ES2372707T3 - Inhibidores de la ikk-beta serina-treonina proteína quinasa. - Google Patents
Inhibidores de la ikk-beta serina-treonina proteína quinasa. Download PDFInfo
- Publication number
- ES2372707T3 ES2372707T3 ES07824358T ES07824358T ES2372707T3 ES 2372707 T3 ES2372707 T3 ES 2372707T3 ES 07824358 T ES07824358 T ES 07824358T ES 07824358 T ES07824358 T ES 07824358T ES 2372707 T3 ES2372707 T3 ES 2372707T3
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- Prior art keywords
- cyclopentyl
- carbamoylamino
- carbamoyl
- alkyl
- phenyl
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Classifications
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- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
- A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
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- Hematology (AREA)
- Reproductive Health (AREA)
- Emergency Medicine (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Enzymes And Modification Thereof (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0621720 | 2006-11-01 | ||
| GB0621720A GB0621720D0 (en) | 2006-11-01 | 2006-11-01 | Inhibitors of ikk- serine-threonine protein kinase |
| GB0715470A GB0715470D0 (en) | 2007-08-09 | 2007-08-09 | IKK- serine-threonine protein kinase inhibitors |
| GB0715470 | 2007-08-09 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2372707T3 true ES2372707T3 (es) | 2012-01-25 |
Family
ID=39015937
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES07824358T Active ES2372707T3 (es) | 2006-11-01 | 2007-10-29 | Inhibidores de la ikk-beta serina-treonina proteína quinasa. |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US8003695B2 (enExample) |
| EP (1) | EP2078007B1 (enExample) |
| JP (1) | JP2010508336A (enExample) |
| KR (1) | KR20090077975A (enExample) |
| AT (1) | ATE522516T1 (enExample) |
| AU (1) | AU2007315943A1 (enExample) |
| BR (1) | BRPI0718056A2 (enExample) |
| CA (1) | CA2668338A1 (enExample) |
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| EA (1) | EA200900616A1 (enExample) |
| ES (1) | ES2372707T3 (enExample) |
| IL (1) | IL198267A0 (enExample) |
| MX (1) | MX2009004442A (enExample) |
| NZ (1) | NZ576705A (enExample) |
| WO (1) | WO2008053182A1 (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0619753D0 (en) | 2006-10-06 | 2006-11-15 | Chroma Therapeutics Ltd | Enzyme inhibitors |
| GB0803747D0 (en) | 2008-02-29 | 2008-04-09 | Martin | Enzyme and receptor modulation |
| MX2010011501A (es) * | 2008-04-23 | 2010-11-30 | Chroma Therapeutics Ltd | Inhibidores de proteina cinasa de serina-treonina ikk-beta. |
| BRPI0911480A2 (pt) * | 2008-04-26 | 2018-04-03 | Chroma Therapeutics Ltd | inibidores de proteínas serina-treonina quinase ikk-beta |
| EP2361245A4 (en) * | 2008-11-26 | 2012-06-13 | Trt Pharma Inc | HYBRID-IONONE AND CURCUMINE MOLECULES AS ANTICREBIALS |
| GB0903480D0 (en) | 2009-02-27 | 2009-04-08 | Chroma Therapeutics Ltd | Enzyme Inhibitors |
| GB0907120D0 (en) * | 2009-04-24 | 2009-06-03 | Chroma Therapeutics Ltd | Inhibitors of IKK-ß serine-threonine protein kinase |
| GB201211310D0 (en) | 2012-06-26 | 2012-08-08 | Chroma Therapeutics Ltd | CSF-1R kinase inhibitors |
| HRP20171320T1 (hr) | 2012-10-17 | 2017-10-20 | Macrophage Pharma Limited | Terc-butil n-[2-{4-[6-amino-5-(2,4-difluorobenzoil)-2-oksopiridin-1(2h)-il]-3,5-difluorofenil}etil]-l-alaninat ili njegova sol, hidrat ili solvat |
| US9809577B2 (en) * | 2013-12-11 | 2017-11-07 | Biogen Ma Inc. | Biaryl inhibitors of Bruton's tyrosine kinase |
| GB201713975D0 (en) | 2017-08-31 | 2017-10-18 | Macrophage Pharma Ltd | Medical use |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE0102616D0 (sv) * | 2001-07-25 | 2001-07-25 | Astrazeneca Ab | Novel compounds |
| SE0300092D0 (sv) | 2003-01-15 | 2003-01-15 | Astrazeneca Ab | Novel compounds |
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2007
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- 2007-10-29 AT AT07824358T patent/ATE522516T1/de not_active IP Right Cessation
- 2007-10-29 AU AU2007315943A patent/AU2007315943A1/en not_active Abandoned
- 2007-10-29 JP JP2009535115A patent/JP2010508336A/ja not_active Withdrawn
- 2007-10-29 EA EA200900616A patent/EA200900616A1/ru unknown
- 2007-10-29 US US12/513,206 patent/US8003695B2/en not_active Expired - Fee Related
- 2007-10-29 CA CA002668338A patent/CA2668338A1/en not_active Abandoned
- 2007-10-29 DK DK07824358.1T patent/DK2078007T3/da active
- 2007-10-29 MX MX2009004442A patent/MX2009004442A/es active IP Right Grant
- 2007-10-29 BR BRPI0718056-0A patent/BRPI0718056A2/pt not_active IP Right Cessation
- 2007-10-29 ES ES07824358T patent/ES2372707T3/es active Active
- 2007-10-29 NZ NZ576705A patent/NZ576705A/en not_active IP Right Cessation
- 2007-10-29 KR KR1020097011261A patent/KR20090077975A/ko not_active Withdrawn
- 2007-10-29 EP EP07824358A patent/EP2078007B1/en not_active Not-in-force
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2009
- 2009-04-21 IL IL198267A patent/IL198267A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NZ576705A (en) | 2011-12-22 |
| EP2078007A1 (en) | 2009-07-15 |
| DK2078007T3 (da) | 2011-12-12 |
| US8003695B2 (en) | 2011-08-23 |
| WO2008053182A1 (en) | 2008-05-08 |
| IL198267A0 (en) | 2009-12-24 |
| EA200900616A1 (ru) | 2010-04-30 |
| BRPI0718056A2 (pt) | 2013-11-05 |
| JP2010508336A (ja) | 2010-03-18 |
| EP2078007B1 (en) | 2011-08-31 |
| MX2009004442A (es) | 2009-05-22 |
| CA2668338A1 (en) | 2008-05-08 |
| KR20090077975A (ko) | 2009-07-16 |
| ATE522516T1 (de) | 2011-09-15 |
| AU2007315943A1 (en) | 2008-05-08 |
| US20100087515A1 (en) | 2010-04-08 |
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