000-09-18 | 2006-11-15 | 威克斯医药有限公司 | 河豚毒素或蛤蚌毒素及其类似物在制备用于全身镇痛的镇痛药中的应用 |
| EP1443932B1 (en) * | 2001-11-15 | 2012-12-26 | Micro Algae Corporation | Pharmaceutical compositions containing 3,4-propinoperhydropurines and uses thereof for blocking neuronal transmission |
| EP1796676B1 (en) * | 2004-05-07 | 2016-03-09 | Phytotox Limited | Transdermal administration of phycotoxins |
| BRPI0510761A (pt) | 2004-05-07 | 2007-11-20 | Phytotox Ltd | métodos de tratar um paciente afligido com pelo menos uma enfermidade e de reduzir ou eliminar rugas |
| KR20070083650A (ko) * | 2004-09-21 | 2007-08-24 | 라보라토리오스 델 드라. 에스테브.에스.에이. | 중추 신경적으로 유발된 신경병증성 통증을 치료하기 위한테트로도톡신 및 그것의 유도체 |
| EP1799220A1 (en) | 2004-09-22 | 2007-06-27 | Laboratorios del Dr. Esteve S.A. | Tetrodotoxin and its derivatives for the treatment of peripheral-nervously derived neuropathic pain |
| ES2691411T3 (es) * | 2006-03-27 | 2018-11-27 | Wex Medical Limited | Uso de bloqueadores de los canales de sodio para el tratamiento del dolor neuropático que se desarrolla como consecuencia de la quimioterapia |
| US9107925B2 (en) * | 2010-02-10 | 2015-08-18 | Phytotox Limited | Sodium channel blocker for treatment of loss of superficial sensitivity |
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2011
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- 2011-02-10 CN CN2011800149701A patent/CN102811722A/zh active Pending
- 2011-02-10 WO PCT/EP2011/051992 patent/WO2011098539A1/en not_active Ceased
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2015
- 2015-07-08 US US14/794,428 patent/US20160000793A1/en not_active Abandoned
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2016
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Also Published As
| Publication number | Publication date |
|---|---|
| CN102811722A (zh) | 2012-12-05 |
| US20160000793A1 (en) | 2016-01-07 |
| JP2013519653A (ja) | 2013-05-30 |
| EP2533785A1 (en) | 2012-12-19 |
| US9107925B2 (en) | 2015-08-18 |
| EP2533785B1 (en) | 2014-04-23 |
| US20130039976A1 (en) | 2013-02-14 |
| JP6112867B2 (ja) | 2017-04-12 |
| WO2011098539A1 (en) | 2011-08-18 |
| JP2017081920A (ja) | 2017-05-18 |
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